BRPI0413067A - processo para controlar a estrututra cristalina do risedronato - Google Patents
processo para controlar a estrututra cristalina do risedronatoInfo
- Publication number
- BRPI0413067A BRPI0413067A BRPI0413067-7A BRPI0413067A BRPI0413067A BR PI0413067 A BRPI0413067 A BR PI0413067A BR PI0413067 A BRPI0413067 A BR PI0413067A BR PI0413067 A BRPI0413067 A BR PI0413067A
- Authority
- BR
- Brazil
- Prior art keywords
- risedronate
- control
- crystal structure
- hydrate
- ethylidene
- Prior art date
Links
- 238000000034 method Methods 0.000 title abstract 3
- IIDJRNMFWXDHID-UHFFFAOYSA-N Risedronic acid Chemical compound OP(=O)(O)C(P(O)(O)=O)(O)CC1=CC=CN=C1 IIDJRNMFWXDHID-UHFFFAOYSA-N 0.000 title abstract 2
- 239000013078 crystal Substances 0.000 title abstract 2
- 229940089617 risedronate Drugs 0.000 title abstract 2
- 239000002253 acid Substances 0.000 abstract 1
- 230000006911 nucleation Effects 0.000 abstract 1
- 238000010899 nucleation Methods 0.000 abstract 1
- 238000010979 pH adjustment Methods 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/553—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
- C07F9/576—Six-membered rings
- C07F9/58—Pyridine rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Biochemistry (AREA)
- General Health & Medical Sciences (AREA)
- Molecular Biology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Crystals, And After-Treatments Of Crystals (AREA)
- Glass Compositions (AREA)
- Steroid Compounds (AREA)
- Seasonings (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Pyridine Compounds (AREA)
- Pens And Brushes (AREA)
- Yarns And Mechanical Finishing Of Yarns Or Ropes (AREA)
Abstract
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US49122203P | 2003-07-30 | 2003-07-30 | |
PCT/US2004/022703 WO2005012314A1 (en) | 2003-07-30 | 2004-07-15 | Process for controlling crystal structure of risedronate |
Publications (1)
Publication Number | Publication Date |
---|---|
BRPI0413067A true BRPI0413067A (pt) | 2006-10-17 |
Family
ID=34115482
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI0413067-7A BRPI0413067A (pt) | 2003-07-30 | 2004-07-15 | processo para controlar a estrututra cristalina do risedronato |
Country Status (20)
Country | Link |
---|---|
US (1) | US7002014B2 (pt) |
EP (1) | EP1651656B1 (pt) |
JP (1) | JP4423614B2 (pt) |
KR (1) | KR100786044B1 (pt) |
CN (1) | CN100439377C (pt) |
AT (1) | ATE493423T1 (pt) |
AU (1) | AU2004261561B9 (pt) |
BR (1) | BRPI0413067A (pt) |
CA (1) | CA2529470C (pt) |
CO (1) | CO5660304A2 (pt) |
DE (1) | DE602004030801D1 (pt) |
IL (1) | IL172676A (pt) |
IS (1) | IS2915B (pt) |
MA (1) | MA27914A1 (pt) |
MX (1) | MXPA06001129A (pt) |
NO (1) | NO335393B1 (pt) |
NZ (1) | NZ544030A (pt) |
RU (1) | RU2319706C2 (pt) |
SG (1) | SG144151A1 (pt) |
WO (1) | WO2005012314A1 (pt) |
Families Citing this family (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP1775302A1 (en) | 2005-10-11 | 2007-04-18 | Sandoz A/S | Method for preparing crystalline sodium risedronate |
JP5052816B2 (ja) * | 2006-04-26 | 2012-10-17 | 株式会社パーマケム・アジア | 3−ピリジル−1−ヒドロキシエチリデン−1、1−ビスホスホン酸ナトリウム塩2.5水和物a型結晶の製造方法 |
JP5354858B2 (ja) * | 2006-05-09 | 2013-11-27 | 株式会社Adeka | スルホンアミド化合物の金属塩を含有するポリエステル樹脂組成物 |
KR20090005206A (ko) | 2006-05-11 | 2009-01-12 | 인드-스위프트 래버러토리즈 리미티드 | 순수한 리세드론산 또는 염의 제조 방법 |
WO2008044245A2 (en) * | 2006-10-10 | 2008-04-17 | Matrix Laboratories Ltd | A process for the preparation of risedronate sodium hemipentahydrate |
KR100828705B1 (ko) * | 2006-12-04 | 2008-05-09 | 씨제이제일제당 (주) | 리세드론산 나트륨 수화물의 제조방법 |
KR100775440B1 (ko) * | 2006-12-20 | 2007-11-12 | 동우신테크 주식회사 | 리세드로네이트 나트륨 헤미펜타히드레이트의 제조방법 |
KR100798855B1 (ko) * | 2007-02-14 | 2008-01-28 | 주식회사 엔지켐 | 리세드론산 나트륨 헤미펜타하이드레이트의 제조방법 |
KR100812528B1 (ko) * | 2007-04-12 | 2008-03-12 | 보령제약 주식회사 | 리세드로네이트 나트륨염의 헤미펜타히드레이트의 선택적결정화방법 |
WO2009050731A2 (en) * | 2007-06-20 | 2009-04-23 | Alkem Laboratories Ltd | Novel process for preparing risedronic acid |
WO2009034580A1 (en) * | 2007-09-11 | 2009-03-19 | Fleming Laboratories Limited | Improved process for the preparation of risedronate sodium hemipentahydrate |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IL77243A (en) * | 1984-12-21 | 1996-11-14 | Procter & Gamble | Pharmaceutical compositions containing geminal diphosphonic acid compounds and certain such novel compounds |
CZ282760B6 (cs) * | 1991-11-22 | 1997-09-17 | Procter And Gamble Pharmaceuticals, Inc. | Risedronátové prostředky se zpožděným uvolňováním |
PE20011061A1 (es) * | 2000-02-01 | 2001-11-20 | Procter & Gamble | Cristalizacion selectiva del acido 3-piridil-1-hidroxi-etiliden-1,1-bisfosfonico sodio como el hemipentahidrato o el monohidrato |
-
2004
- 2004-07-15 MX MXPA06001129A patent/MXPA06001129A/es active IP Right Grant
- 2004-07-15 CA CA2529470A patent/CA2529470C/en active Active
- 2004-07-15 BR BRPI0413067-7A patent/BRPI0413067A/pt not_active Application Discontinuation
- 2004-07-15 EP EP04778281A patent/EP1651656B1/en active Active
- 2004-07-15 JP JP2006521878A patent/JP4423614B2/ja active Active
- 2004-07-15 AT AT04778281T patent/ATE493423T1/de not_active IP Right Cessation
- 2004-07-15 NZ NZ544030A patent/NZ544030A/en unknown
- 2004-07-15 CN CNB2004800205190A patent/CN100439377C/zh active Active
- 2004-07-15 DE DE602004030801T patent/DE602004030801D1/de active Active
- 2004-07-15 AU AU2004261561A patent/AU2004261561B9/en active Active
- 2004-07-15 WO PCT/US2004/022703 patent/WO2005012314A1/en active Application Filing
- 2004-07-15 KR KR1020067000683A patent/KR100786044B1/ko active IP Right Grant
- 2004-07-15 RU RU2006102357/04A patent/RU2319706C2/ru active
- 2004-07-15 SG SG200804444-8A patent/SG144151A1/en unknown
- 2004-07-29 US US10/901,692 patent/US7002014B2/en active Active
-
2005
- 2005-12-18 IL IL172676A patent/IL172676A/en active IP Right Grant
-
2006
- 2006-01-25 IS IS8262A patent/IS2915B/is unknown
- 2006-01-26 MA MA28754A patent/MA27914A1/fr unknown
- 2006-02-27 NO NO20060950A patent/NO335393B1/no unknown
- 2006-02-27 CO CO06019211A patent/CO5660304A2/es not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
CN100439377C (zh) | 2008-12-03 |
EP1651656A1 (en) | 2006-05-03 |
IL172676A0 (en) | 2006-04-10 |
IS2915B (is) | 2014-12-15 |
EP1651656B1 (en) | 2010-12-29 |
RU2319706C2 (ru) | 2008-03-20 |
CA2529470C (en) | 2010-11-23 |
CO5660304A2 (es) | 2006-07-31 |
NO20060950L (no) | 2006-02-27 |
WO2005012314A1 (en) | 2005-02-10 |
ATE493423T1 (de) | 2011-01-15 |
US7002014B2 (en) | 2006-02-21 |
NZ544030A (en) | 2008-05-30 |
MA27914A1 (fr) | 2006-05-02 |
JP2007500189A (ja) | 2007-01-11 |
KR100786044B1 (ko) | 2007-12-17 |
DE602004030801D1 (de) | 2011-02-10 |
AU2004261561B9 (en) | 2008-10-30 |
KR20060054297A (ko) | 2006-05-22 |
CN1823078A (zh) | 2006-08-23 |
MXPA06001129A (es) | 2006-04-11 |
IS8262A (is) | 2006-01-25 |
AU2004261561A1 (en) | 2005-02-10 |
SG144151A1 (en) | 2008-07-29 |
US20050026869A1 (en) | 2005-02-03 |
RU2006102357A (ru) | 2006-07-27 |
NO335393B1 (no) | 2014-12-08 |
JP4423614B2 (ja) | 2010-03-03 |
CA2529470A1 (en) | 2005-02-10 |
AU2004261561B2 (en) | 2008-06-26 |
IL172676A (en) | 2010-12-30 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B25A | Requested transfer of rights approved |
Owner name: WARNER CHILCOTT COMPANY, LLC (PR) |
|
B06F | Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette] | ||
B07D | Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette] | ||
B25E | Requested change of name of applicant rejected |
Owner name: WARNER CHILCOTT COMPANY, LLC (PR) |
|
B07E | Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette] | ||
B07A | Application suspended after technical examination (opinion) [chapter 7.1 patent gazette] | ||
B06G | Technical and formal requirements: other requirements [chapter 6.7 patent gazette] | ||
B06I | Publication of requirement cancelled [chapter 6.9 patent gazette] |
Free format text: ANULADA A PUBLICACAO CODIGO 6.7 NA RPI NO 2505 DE 08/01/2019 POR TER SIDO INDEVIDA. |
|
B09B | Patent application refused [chapter 9.2 patent gazette] | ||
B12B | Appeal against refusal [chapter 12.2 patent gazette] | ||
B25E | Requested change of name of applicant rejected |
Owner name: WARNER CHILCOTT COMPANY, LLC (PR) Free format text: INDEFERIDO O PEDIDO DE ALTERACAO DE NOME CONTIDO NA PETICAO 870220023201 DE 17/03/2022, EM VIRTUDE DA MANUTENCAO DO INDEFERIMENTO DO PEDIDO, CONFORME PUBLICADO NA RPI2620 DE 23/03/2021. |
|
B25B | Requested transfer of rights rejected |
Owner name: WARNER CHILCOTT COMPANY, LLC (PR) Free format text: INDEFERIDO O PEDIDO DE TRANSFERENCIA CONTIDO NA PETICAO 870220023212 DE 17/03/2022, EM VIRTUDE DE TER SIDO MANTIDO O INDEFERIMENTO DO PEDIDO, CONFORME PUBLICADO NA RPI2620 DE 23/03/2021. |