MXPA06001129A - Proceso para controlar una estructura cristalina de risedronato. - Google Patents
Proceso para controlar una estructura cristalina de risedronato.Info
- Publication number
- MXPA06001129A MXPA06001129A MXPA06001129A MXPA06001129A MXPA06001129A MX PA06001129 A MXPA06001129 A MX PA06001129A MX PA06001129 A MXPA06001129 A MX PA06001129A MX PA06001129 A MXPA06001129 A MX PA06001129A MX PA06001129 A MXPA06001129 A MX PA06001129A
- Authority
- MX
- Mexico
- Prior art keywords
- risedronate
- crystal structure
- controlling crystal
- controlling
- hydrate
- Prior art date
Links
- 238000000034 method Methods 0.000 title abstract 3
- IIDJRNMFWXDHID-UHFFFAOYSA-N Risedronic acid Chemical compound OP(=O)(O)C(P(O)(O)=O)(O)CC1=CC=CN=C1 IIDJRNMFWXDHID-UHFFFAOYSA-N 0.000 title abstract 2
- 239000013078 crystal Substances 0.000 title abstract 2
- 229940089617 risedronate Drugs 0.000 title abstract 2
- 239000002253 acid Substances 0.000 abstract 1
- 230000006911 nucleation Effects 0.000 abstract 1
- 238000010899 nucleation Methods 0.000 abstract 1
- 238000010979 pH adjustment Methods 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/553—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
- C07F9/576—Six-membered rings
- C07F9/58—Pyridine rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Biochemistry (AREA)
- General Health & Medical Sciences (AREA)
- Molecular Biology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Crystals, And After-Treatments Of Crystals (AREA)
- Glass Compositions (AREA)
- Steroid Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Pyridine Compounds (AREA)
- Yarns And Mechanical Finishing Of Yarns Or Ropes (AREA)
- Pens And Brushes (AREA)
- Seasonings (AREA)
Abstract
La presente invencion se relaciona con un proceso para controlar la forma cristalina de una sal del acido 3-piridil-1-hidroxil-etilideno-1,1-bisfosfonico (Risedronato); el proceso emplea un ajuste del pH para inducir la forma hidratada correcta y en consecuencia evitar la nucleacion accidental de las formas hidratadas no deseadas.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US49122203P | 2003-07-30 | 2003-07-30 | |
| PCT/US2004/022703 WO2005012314A1 (en) | 2003-07-30 | 2004-07-15 | Process for controlling crystal structure of risedronate |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MXPA06001129A true MXPA06001129A (es) | 2006-04-11 |
Family
ID=34115482
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MXPA06001129A MXPA06001129A (es) | 2003-07-30 | 2004-07-15 | Proceso para controlar una estructura cristalina de risedronato. |
Country Status (20)
| Country | Link |
|---|---|
| US (1) | US7002014B2 (es) |
| EP (1) | EP1651656B1 (es) |
| JP (1) | JP4423614B2 (es) |
| KR (1) | KR100786044B1 (es) |
| CN (1) | CN100439377C (es) |
| AT (1) | ATE493423T1 (es) |
| AU (1) | AU2004261561B9 (es) |
| BR (1) | BRPI0413067A (es) |
| CA (1) | CA2529470C (es) |
| CO (1) | CO5660304A2 (es) |
| DE (1) | DE602004030801D1 (es) |
| IL (1) | IL172676A (es) |
| IS (1) | IS2915B (es) |
| MA (1) | MA27914A1 (es) |
| MX (1) | MXPA06001129A (es) |
| NO (1) | NO335393B1 (es) |
| NZ (1) | NZ544030A (es) |
| RU (1) | RU2319706C2 (es) |
| SG (1) | SG144151A1 (es) |
| WO (1) | WO2005012314A1 (es) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1775302A1 (en) | 2005-10-11 | 2007-04-18 | Sandoz A/S | Method for preparing crystalline sodium risedronate |
| JP5052816B2 (ja) * | 2006-04-26 | 2012-10-17 | 株式会社パーマケム・アジア | ３−ピリジル−１−ヒドロキシエチリデン−１、１−ビスホスホン酸ナトリウム塩２．５水和物ａ型結晶の製造方法 |
| JP5354858B2 (ja) * | 2006-05-09 | 2013-11-27 | 株式会社Ａｄｅｋａ | スルホンアミド化合物の金属塩を含有するポリエステル樹脂組成物 |
| US8076483B2 (en) | 2006-05-11 | 2011-12-13 | M/S. Ind Swift Laboratories Limited | Process for the preparation of pure risedronic acid or salts |
| WO2008044245A2 (en) * | 2006-10-10 | 2008-04-17 | Matrix Laboratories Ltd | A process for the preparation of risedronate sodium hemipentahydrate |
| KR100828705B1 (ko) * | 2006-12-04 | 2008-05-09 | 씨제이제일제당 (주) | 리세드론산 나트륨 수화물의 제조방법 |
| KR100775440B1 (ko) * | 2006-12-20 | 2007-11-12 | 동우신테크 주식회사 | 리세드로네이트 나트륨 헤미펜타히드레이트의 제조방법 |
| KR100798855B1 (ko) * | 2007-02-14 | 2008-01-28 | 주식회사 엔지켐 | 리세드론산 나트륨 헤미펜타하이드레이트의 제조방법 |
| KR100812528B1 (ko) * | 2007-04-12 | 2008-03-12 | 보령제약 주식회사 | 리세드로네이트 나트륨염의 헤미펜타히드레이트의 선택적결정화방법 |
| WO2009050731A2 (en) * | 2007-06-20 | 2009-04-23 | Alkem Laboratories Ltd | Novel process for preparing risedronic acid |
| WO2009034580A1 (en) * | 2007-09-11 | 2009-03-19 | Fleming Laboratories Limited | Improved process for the preparation of risedronate sodium hemipentahydrate |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IL77243A (en) | 1984-12-21 | 1996-11-14 | Procter & Gamble | Pharmaceutical compositions containing geminal diphosphonic acid compounds and certain such novel compounds |
| SK279589B6 (sk) | 1991-11-22 | 1999-01-11 | Procter And Gamble Pharmaceuticals | Farmaceutický prípravok s retardovaným uvoľňovaním |
| PE20011061A1 (es) * | 2000-02-01 | 2001-11-20 | Procter & Gamble | Cristalizacion selectiva del acido 3-piridil-1-hidroxi-etiliden-1,1-bisfosfonico sodio como el hemipentahidrato o el monohidrato |
-
2004
- 2004-07-15 CA CA2529470A patent/CA2529470C/en active Active
- 2004-07-15 EP EP04778281A patent/EP1651656B1/en active Active
- 2004-07-15 SG SG200804444-8A patent/SG144151A1/en unknown
- 2004-07-15 KR KR1020067000683A patent/KR100786044B1/ko active IP Right Grant
- 2004-07-15 MX MXPA06001129A patent/MXPA06001129A/es active IP Right Grant
- 2004-07-15 JP JP2006521878A patent/JP4423614B2/ja active Active
- 2004-07-15 NZ NZ544030A patent/NZ544030A/en unknown
- 2004-07-15 AU AU2004261561A patent/AU2004261561B9/en active Active
- 2004-07-15 CN CNB2004800205190A patent/CN100439377C/zh active Active
- 2004-07-15 RU RU2006102357/04A patent/RU2319706C2/ru active
- 2004-07-15 DE DE602004030801T patent/DE602004030801D1/de active Active
- 2004-07-15 BR BRPI0413067-7A patent/BRPI0413067A/pt not_active Application Discontinuation
- 2004-07-15 WO PCT/US2004/022703 patent/WO2005012314A1/en active Application Filing
- 2004-07-15 AT AT04778281T patent/ATE493423T1/de not_active IP Right Cessation
- 2004-07-29 US US10/901,692 patent/US7002014B2/en active Active
-
2005
- 2005-12-18 IL IL172676A patent/IL172676A/en active IP Right Grant
-
2006
- 2006-01-25 IS IS8262A patent/IS2915B/is unknown
- 2006-01-26 MA MA28754A patent/MA27914A1/fr unknown
- 2006-02-27 CO CO06019211A patent/CO5660304A2/es not_active Application Discontinuation
- 2006-02-27 NO NO20060950A patent/NO335393B1/no unknown
Also Published As
| Publication number | Publication date |
|---|---|
| AU2004261561A1 (en) | 2005-02-10 |
| IS8262A (is) | 2006-01-25 |
| AU2004261561B2 (en) | 2008-06-26 |
| WO2005012314A1 (en) | 2005-02-10 |
| KR20060054297A (ko) | 2006-05-22 |
| JP4423614B2 (ja) | 2010-03-03 |
| US7002014B2 (en) | 2006-02-21 |
| AU2004261561B9 (en) | 2008-10-30 |
| CA2529470C (en) | 2010-11-23 |
| IS2915B (is) | 2014-12-15 |
| RU2006102357A (ru) | 2006-07-27 |
| MA27914A1 (fr) | 2006-05-02 |
| US20050026869A1 (en) | 2005-02-03 |
| NZ544030A (en) | 2008-05-30 |
| NO335393B1 (no) | 2014-12-08 |
| CA2529470A1 (en) | 2005-02-10 |
| IL172676A0 (en) | 2006-04-10 |
| EP1651656A1 (en) | 2006-05-03 |
| CN1823078A (zh) | 2006-08-23 |
| CN100439377C (zh) | 2008-12-03 |
| IL172676A (en) | 2010-12-30 |
| JP2007500189A (ja) | 2007-01-11 |
| CO5660304A2 (es) | 2006-07-31 |
| BRPI0413067A (pt) | 2006-10-17 |
| SG144151A1 (en) | 2008-07-29 |
| ATE493423T1 (de) | 2011-01-15 |
| RU2319706C2 (ru) | 2008-03-20 |
| EP1651656B1 (en) | 2010-12-29 |
| DE602004030801D1 (de) | 2011-02-10 |
| KR100786044B1 (ko) | 2007-12-17 |
| NO20060950L (no) | 2006-02-27 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FG | Grant or registration | ||
| GB | Transfer or rights |