NL7906214A - Acetyleenderivaten van androst-4-een en werkwijze voor de bereiding en toepassing ervan, alsmede farmaceuti- sche preparaten die deze derivaten bevatten. - Google Patents

Acetyleenderivaten van androst-4-een en werkwijze voor de bereiding en toepassing ervan, alsmede farmaceuti- sche preparaten die deze derivaten bevatten. Download PDF

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Publication number
NL7906214A
NL7906214A NL7906214A NL7906214A NL7906214A NL 7906214 A NL7906214 A NL 7906214A NL 7906214 A NL7906214 A NL 7906214A NL 7906214 A NL7906214 A NL 7906214A NL 7906214 A NL7906214 A NL 7906214A
Authority
NL
Netherlands
Prior art keywords
formula
compounds
radical
carbon atoms
hydrogen atom
Prior art date
Application number
NL7906214A
Other languages
English (en)
Dutch (nl)
Original Assignee
Roussel Uclaf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Uclaf filed Critical Roussel Uclaf
Publication of NL7906214A publication Critical patent/NL7906214A/nl

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C07J71/0005—Oxygen-containing hetero ring
    • C07J71/001—Oxiranes
    • C07J71/0015—Oxiranes at position 9(11)
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0003—Androstane derivatives
    • C07J1/0011—Androstane derivatives substituted in position 17 by a keto group
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0003—Androstane derivatives
    • C07J1/0033—Androstane derivatives substituted in position 17 alfa and 17 beta
    • C07J1/004—Androstane derivatives substituted in position 17 alfa and 17 beta the substituent in position 17 alfa being an unsaturated hydrocarbon group
    • C07J1/0048—Alkynyl derivatives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Rheumatology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
NL7906214A 1978-08-16 1979-08-15 Acetyleenderivaten van androst-4-een en werkwijze voor de bereiding en toepassing ervan, alsmede farmaceuti- sche preparaten die deze derivaten bevatten. NL7906214A (nl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR7823851A FR2433536A1 (fr) 1978-08-16 1978-08-16 Nouveaux derives de l'androst 4-ene, leur procede de preparation et leur application comme medicament
FR7823851 1978-08-16

Publications (1)

Publication Number Publication Date
NL7906214A true NL7906214A (nl) 1980-02-19

Family

ID=9211827

Family Applications (1)

Application Number Title Priority Date Filing Date
NL7906214A NL7906214A (nl) 1978-08-16 1979-08-15 Acetyleenderivaten van androst-4-een en werkwijze voor de bereiding en toepassing ervan, alsmede farmaceuti- sche preparaten die deze derivaten bevatten.

Country Status (16)

Country Link
US (1) US4232015A (fr)
JP (1) JPS5528982A (fr)
AT (1) AT368520B (fr)
AU (1) AU524232B2 (fr)
BE (1) BE878256A (fr)
CH (1) CH641814A5 (fr)
DE (1) DE2933258A1 (fr)
FR (1) FR2433536A1 (fr)
GB (1) GB2029833B (fr)
HU (1) HU180520B (fr)
IE (1) IE48931B1 (fr)
IT (1) IT1164040B (fr)
NL (1) NL7906214A (fr)
PT (1) PT70060A (fr)
SE (1) SE435186B (fr)
ZA (1) ZA793967B (fr)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4424218A (en) 1979-08-17 1984-01-03 Roussel Uclaf Novel 3 α-amino steroids
FR2468617A1 (fr) * 1979-10-26 1981-05-08 Roussel Uclaf Nouveaux derives acetyleniques chlores de l'androst-4-ene leur procede de preparation, et leur application a titre de medicament et les compositions pharmaceutiques les renfermant
US4383947A (en) * 1981-07-24 1983-05-17 The Upjohn Company Introduction of a fluorine atom
US4488995A (en) * 1984-02-06 1984-12-18 E. R. Squibb & Sons, Inc. Androstene-17β-alkylthiomethyl ethers
US6740646B2 (en) * 2002-01-16 2004-05-25 Biotest Laboratories, Llc Bioavailable prodrugs of androgenic steroids and related method
JP4636847B2 (ja) * 2004-10-13 2011-02-23 株式会社ロッテ 全粒粉からなる小麦粉の加工方法及びその加工方法により得られた加工小麦粉並びにその加工小麦粉を使用した食品

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2740798A (en) * 1953-05-25 1956-04-03 Searle & Co 11 beta-hydroxy-17-ethynyl testosterone and esters thereof
US3010957A (en) * 1958-11-26 1961-11-28 Schering Corp Ethinyl androstadienes
FR1349113A (fr) * 1959-01-28 1964-01-17 Upjohn Co Procédé de fabrication de 6-fluoro-11 oxygéné-17-bêta-hydroxy-17 alpha-alkynyl inférieur-4-androstène-3-ones et leurs dérivés acylés
GB1081494A (en) * 1965-09-14 1967-08-31 British Drug Houses Ltd 17ª‡-(alka-1',3'-diynyl)-steroids
US3793308A (en) * 1972-11-08 1974-02-19 Upjohn Co 4-spiro(cyclopropyl)androstenes and process for their production
SE7801152L (sv) * 1977-02-22 1978-08-23 Roussel Uclaf Sett att framstella 17alfa-acetylen-derivat av androst-4-en

Also Published As

Publication number Publication date
SE7905865L (sv) 1980-02-17
IT7950049A0 (it) 1979-08-14
AU524232B2 (en) 1982-09-09
DE2933258C2 (fr) 1990-10-25
IT1164040B (it) 1987-04-08
AT368520B (de) 1982-10-25
AU4995879A (en) 1980-03-06
DE2933258A1 (de) 1980-02-28
CH641814A5 (fr) 1984-03-15
GB2029833B (en) 1983-04-27
US4232015A (en) 1980-11-04
FR2433536B1 (fr) 1981-07-24
JPS636559B2 (fr) 1988-02-10
SE435186B (sv) 1984-09-10
PT70060A (fr) 1979-09-01
ATA553479A (de) 1982-02-15
GB2029833A (en) 1980-03-26
FR2433536A1 (fr) 1980-03-14
IE48931B1 (en) 1985-06-26
IE791578L (en) 1980-02-16
JPS5528982A (en) 1980-02-29
ZA793967B (en) 1980-07-30
HU180520B (en) 1983-03-28
BE878256A (fr) 1980-02-14

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Legal Events

Date Code Title Description
A85 Still pending on 85-01-01
BA A request for search or an international-type search has been filed
BB A search report has been drawn up
BC A request for examination has been filed
BV The patent application has lapsed