MXPA05007571A - Tratamiento para hiperplasia protatica benigna utilizando agentes energoliticos. - Google Patents
Tratamiento para hiperplasia protatica benigna utilizando agentes energoliticos.Info
- Publication number
- MXPA05007571A MXPA05007571A MXPA05007571A MXPA05007571A MXPA05007571A MX PA05007571 A MXPA05007571 A MX PA05007571A MX PA05007571 A MXPA05007571 A MX PA05007571A MX PA05007571 A MXPA05007571 A MX PA05007571A MX PA05007571 A MXPA05007571 A MX PA05007571A
- Authority
- MX
- Mexico
- Prior art keywords
- cells
- bph
- agent
- citrate
- treatment
- Prior art date
Links
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- JOXIMZWYDAKGHI-UHFFFAOYSA-N toluene-4-sulfonic acid Chemical compound CC1=CC=C(S(O)(=O)=O)C=C1 JOXIMZWYDAKGHI-UHFFFAOYSA-N 0.000 description 1
- 239000012049 topical pharmaceutical composition Substances 0.000 description 1
- 231100000041 toxicology testing Toxicity 0.000 description 1
- 238000012546 transfer Methods 0.000 description 1
- 230000009466 transformation Effects 0.000 description 1
- 150000003627 tricarboxylic acid derivatives Chemical class 0.000 description 1
- WGIWBXUNRXCYRA-UHFFFAOYSA-H trizinc;2-hydroxypropane-1,2,3-tricarboxylate Chemical compound [Zn+2].[Zn+2].[Zn+2].[O-]C(=O)CC(O)(CC([O-])=O)C([O-])=O.[O-]C(=O)CC(O)(CC([O-])=O)C([O-])=O WGIWBXUNRXCYRA-UHFFFAOYSA-H 0.000 description 1
- 208000014001 urinary system disease Diseases 0.000 description 1
- 210000001635 urinary tract Anatomy 0.000 description 1
- 208000019206 urinary tract infection Diseases 0.000 description 1
- 230000003202 urodynamic effect Effects 0.000 description 1
- 235000012431 wafers Nutrition 0.000 description 1
- 238000004804 winding Methods 0.000 description 1
- 239000004246 zinc acetate Substances 0.000 description 1
- 229960000314 zinc acetate Drugs 0.000 description 1
- 229940062776 zinc aspartate Drugs 0.000 description 1
- 239000011592 zinc chloride Substances 0.000 description 1
- 235000005074 zinc chloride Nutrition 0.000 description 1
- 229960001939 zinc chloride Drugs 0.000 description 1
- 239000011746 zinc citrate Substances 0.000 description 1
- 235000006076 zinc citrate Nutrition 0.000 description 1
- 229940068475 zinc citrate Drugs 0.000 description 1
- 239000011670 zinc gluconate Substances 0.000 description 1
- 235000011478 zinc gluconate Nutrition 0.000 description 1
- 229960000306 zinc gluconate Drugs 0.000 description 1
- 239000011787 zinc oxide Substances 0.000 description 1
- 229940032991 zinc picolinate Drugs 0.000 description 1
- NWONKYPBYAMBJT-UHFFFAOYSA-L zinc sulfate Chemical compound [Zn+2].[O-]S([O-])(=O)=O NWONKYPBYAMBJT-UHFFFAOYSA-L 0.000 description 1
- 229960001763 zinc sulfate Drugs 0.000 description 1
- 229910000368 zinc sulfate Inorganic materials 0.000 description 1
- POEVDIARYKIEGF-CEOVSRFSSA-L zinc;(2s)-2-aminobutanedioate;hydron Chemical compound [Zn+2].[O-]C(=O)[C@@H](N)CC(O)=O.[O-]C(=O)[C@@H](N)CC(O)=O POEVDIARYKIEGF-CEOVSRFSSA-L 0.000 description 1
- JNPQFTCBVDSMDO-UHFFFAOYSA-L zinc;2,3-dihydroxypropanoate Chemical compound [Zn+2].OCC(O)C([O-])=O.OCC(O)C([O-])=O JNPQFTCBVDSMDO-UHFFFAOYSA-L 0.000 description 1
- NHVUUBRKFZWXRN-UHFFFAOYSA-L zinc;pyridine-2-carboxylate Chemical compound C=1C=CC=NC=1C(=O)O[Zn]OC(=O)C1=CC=CC=N1 NHVUUBRKFZWXRN-UHFFFAOYSA-L 0.000 description 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
- A61K31/416—1,2-Diazoles condensed with carbocyclic ring systems, e.g. indazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/08—Drugs for disorders of the urinary system of the prostate
-
- G—PHYSICS
- G01—MEASURING; TESTING
- G01N—INVESTIGATING OR ANALYSING MATERIALS BY DETERMINING THEIR CHEMICAL OR PHYSICAL PROPERTIES
- G01N2800/00—Detection or diagnosis of diseases
- G01N2800/34—Genitourinary disorders
- G01N2800/342—Prostate diseases, e.g. BPH, prostatitis
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Molecular Biology (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Urology & Nephrology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
- Micro-Organisms Or Cultivation Processes Thereof (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Steroid Compounds (AREA)
Applications Claiming Priority (10)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US44111003P | 2003-01-17 | 2003-01-17 | |
| US44234403P | 2003-01-23 | 2003-01-23 | |
| US45866503P | 2003-03-28 | 2003-03-28 | |
| US45866303P | 2003-03-28 | 2003-03-28 | |
| US45884603P | 2003-03-28 | 2003-03-28 | |
| US46001203P | 2003-04-02 | 2003-04-02 | |
| US47290703P | 2003-05-22 | 2003-05-22 | |
| US48826503P | 2003-07-18 | 2003-07-18 | |
| US49616303P | 2003-08-18 | 2003-08-18 | |
| PCT/US2004/001146 WO2004064736A2 (en) | 2003-01-17 | 2004-01-16 | Treatment of benign prostatic hyperplasia using energolytic agents |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MXPA05007571A true MXPA05007571A (es) | 2005-11-17 |
Family
ID=32777423
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MXPA05007571A MXPA05007571A (es) | 2003-01-17 | 2004-01-16 | Tratamiento para hiperplasia protatica benigna utilizando agentes energoliticos. |
| MXPA05007572A MXPA05007572A (es) | 2003-01-17 | 2004-01-16 | Tratamiento de hiperplasia prostatica benigna. |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MXPA05007572A MXPA05007572A (es) | 2003-01-17 | 2004-01-16 | Tratamiento de hiperplasia prostatica benigna. |
Country Status (13)
| Country | Link |
|---|---|
| US (4) | US6989400B2 (enExample) |
| EP (2) | EP1610778A4 (enExample) |
| JP (2) | JP2006518343A (enExample) |
| KR (2) | KR20050098250A (enExample) |
| AU (2) | AU2004206870A1 (enExample) |
| BR (1) | BRPI0406796A (enExample) |
| CA (2) | CA2513572A1 (enExample) |
| DE (1) | DE04702967T1 (enExample) |
| ES (1) | ES2254046T1 (enExample) |
| IL (1) | IL169685A0 (enExample) |
| MX (2) | MXPA05007571A (enExample) |
| NO (1) | NO20053783L (enExample) |
| WO (2) | WO2004064735A2 (enExample) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7795227B2 (en) | 2004-06-17 | 2010-09-14 | Wisconsin Alumni Research Foundation | Compounds and methods for treating seizure disorders |
Families Citing this family (21)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7547673B2 (en) * | 2001-09-13 | 2009-06-16 | The Johns Hopkins University | Therapeutics for cancer using 3-bromopyruvate and other selective inhibitors of ATP production |
| US7524885B2 (en) * | 2002-04-01 | 2009-04-28 | The Governors Of The University Of Alberta | Compounds that stimulate glucose utilization and methods of use |
| WO2004064735A2 (en) | 2003-01-17 | 2004-08-05 | Threshold Pharmaceuticals, Inc. | Treatment of benign prostatic hyperplasia |
| WO2006091790A1 (en) | 2005-02-23 | 2006-08-31 | Xenoport, Inc. | Platinum-containing compounds exhibiting cytostatic activity, synthesis and methods of use |
| US20060287253A1 (en) * | 2005-06-17 | 2006-12-21 | Kriegler Steven M | Compounds and methods for treating seizure disorders |
| US8324175B2 (en) | 2006-02-16 | 2012-12-04 | Young Hee Ko | Compositions and methods for the treatment of cancer |
| WO2007101148A2 (en) * | 2006-02-24 | 2007-09-07 | Board Of Regents, The University Of Texas System | Hexose compounds to treat cancer |
| CA2644809A1 (en) | 2006-03-02 | 2007-09-07 | Astellas Pharma Inc. | 17 .beta. hsd type 5 inhibitor |
| WO2008076964A1 (en) * | 2006-12-18 | 2008-06-26 | The Johns Hopkins University | Therapeutics for cancer using 3-bromopyruvate and other selective inhibitors of atp production |
| US20080245375A1 (en) * | 2007-04-05 | 2008-10-09 | Medtronic Vascular, Inc. | Benign Prostatic Hyperplasia Treatments |
| WO2009014150A1 (ja) | 2007-07-24 | 2009-01-29 | Astellas Pharma Inc. | ベンズイミダゾール誘導体 |
| SI2181990T1 (sl) | 2007-08-31 | 2012-10-30 | Astellas Pharma Inc | Piperidinski derivat |
| US8603123B2 (en) | 2008-04-28 | 2013-12-10 | Urotech, Inc. | Benign prostatic hyperplasia surgical system featuring mechanical coring probe with live aspiration |
| DK2331092T3 (da) | 2008-08-21 | 2014-05-19 | Univ Johns Hopkins | Fremgangsmåder og sammensætninger til indgivelse af 3-halopyruvat og associerede forbindelser til behandling af cancer |
| AU2010208062B2 (en) * | 2009-01-29 | 2014-07-24 | Kodiscovery, Llc | Compositions and methods for the treatment of cancer |
| WO2013153821A1 (ja) * | 2012-04-12 | 2013-10-17 | Omura Satoshi | Ｐｄｋ４阻害剤及びその利用 |
| US10441561B2 (en) | 2012-07-26 | 2019-10-15 | The William M. Yanbrough Foundation | Method for treating benign prostatic hyperplasia (BPH), prostatitis, and prostate cancer |
| JP6552509B2 (ja) | 2014-01-14 | 2019-07-31 | ザ・ジョンズ・ホプキンス・ユニバーシティー | 選択的ａｔｐ阻害剤をカプセル化するシクロデキストリン組成物およびその使用 |
| WO2017079563A1 (en) | 2015-11-06 | 2017-05-11 | The Johns Hopkins University | Methods of treating liver fibrosis by administering 3-bromopyruvate |
| EP3564214B1 (en) | 2018-05-04 | 2024-07-03 | Universita' Degli Studi G. D'annunzio Chieti - Pescara | Indazole derivatives as modulators of the cannabinoid system |
| CN116438162A (zh) * | 2020-09-17 | 2023-07-14 | 伊赛恩特制药公司 | Mas相关g蛋白受体x4的调节剂及相关产物和方法 |
Family Cites Families (20)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IT1052111B (it) * | 1972-02-29 | 1981-06-20 | Acraf | Acidi i benzil i h indazol 3 carbossilici sostituiti e loro derivati |
| US4684627A (en) * | 1981-09-08 | 1987-08-04 | Leveen Harry H | Treatment of cancer with phlorizin and its derivatives |
| CA1289077C (en) * | 1984-08-13 | 1991-09-17 | Harry H. Leveen | Treatment of cancer with phlorizin and its derivatives |
| US5260327A (en) * | 1985-10-02 | 1993-11-09 | Sloan-Kettering Institute For Cancer Research | Methods for inhibiting the proliferation of brain and hepatic metastases by using lonidamine |
| WO1992018132A1 (en) * | 1991-04-17 | 1992-10-29 | Merck & Co., Inc. | Pharmaceutical combination for the treatment of benign prostatic hyperplasia comtaining a 5 alpha-reductase inhibitor |
| US6063911A (en) * | 1993-12-01 | 2000-05-16 | Marine Polymer Technologies, Inc. | Methods and compositions for treatment of cell proliferative disorders |
| US5654320A (en) * | 1995-03-16 | 1997-08-05 | Eli Lilly And Company | Indazolecarboxamides |
| SK72996A3 (en) | 1995-06-07 | 1997-04-09 | Pfizer | Heterocyclic ring-fused pyrimidine derivatives and pharmaceutical compositions on their base |
| FR2737721B1 (fr) * | 1995-08-08 | 1997-09-05 | Roussel Uclaf | Nouveaux composes biphenyles, leur procede de preparation et les intermediaires de ce procede, leur application a titre de medicament et les compositions pharmaceutiques les contenant |
| ATE202551T1 (de) | 1995-10-18 | 2001-07-15 | Kanoldt Arzneimittel Gmbh | Lignane, verfahren zu ihrer herstellung, ihre pharmazeutische compositionen und anwendungen |
| DE19621319A1 (de) | 1996-05-28 | 1997-12-04 | Hoechst Ag | Bis-ortho-substituierte Benzoylguanidine, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament |
| US6054432A (en) | 1996-09-12 | 2000-04-25 | Asta Medica Aktiengesellschaft | Means for treating prostate hypertrophy and prostate cancer |
| IT1289938B1 (it) * | 1997-02-20 | 1998-10-19 | Angelini Ricerche Spa | Preparazione farmaceutica comprendente liposomi liofilizzati in cui e' incapsulato un principio attivo altamente insolubile in acqua e |
| IT1289939B1 (it) * | 1997-02-20 | 1998-10-19 | Angelini Ricerche Spa | Composizione farmaceutica acquosa comprendente un principio attivo altamente insolubile in acqua |
| CN1078462C (zh) * | 1997-07-09 | 2002-01-30 | 辛国芳 | 棉酚和/或其衍生物作为有效成分在制备用于治疗前列腺炎的栓剂中的应用 |
| EP1083896A4 (en) * | 1998-05-11 | 2002-09-11 | Endowment For Res In Human Bio | USE OF NEOMYCIN FOR TREATING ANGIOGENESIS-RELATED DISEASES |
| US6428968B1 (en) * | 1999-03-15 | 2002-08-06 | The Trustees Of The University Of Pennsylvania | Combined therapy with a chemotherapeutic agent and an oncolytic virus for killing tumor cells in a subject |
| US6001865A (en) * | 1999-05-04 | 1999-12-14 | Angelini Pharmaceuticals Inc. | 3-substituted 1-benzyl-1H-indazole derivatives as antifertility agents |
| WO2004064735A2 (en) | 2003-01-17 | 2004-08-05 | Threshold Pharmaceuticals, Inc. | Treatment of benign prostatic hyperplasia |
| SG151299A1 (en) * | 2004-03-25 | 2009-04-30 | Univ Michigan | Gossypol co-crystals and the use thereof |
-
2004
- 2004-01-16 WO PCT/US2004/001141 patent/WO2004064735A2/en not_active Ceased
- 2004-01-16 AU AU2004206870A patent/AU2004206870A1/en not_active Abandoned
- 2004-01-16 BR BR0406796-7A patent/BRPI0406796A/pt not_active Application Discontinuation
- 2004-01-16 MX MXPA05007571A patent/MXPA05007571A/es unknown
- 2004-01-16 JP JP2006500983A patent/JP2006518343A/ja not_active Withdrawn
- 2004-01-16 EP EP04702967A patent/EP1610778A4/en not_active Withdrawn
- 2004-01-16 CA CA002513572A patent/CA2513572A1/en not_active Abandoned
- 2004-01-16 KR KR1020057013200A patent/KR20050098250A/ko not_active Withdrawn
- 2004-01-16 WO PCT/US2004/001146 patent/WO2004064736A2/en not_active Ceased
- 2004-01-16 AU AU2004206869A patent/AU2004206869A1/en not_active Abandoned
- 2004-01-16 US US10/759,337 patent/US6989400B2/en not_active Expired - Fee Related
- 2004-01-16 MX MXPA05007572A patent/MXPA05007572A/es unknown
- 2004-01-16 CA CA002513575A patent/CA2513575A1/en not_active Abandoned
- 2004-01-16 DE DE04702967T patent/DE04702967T1/de active Pending
- 2004-01-16 EP EP04702976A patent/EP1592430A4/en not_active Withdrawn
- 2004-01-16 ES ES04702967T patent/ES2254046T1/es active Pending
- 2004-01-16 JP JP2006500981A patent/JP2006516571A/ja active Pending
- 2004-01-16 KR KR1020057013198A patent/KR20050098249A/ko not_active Withdrawn
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2005
- 2005-06-29 US US11/171,138 patent/US20050272796A1/en not_active Abandoned
- 2005-06-29 US US11/172,050 patent/US20050271723A1/en not_active Abandoned
- 2005-06-29 US US11/171,020 patent/US20050272795A1/en not_active Abandoned
- 2005-07-14 IL IL169685A patent/IL169685A0/en unknown
- 2005-08-09 NO NO20053783A patent/NO20053783L/no unknown
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7795227B2 (en) | 2004-06-17 | 2010-09-14 | Wisconsin Alumni Research Foundation | Compounds and methods for treating seizure disorders |
Also Published As
| Publication number | Publication date |
|---|---|
| AU2004206870A1 (en) | 2004-08-05 |
| JP2006518343A (ja) | 2006-08-10 |
| US20050272796A1 (en) | 2005-12-08 |
| WO2004064736A2 (en) | 2004-08-05 |
| AU2004206869A1 (en) | 2004-08-05 |
| US20050271723A1 (en) | 2005-12-08 |
| NO20053783D0 (no) | 2005-08-09 |
| US20040167196A1 (en) | 2004-08-26 |
| MXPA05007572A (es) | 2005-11-17 |
| KR20050098249A (ko) | 2005-10-11 |
| BRPI0406796A (pt) | 2006-01-17 |
| EP1592430A2 (en) | 2005-11-09 |
| EP1592430A4 (en) | 2006-05-31 |
| JP2006516571A (ja) | 2006-07-06 |
| US6989400B2 (en) | 2006-01-24 |
| IL169685A0 (en) | 2007-07-04 |
| US20050272795A1 (en) | 2005-12-08 |
| WO2004064735A3 (en) | 2004-12-16 |
| WO2004064736A3 (en) | 2005-05-06 |
| NO20053783L (no) | 2005-09-27 |
| CA2513572A1 (en) | 2004-08-05 |
| EP1610778A2 (en) | 2006-01-04 |
| EP1610778A4 (en) | 2006-05-31 |
| DE04702967T1 (de) | 2006-06-22 |
| CA2513575A1 (en) | 2004-08-05 |
| KR20050098250A (ko) | 2005-10-11 |
| ES2254046T1 (es) | 2006-06-16 |
| WO2004064735A2 (en) | 2004-08-05 |
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