RS57881B1 - Formulacija solubilizovane kapsule 1,1-dimetiletil [(1s)-1-{[(2s,4r)-4-(7-hloro-4metoksiizohinolin-1-iloksi)-2-({(1r,2s)-1-[(ciklopropilsulfonil)karbamoil]-2-etenilciklopropil}karbamoil)pirolidin-1-il]karbonil}-2,2-dimetilpropil]karbamata - Google Patents

Formulacija solubilizovane kapsule 1,1-dimetiletil [(1s)-1-{[(2s,4r)-4-(7-hloro-4metoksiizohinolin-1-iloksi)-2-({(1r,2s)-1-[(ciklopropilsulfonil)karbamoil]-2-etenilciklopropil}karbamoil)pirolidin-1-il]karbonil}-2,2-dimetilpropil]karbamata

Info

Publication number
RS57881B1
RS57881B1 RS20181141A RSP20181141A RS57881B1 RS 57881 B1 RS57881 B1 RS 57881B1 RS 20181141 A RS20181141 A RS 20181141A RS P20181141 A RSP20181141 A RS P20181141A RS 57881 B1 RS57881 B1 RS 57881B1
Authority
RS
Serbia
Prior art keywords
carbamoyl
ethenylcyclopropyl
cyclopropylsulfonyl
dimethylpropyl
dimethylethyl
Prior art date
Application number
RS20181141A
Other languages
English (en)
Inventor
Robert Kevin Perrone
Original Assignee
Bristol Myers Squibb Holdings Ireland
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=48428670&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=RS57881(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bristol Myers Squibb Holdings Ireland filed Critical Bristol Myers Squibb Holdings Ireland
Publication of RS57881B1 publication Critical patent/RS57881B1/sr

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841—Filling excipients; Inactive ingredients
    • A61K9/4858—Organic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/472—Non-condensed isoquinolines, e.g. papaverine
    • A61K31/4725—Non-condensed isoquinolines, e.g. papaverine containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/06—Tripeptides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Oncology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • General Chemical & Material Sciences (AREA)
  • Virology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
RS20181141A 2012-05-07 2013-04-30 Formulacija solubilizovane kapsule 1,1-dimetiletil [(1s)-1-{[(2s,4r)-4-(7-hloro-4metoksiizohinolin-1-iloksi)-2-({(1r,2s)-1-[(ciklopropilsulfonil)karbamoil]-2-etenilciklopropil}karbamoil)pirolidin-1-il]karbonil}-2,2-dimetilpropil]karbamata RS57881B1 (sr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201261643454P 2012-05-07 2012-05-07
PCT/US2013/038770 WO2013169520A1 (en) 2012-05-07 2013-04-30 Solubilized capsule formulation of 1,1-dimethylethyl [(1s)-1-{[(2s,4r)-4-(7-chloro-4methoxyisoquinolin-1-yloxy)-2-({(1r,2s)-1-[(cyclopropylsulfonyl)carbamoyl]-2-ethenylcyclopropyl}carbamoyl)pyrrolidin-1-yl]carbonyl}-2,2-dimethylpropyl]carbamate
EP13722217.0A EP2846780B1 (en) 2012-05-07 2013-04-30 Solubilized capsule formulation of 1,1-dimethylethyl [(1s)-1-{[(2s,4r)-4-(7-chloro-4methoxyisoquinolin-1-yloxy)-2-({(1r,2s)-1-[(cyclopropylsulfonyl)carbamoyl]-2-ethenylcyclopropyl}carbamoyl)pyrrolidin-1-yl]carbonyl}-2,2-dimethylpropyl]carbamate

Publications (1)

Publication Number Publication Date
RS57881B1 true RS57881B1 (sr) 2019-01-31

Family

ID=48428670

Family Applications (1)

Application Number Title Priority Date Filing Date
RS20181141A RS57881B1 (sr) 2012-05-07 2013-04-30 Formulacija solubilizovane kapsule 1,1-dimetiletil [(1s)-1-{[(2s,4r)-4-(7-hloro-4metoksiizohinolin-1-iloksi)-2-({(1r,2s)-1-[(ciklopropilsulfonil)karbamoil]-2-etenilciklopropil}karbamoil)pirolidin-1-il]karbonil}-2,2-dimetilpropil]karbamata

Country Status (33)

Country Link
US (1) US20130302414A1 (sr)
EP (1) EP2846780B1 (sr)
JP (1) JP6276756B2 (sr)
KR (1) KR20150004921A (sr)
CN (1) CN104363899A (sr)
AR (1) AR090954A1 (sr)
AU (1) AU2013260005B2 (sr)
BR (1) BR112014027676A2 (sr)
CA (1) CA2872765A1 (sr)
CL (1) CL2014003012A1 (sr)
CO (1) CO7141457A2 (sr)
CY (1) CY1120756T1 (sr)
DK (1) DK2846780T3 (sr)
EA (1) EA028749B1 (sr)
ES (1) ES2688817T3 (sr)
HK (1) HK1204552A1 (sr)
HR (1) HRP20181583T1 (sr)
IL (1) IL235466B (sr)
LT (1) LT2846780T (sr)
MX (1) MX358545B (sr)
MY (1) MY171378A (sr)
NZ (1) NZ630248A (sr)
PE (1) PE20142439A1 (sr)
PH (1) PH12014502405A1 (sr)
PL (1) PL2846780T3 (sr)
PT (1) PT2846780T (sr)
RS (1) RS57881B1 (sr)
SG (1) SG11201406964QA (sr)
SI (1) SI2846780T1 (sr)
TW (1) TWI577392B (sr)
UY (1) UY34785A (sr)
WO (1) WO2013169520A1 (sr)
ZA (1) ZA201408967B (sr)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20150119317A1 (en) * 2012-05-07 2015-04-30 Bristol-Myers Squibb Company Oral solid dosage formulation of 1,1-dimethylethyl [(1s)-1-carbamoyl)pyrrolidin-1-yl]carbonyl}-2,2-dimethylpropyl]carbamate
KR20150074051A (ko) 2012-10-19 2015-07-01 브리스톨-마이어스 스큅 컴퍼니 C형 간염 바이러스 억제제
WO2014070964A1 (en) 2012-11-02 2014-05-08 Bristol-Myers Squibb Company Hepatitis c virus inhibitors
WO2014071007A1 (en) 2012-11-02 2014-05-08 Bristol-Myers Squibb Company Hepatitis c virus inhibitors
US9643999B2 (en) 2012-11-02 2017-05-09 Bristol-Myers Squibb Company Hepatitis C virus inhibitors
US9409943B2 (en) 2012-11-05 2016-08-09 Bristol-Myers Squibb Company Hepatitis C virus inhibitors
JP6342922B2 (ja) 2013-03-07 2018-06-13 ブリストル−マイヤーズ スクイブ カンパニーＢｒｉｓｔｏｌ−Ｍｙｅｒｓ Ｓｑｕｉｂｂ Ｃｏｍｐａｎｙ Ｃ型肝炎ウイルス阻害剤
WO2019130341A1 (en) * 2017-12-26 2019-07-04 Hetero Labs Limited Capsule compositions comprising lopinavir and ritonavir

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA9710071B (en) * 1996-11-21 1998-05-25 Abbott Lab Pharmaceutical composition.
ATE381922T1 (de) * 2000-10-31 2008-01-15 Boehringer Ingelheim Pharma Perorale, selbst-emulgierende darreichungsformen von pyranon-proteaseinhibitoren
US6828301B2 (en) * 2002-02-07 2004-12-07 Boehringer Ingelheim International Gmbh Pharmaceutical compositions for hepatitis C viral protease inhibitors
MY140680A (en) 2002-05-20 2010-01-15 Bristol Myers Squibb Co Hepatitis c virus inhibitors
WO2010042834A1 (en) * 2008-10-09 2010-04-15 Anadys Pharmaceuticals, Inc. A method of inhibiting hepatitis c virus by combination of a 5,6-dihydro-1h-pyridin-2-one and one or more additional antiviral compounds
US8252821B2 (en) * 2009-04-14 2012-08-28 Bristol-Myers Squibb Company Bioavailable capsule compositions of amorphous alpha-(N-sulfonamido)acetamide compound

Also Published As

Publication number Publication date
PH12014502405A1 (en) 2015-01-12
BR112014027676A2 (pt) 2017-06-27
MX2014013220A (es) 2015-05-11
PT2846780T (pt) 2018-10-26
ZA201408967B (en) 2016-10-26
PE20142439A1 (es) 2015-01-28
EA201492039A1 (ru) 2015-02-27
WO2013169520A1 (en) 2013-11-14
US20130302414A1 (en) 2013-11-14
AU2013260005A1 (en) 2015-01-15
AU2013260005B2 (en) 2017-07-13
CO7141457A2 (es) 2014-12-12
CN104363899A (zh) 2015-02-18
CA2872765A1 (en) 2013-11-14
PL2846780T3 (pl) 2018-11-30
DK2846780T3 (en) 2018-09-17
AR090954A1 (es) 2014-12-17
EP2846780A1 (en) 2015-03-18
EA028749B1 (ru) 2017-12-29
ES2688817T3 (es) 2018-11-07
SI2846780T1 (sl) 2018-09-28
CY1120756T1 (el) 2019-12-11
LT2846780T (lt) 2018-11-12
SG11201406964QA (en) 2014-11-27
MY171378A (en) 2019-10-10
UY34785A (es) 2013-11-29
IL235466B (en) 2019-03-31
NZ630248A (en) 2016-11-25
HK1204552A1 (en) 2015-11-27
CL2014003012A1 (es) 2015-07-10
TW201350145A (zh) 2013-12-16
JP6276756B2 (ja) 2018-02-07
TWI577392B (zh) 2017-04-11
EP2846780B1 (en) 2018-07-18
HRP20181583T1 (hr) 2018-11-30
JP2015516418A (ja) 2015-06-11
MX358545B (es) 2018-08-24
KR20150004921A (ko) 2015-01-13

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