MY171378A - Solubilized capsule formulation of 1,1-dimethylethyl [(1s)-1-{[(2s,4r)-4-(7-chloro-4methoxyisoquinolin-1-yloxy)-2-({(1r,2s)-1-[(cyclopropylsulfonyl)carbamoyl]-2-ethenylcyclopropyl}carbamoyl)pyrrolidin-1-yl]carbonyl}-2,2-dimethylpropyl]carbamate - Google Patents

Solubilized capsule formulation of 1,1-dimethylethyl [(1s)-1-{[(2s,4r)-4-(7-chloro-4methoxyisoquinolin-1-yloxy)-2-({(1r,2s)-1-[(cyclopropylsulfonyl)carbamoyl]-2-ethenylcyclopropyl}carbamoyl)pyrrolidin-1-yl]carbonyl}-2,2-dimethylpropyl]carbamate

Info

Publication number
MY171378A
MY171378A MYPI2014703294A MYPI2014703294A MY171378A MY 171378 A MY171378 A MY 171378A MY PI2014703294 A MYPI2014703294 A MY PI2014703294A MY PI2014703294 A MYPI2014703294 A MY PI2014703294A MY 171378 A MY171378 A MY 171378A
Authority
MY
Malaysia
Prior art keywords
carbamoyl
ethenylcyclopropyl
cyclopropylsulfonyl
dimethylpropyl
dimethylethyl
Prior art date
Application number
MYPI2014703294A
Other languages
English (en)
Inventor
Robert Kevin Perrone
Original Assignee
Bristol Myers Squibb Holdings Ireland
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=48428670&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MY171378(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bristol Myers Squibb Holdings Ireland filed Critical Bristol Myers Squibb Holdings Ireland
Publication of MY171378A publication Critical patent/MY171378A/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841Filling excipients; Inactive ingredients
    • A61K9/4858Organic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/472Non-condensed isoquinolines, e.g. papaverine
    • A61K31/4725Non-condensed isoquinolines, e.g. papaverine containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/06Tripeptides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Virology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
MYPI2014703294A 2012-05-07 2013-04-30 Solubilized capsule formulation of 1,1-dimethylethyl [(1s)-1-{[(2s,4r)-4-(7-chloro-4methoxyisoquinolin-1-yloxy)-2-({(1r,2s)-1-[(cyclopropylsulfonyl)carbamoyl]-2-ethenylcyclopropyl}carbamoyl)pyrrolidin-1-yl]carbonyl}-2,2-dimethylpropyl]carbamate MY171378A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201261643454P 2012-05-07 2012-05-07

Publications (1)

Publication Number Publication Date
MY171378A true MY171378A (en) 2019-10-10

Family

ID=48428670

Family Applications (1)

Application Number Title Priority Date Filing Date
MYPI2014703294A MY171378A (en) 2012-05-07 2013-04-30 Solubilized capsule formulation of 1,1-dimethylethyl [(1s)-1-{[(2s,4r)-4-(7-chloro-4methoxyisoquinolin-1-yloxy)-2-({(1r,2s)-1-[(cyclopropylsulfonyl)carbamoyl]-2-ethenylcyclopropyl}carbamoyl)pyrrolidin-1-yl]carbonyl}-2,2-dimethylpropyl]carbamate

Country Status (33)

Country Link
US (1) US20130302414A1 (https=)
EP (1) EP2846780B1 (https=)
JP (1) JP6276756B2 (https=)
KR (1) KR20150004921A (https=)
CN (1) CN104363899A (https=)
AR (1) AR090954A1 (https=)
AU (1) AU2013260005B2 (https=)
BR (1) BR112014027676A2 (https=)
CA (1) CA2872765A1 (https=)
CL (1) CL2014003012A1 (https=)
CO (1) CO7141457A2 (https=)
CY (1) CY1120756T1 (https=)
DK (1) DK2846780T3 (https=)
EA (1) EA028749B1 (https=)
ES (1) ES2688817T3 (https=)
HR (1) HRP20181583T1 (https=)
IL (1) IL235466B (https=)
LT (1) LT2846780T (https=)
MX (1) MX358545B (https=)
MY (1) MY171378A (https=)
NZ (1) NZ630248A (https=)
PE (1) PE20142439A1 (https=)
PH (1) PH12014502405A1 (https=)
PL (1) PL2846780T3 (https=)
PT (1) PT2846780T (https=)
RS (1) RS57881B1 (https=)
SG (1) SG11201406964QA (https=)
SI (1) SI2846780T1 (https=)
SM (1) SMT201800506T1 (https=)
TW (1) TWI577392B (https=)
UY (1) UY34785A (https=)
WO (1) WO2013169520A1 (https=)
ZA (1) ZA201408967B (https=)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2846778B1 (en) * 2012-05-07 2018-04-25 Bristol-Myers Squibb Holdings Ireland Oral solid dosage formulation of 1,1-dimethylethyl [(1s)-1-{[(2s,4r)-4-(7-chloro-4methoxyisoquinolin-1-yloxy)-2-({(1r,2s)-1-[(cyclopropylsulfonyl)carbamoyl]-2-ethenylcyclopropyl}carbamoyl)pyrrolidin-1-yl]carbonyl}-2,2-dimethylpropyl]carbamate
EA025560B1 (ru) 2012-10-19 2017-01-30 Бристол-Майерс Сквибб Компани Ингибиторы вируса гепатита с
WO2014070964A1 (en) 2012-11-02 2014-05-08 Bristol-Myers Squibb Company Hepatitis c virus inhibitors
WO2014071007A1 (en) 2012-11-02 2014-05-08 Bristol-Myers Squibb Company Hepatitis c virus inhibitors
US9643999B2 (en) 2012-11-02 2017-05-09 Bristol-Myers Squibb Company Hepatitis C virus inhibitors
EP2914614B1 (en) 2012-11-05 2017-08-16 Bristol-Myers Squibb Company Hepatitis c virus inhibitors
WO2014137869A1 (en) 2013-03-07 2014-09-12 Bristol-Myers Squibb Company Hepatitis c virus inhibitors
WO2019130341A1 (en) * 2017-12-26 2019-07-04 Hetero Labs Limited Capsule compositions comprising lopinavir and ritonavir
JP7433252B2 (ja) 2018-03-14 2024-02-19 キャンディ・セラピューティクス・リミテッド Nk-1/nk-3受容体二重アンタゴニストを含む新規な医薬製剤
US11464764B2 (en) * 2018-12-19 2022-10-11 Corcept Therapeutics Incorporated Pharmaceutical formulations containing relacorilant, a heteroaryl-ketone fused azadecalin compound
US12533358B1 (en) 2025-05-14 2026-01-27 Bayer Consumer Care Ag Methods of treatment with elinzanetant

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA9710071B (en) * 1996-11-21 1998-05-25 Abbott Lab Pharmaceutical composition.
NZ526169A (en) * 2000-10-31 2005-12-23 Boehringer Ingelheim Pharma Oral dosage self-emulsifying formulations of pyranone protease inhibitors
US6828301B2 (en) * 2002-02-07 2004-12-07 Boehringer Ingelheim International Gmbh Pharmaceutical compositions for hepatitis C viral protease inhibitors
MY140680A (en) * 2002-05-20 2010-01-15 Bristol Myers Squibb Co Hepatitis c virus inhibitors
WO2010042834A1 (en) * 2008-10-09 2010-04-15 Anadys Pharmaceuticals, Inc. A method of inhibiting hepatitis c virus by combination of a 5,6-dihydro-1h-pyridin-2-one and one or more additional antiviral compounds
US8252821B2 (en) * 2009-04-14 2012-08-28 Bristol-Myers Squibb Company Bioavailable capsule compositions of amorphous alpha-(N-sulfonamido)acetamide compound

Also Published As

Publication number Publication date
IL235466B (en) 2019-03-31
CY1120756T1 (el) 2019-12-11
SG11201406964QA (en) 2014-11-27
ES2688817T3 (es) 2018-11-07
KR20150004921A (ko) 2015-01-13
TWI577392B (zh) 2017-04-11
PE20142439A1 (es) 2015-01-28
LT2846780T (lt) 2018-11-12
CN104363899A (zh) 2015-02-18
UY34785A (es) 2013-11-29
RS57881B1 (sr) 2019-01-31
JP2015516418A (ja) 2015-06-11
AR090954A1 (es) 2014-12-17
EP2846780B1 (en) 2018-07-18
BR112014027676A2 (pt) 2017-06-27
PL2846780T3 (pl) 2018-11-30
MX358545B (es) 2018-08-24
AU2013260005B2 (en) 2017-07-13
HK1204552A1 (en) 2015-11-27
CA2872765A1 (en) 2013-11-14
PT2846780T (pt) 2018-10-26
DK2846780T3 (en) 2018-09-17
ZA201408967B (en) 2016-10-26
EA201492039A1 (ru) 2015-02-27
WO2013169520A1 (en) 2013-11-14
EA028749B1 (ru) 2017-12-29
NZ630248A (en) 2016-11-25
CO7141457A2 (es) 2014-12-12
SMT201800506T1 (it) 2018-11-09
TW201350145A (zh) 2013-12-16
SI2846780T1 (sl) 2018-09-28
JP6276756B2 (ja) 2018-02-07
CL2014003012A1 (es) 2015-07-10
AU2013260005A1 (en) 2015-01-15
EP2846780A1 (en) 2015-03-18
PH12014502405A1 (en) 2015-01-12
HRP20181583T1 (hr) 2018-11-30
MX2014013220A (es) 2015-05-11
US20130302414A1 (en) 2013-11-14

Similar Documents

Publication Publication Date Title
MY171378A (en) Solubilized capsule formulation of 1,1-dimethylethyl [(1s)-1-{[(2s,4r)-4-(7-chloro-4methoxyisoquinolin-1-yloxy)-2-({(1r,2s)-1-[(cyclopropylsulfonyl)carbamoyl]-2-ethenylcyclopropyl}carbamoyl)pyrrolidin-1-yl]carbonyl}-2,2-dimethylpropyl]carbamate
WO2014052360A3 (en) Glycoprotein preparations
AU2013225533A8 (en) Amido spirocyclic amide and sulfonamide derivatives
CA2902938C (en) Peptides for skin rejuvenation and methods of using the same
HK1206055A1 (en) Methods and processes for non-invasive assessment of genetic variations
MX2013012542A (es) Compuestos de amida y aplicacion farmaceutica para el mismo.
WO2015081085A3 (en) Methods of treating a tauopathy
UA95283C2 (ru) Активное косметическое начало, состоящее из экстракта микроводорослей класса chlorophyceae и феррулата аргинина, и его применение
HUE045111T2 (hu) N-(2-metoxibenzil)-4-[(metilaminokarbonil)amino]benzolszulfonamid inszekticidekkel vagy fungicidekkel képzett kombinációjának alkalmazása növénytermesztés hatásfokának növelésére
PH12015501115B1 (en) Learning and memory improver
MY169048A (en) Polymorph of n- (2-methoxybenzoyl) -4- [(methylaminocarbonyl) amino] benzenesulfonamide
WO2015048503A3 (en) N-arylmethyl sulfonamide negative modulators of nr2a
WO2012099899A3 (en) Topical dermatological compositions for the treatment of acne
WO2015095240A3 (en) Biosynthesis of 1-undecence and related terminal olefins
WO2011054804A3 (en) Skin care compositions comprising phenoxyalkyl amines
IL235657A0 (en) Pharmacy device containing (1r, 4r) - 6' - fluoro - n, n - dimethyl - 4 - phenyl - 4', 9' - dihydro - 3'h - spiro [cyclohexane - 1, 1' - pyrano [3, 4 ,b] indole] – 4 – amine and antidepressants
MX352596B (es) Composicion farmaceutica que comprende (1r,4r)-6´-fluoro-n,n-dimet il-4-fenil-4´,9´-dihidro-3´h-espiro[ciclohexan-1,1´-piran-[3,4,b] indol]-4-amina y paracetamol o propacetamol.
CA2852067C (en) Sugar chain-containing polymer, and sugar chain-containing polymer complex
WO2013072770A3 (en) Pharmaceutical formulations comprising atorvastatin and glimepiride
TH1401006625A (th) สูตรผสมแคปซูลที่ละลายได้ของ 1,1-ไดเมธิลเอธิล[(1s)-1{[2s,4r)-4-(7-คลอโร-4เมธอกซีไอโซควิโนลิน-1-อิลออกซี)-2-({1r,2s)-1-[(ไซโคลโพรพิลซัลโฟนิล) คาร์บาโมอิล]-2-เอธีนิลไซโคลโพรพิล}คาร์บาโมอิล)ไพร์โรลิดิน-1-อิล]คาร์บอนิล}-2,2-ไดเมธิลโพรพิล]คาร์บาเมต
WO2014099109A3 (en) Plod-2 modulators and their use in the treatment of skin
WO2012160713A8 (en) Learning and memory improver
CN105709225A (zh) 一种用于治疗高眼压的药物
TH156288A (th) สูตรผสมแคปซูลที่ละลายได้ของ 1,1-ไดเมธิลเอธิล[(1s)-1{[2s,4r)-4-(7-คลอโร-4เมธอกซีไอโซควิโนลิน-1-อิลออกซี)-2-({1r,2s)-1-[(ไซโคลโพรพิลซัลโฟนิล) คาร์บาโมอิล]-2-เอธีนิลไซโคลโพรพิล}คาร์บาโมอิล)ไพร์โรลิดิน-1-อิล]คาร์บอนิล}-2,2-ไดเมธิลโพรพิล]คาร์บาเมต
BR112014028557A2 (pt) composição farmacêutica compreendendo ( 1r , 4r )-6-fluoro-n ,n-dimetil-4-fenil-4 ,9-di-hidro-3h-espiro[ciclohexano-1 ,1-pirano-[3,4,b]indol]-4- amina e um anticonvulsivo