AU2001270200A1 - Fatty acid synthase inhibitors - Google Patents
Fatty acid synthase inhibitorsInfo
- Publication number
- AU2001270200A1 AU2001270200A1 AU2001270200A AU7020001A AU2001270200A1 AU 2001270200 A1 AU2001270200 A1 AU 2001270200A1 AU 2001270200 A AU2001270200 A AU 2001270200A AU 7020001 A AU7020001 A AU 7020001A AU 2001270200 A1 AU2001270200 A1 AU 2001270200A1
- Authority
- AU
- Australia
- Prior art keywords
- fatty acid
- acid synthase
- synthase inhibitors
- inhibitors
- fatty
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US21428000P | 2000-06-27 | 2000-06-27 | |
US60214280 | 2000-06-27 | ||
PCT/US2001/020458 WO2002000646A1 (en) | 2000-06-27 | 2001-06-27 | Fatty acid synthase inhibitors |
Publications (1)
Publication Number | Publication Date |
---|---|
AU2001270200A1 true AU2001270200A1 (en) | 2002-01-08 |
Family
ID=22798484
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AU2001270200A Abandoned AU2001270200A1 (en) | 2000-06-27 | 2001-06-27 | Fatty acid synthase inhibitors |
Country Status (3)
Country | Link |
---|---|
US (1) | US6608059B1 (en) |
AU (1) | AU2001270200A1 (en) |
WO (1) | WO2002000646A1 (en) |
Families Citing this family (16)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP1553075B1 (en) | 2002-10-03 | 2013-08-14 | Ono Pharmaceutical Co., Ltd. | Lpa receptor antagonists |
WO2006060535A2 (en) * | 2004-11-30 | 2006-06-08 | Plexxikon, Inc. | Indole derivatives for use as ppar active compounds |
RU2416601C2 (en) * | 2005-02-25 | 2011-04-20 | Оно Фармасьютикал Ко., Лтд. | Indole compound and use thereof |
SG165362A1 (en) * | 2005-09-07 | 2010-10-28 | Plexxikon Inc | Ppar active compounds |
CN101117328B (en) * | 2006-08-01 | 2012-11-07 | 中国人民解放军军事医学科学院毒物药物研究所 | Fatty acid synthetase inhibitor and application for treating bacterial infection |
PE20090159A1 (en) * | 2007-03-08 | 2009-02-21 | Plexxikon Inc | INDOL-PROPIONIC ACID DERIVED COMPOUNDS AS PPARs MODULATORS |
AR072297A1 (en) | 2008-06-27 | 2010-08-18 | Novartis Ag | DERIVATIVES OF INDOL-2-IL-PIRIDIN-3-ILO, PHARMACEUTICAL COMPOSITION THAT INCLUDES THEM AND ITS USE IN MEDICINES FOR THE TREATMENT OF DISEASES MEDIATED BY THE SYNTHESIS ALDOSTERONE. |
TWI469965B (en) | 2008-12-22 | 2015-01-21 | Ono Pharmaceutical Co | Ethynylindole compounds |
EP2503890A4 (en) * | 2009-11-24 | 2013-05-15 | Glaxosmithkline Llc | Azabenzimidazoles as fatty acid synthase inhibitors |
US8450350B2 (en) | 2010-05-05 | 2013-05-28 | Infinity Pharmaceuticals, Inc. | Triazoles as inhibitors of fatty acid synthase |
EP2566853B1 (en) | 2010-05-05 | 2017-01-25 | Infinity Pharmaceuticals, Inc. | Tetrazolones as inhibitors of fatty acid synthase |
RU2560147C2 (en) | 2010-06-21 | 2015-08-20 | Оно Фармасьютикал Ко., Лтд. | Novel crystalline forms of 4,4'-[4-fluoro-7({4-[4-(3-fluoro-2-methylphenyl)butoxy]phenyl} ethynyl)-2-methyl-1h-indole-1,3-diiyl]dibutanoic acid, 4,4'-[2-methyl-7-({4-[4-(pentafluorophenyl)butoxy]phenyl} ethynyl)-1h-indole-1,3-diiyl]dibutanoic acid and 4,4'-[4-fluoro-2-methyl-7-({4-[4-(2,3,4,6-tetrafluorophenyl) butoxy]phenyl} ethynyl)-1h-indole-1,3-diiyl]dibutanoic acid |
US20130196971A1 (en) * | 2010-09-17 | 2013-08-01 | Christopher Joseph Aquino | Fatty acid synthase inhibitors |
US20160002188A1 (en) | 2013-03-13 | 2016-01-07 | Forma Therapeutics, Inc. | Novel compounds and compositions for inhibition of fasn |
TWI767148B (en) | 2018-10-10 | 2022-06-11 | 美商弗瑪治療公司 | Inhibiting fatty acid synthase (fasn) |
CN113382633A (en) | 2018-10-29 | 2021-09-10 | 福马治疗股份有限公司 | Solid forms of (4- (2-fluoro-4- (1-methyl-1H-benzo [ d ] imidazol-5-yl) benzoyl) piperazin-1-yl) (1-hydroxycyclopropyl) methanone |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IL109311A0 (en) | 1993-04-16 | 1994-07-31 | Lilly Co Eli | 1H-indole-3-acetamide sPla2 inhibitors |
FR2745003B1 (en) | 1996-02-16 | 1998-04-03 | Adir | NOVEL PSEUDOPEPTIDES DERIVED FROM NEUROKININS, THEIR PREPARATION PROCESS AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM |
US6486211B1 (en) * | 1999-10-22 | 2002-11-26 | Smithkline Beecham Corporation | Indole compounds |
-
2001
- 2001-06-27 WO PCT/US2001/020458 patent/WO2002000646A1/en active Application Filing
- 2001-06-27 AU AU2001270200A patent/AU2001270200A1/en not_active Abandoned
- 2001-06-27 US US10/296,774 patent/US6608059B1/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
US6608059B1 (en) | 2003-08-19 |
WO2002000646A1 (en) | 2002-01-03 |
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