MXPA03000772A - Derivados de acido hexahidro-7-1h-azepin-2-il-hexanoico como inhibidores de oxido nitrico sintasa inducible. - Google Patents

Derivados de acido hexahidro-7-1h-azepin-2-il-hexanoico como inhibidores de oxido nitrico sintasa inducible.

Info

Publication number
MXPA03000772A
MXPA03000772A MXPA03000772A MXPA03000772A MXPA03000772A MX PA03000772 A MXPA03000772 A MX PA03000772A MX PA03000772 A MXPA03000772 A MX PA03000772A MX PA03000772 A MXPA03000772 A MX PA03000772A MX PA03000772 A MXPA03000772 A MX PA03000772A
Authority
MX
Mexico
Prior art keywords
azepin
hexahydro
inhibitors
acid derivatives
nitric oxide
Prior art date
Application number
MXPA03000772A
Other languages
English (en)
Inventor
Donald W Hansen
Original Assignee
Pharmacia Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmacia Corp filed Critical Pharmacia Corp
Publication of MXPA03000772A publication Critical patent/MXPA03000772A/es

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    • C07D223/02—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D223/06—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom not condensed with other rings with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D223/12—Nitrogen atoms not forming part of a nitro radical
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D223/00—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom
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MXPA03000772A 2000-08-01 2001-08-01 Derivados de acido hexahidro-7-1h-azepin-2-il-hexanoico como inhibidores de oxido nitrico sintasa inducible. MXPA03000772A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US22217900P 2000-08-01 2000-08-01
PCT/US2001/024542 WO2002010139A1 (en) 2000-08-01 2001-08-01 Hexahydro-7-1h-azepin-2-yl-haxanoic acid derivatives as inhibitors of inducible nitric oxide synthase

Publications (1)

Publication Number Publication Date
MXPA03000772A true MXPA03000772A (es) 2003-06-04

Family

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Family Applications (1)

Application Number Title Priority Date Filing Date
MXPA03000772A MXPA03000772A (es) 2000-08-01 2001-08-01 Derivados de acido hexahidro-7-1h-azepin-2-il-hexanoico como inhibidores de oxido nitrico sintasa inducible.

Country Status (11)

Country Link
US (1) US6495544B2 (es)
EP (1) EP1305293A1 (es)
JP (1) JP2004512271A (es)
AR (1) AR032360A1 (es)
AU (1) AU2001281083A1 (es)
CA (1) CA2415851A1 (es)
EA (1) EA005817B1 (es)
MX (1) MXPA03000772A (es)
NZ (1) NZ523770A (es)
PE (1) PE20030413A1 (es)
WO (1) WO2002010139A1 (es)

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US7393652B2 (en) 2000-05-10 2008-07-01 The Trustees Of Columbia University In The City Of New York Methods for identifying a chemical compound that directly enhances binding of FKBP12.6 to PKA-phosphorylated type 2 ryanodine receptor (RyR2)
US7879840B2 (en) 2005-08-25 2011-02-01 The Trustees Of Columbia University In The City Of New York Agents for preventing and treating disorders involving modulation of the RyR receptors
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