MX373319B - Derivados de hexahidro-[1-4]diazepino[6,7,1-hi]indol-8-carboxamida como agonistas del receptor 5-ht2c y el uso de los mismos en el tratamiento de enfermedades relacionadas con dicho receptor. - Google Patents

Derivados de hexahidro-[1-4]diazepino[6,7,1-hi]indol-8-carboxamida como agonistas del receptor 5-ht2c y el uso de los mismos en el tratamiento de enfermedades relacionadas con dicho receptor.

Info

Publication number
MX373319B
MX373319B MX2017013902A MX2017013902A MX373319B MX 373319 B MX373319 B MX 373319B MX 2017013902 A MX2017013902 A MX 2017013902A MX 2017013902 A MX2017013902 A MX 2017013902A MX 373319 B MX373319 B MX 373319B
Authority
MX
Mexico
Prior art keywords
tobacco
individual attempting
addiction
smoking
disorders
Prior art date
Application number
MX2017013902A
Other languages
English (en)
Spanish (es)
Other versions
MX2017013902A (es
Inventor
Albert S Ren
Carleton R Sage
Graeme Semple
Xiuwen Zhu
Original Assignee
Arena Pharm Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Arena Pharm Inc filed Critical Arena Pharm Inc
Publication of MX2017013902A publication Critical patent/MX2017013902A/es
Publication of MX373319B publication Critical patent/MX373319B/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
    • A61K31/55131,4-Benzodiazepines, e.g. diazepam or clozapine
    • A61K31/55171,4-Benzodiazepines, e.g. diazepam or clozapine condensed with five-membered rings having nitrogen as a ring hetero atom, e.g. imidazobenzodiazepines, triazolam
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/06Peri-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Child & Adolescent Psychology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
MX2017013902A 2015-04-27 2016-04-26 Derivados de hexahidro-[1-4]diazepino[6,7,1-hi]indol-8-carboxamida como agonistas del receptor 5-ht2c y el uso de los mismos en el tratamiento de enfermedades relacionadas con dicho receptor. MX373319B (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201562153082P 2015-04-27 2015-04-27
PCT/US2016/029308 WO2016176177A1 (en) 2015-04-27 2016-04-26 5-ht2c receptor agonists and compositions and methods of use

Publications (2)

Publication Number Publication Date
MX2017013902A MX2017013902A (es) 2018-03-16
MX373319B true MX373319B (es) 2020-06-13

Family

ID=55949111

Family Applications (2)

Application Number Title Priority Date Filing Date
MX2017013902A MX373319B (es) 2015-04-27 2016-04-26 Derivados de hexahidro-[1-4]diazepino[6,7,1-hi]indol-8-carboxamida como agonistas del receptor 5-ht2c y el uso de los mismos en el tratamiento de enfermedades relacionadas con dicho receptor.
MX2020005898A MX2020005898A (es) 2015-04-27 2017-10-27 Derivados de hexahidro-[1,4]diazepino[6,7,1-hi]indol-8-carboxamida como agonistas del receptor 5-ht2c y el uso de los mismos en el tratamiento de enfermedades relacionadas con dicho receptor.

Family Applications After (1)

Application Number Title Priority Date Filing Date
MX2020005898A MX2020005898A (es) 2015-04-27 2017-10-27 Derivados de hexahidro-[1,4]diazepino[6,7,1-hi]indol-8-carboxamida como agonistas del receptor 5-ht2c y el uso de los mismos en el tratamiento de enfermedades relacionadas con dicho receptor.

Country Status (18)

Country Link
US (1) US10392390B2 (enExample)
EP (1) EP3288946B1 (enExample)
JP (1) JP6675688B2 (enExample)
KR (1) KR102275505B1 (enExample)
CN (1) CN107873030B (enExample)
AU (1) AU2016255009B2 (enExample)
BR (1) BR112017023088B1 (enExample)
CA (1) CA3002544C (enExample)
DK (1) DK3288946T3 (enExample)
EA (1) EA034446B1 (enExample)
ES (1) ES2757922T3 (enExample)
HK (1) HK1244005B (enExample)
HR (1) HRP20192044T1 (enExample)
HU (1) HUE047169T2 (enExample)
IL (1) IL255171A0 (enExample)
MX (2) MX373319B (enExample)
PT (1) PT3288946T (enExample)
WO (1) WO2016176177A1 (enExample)

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US12459965B2 (en) 2017-10-09 2025-11-04 Compass Pathfinder Limited Preparation of psilocybin, different polymorphic forms, intermediates, formulations and their use
GB2571696B (en) 2017-10-09 2020-05-27 Compass Pathways Ltd Large scale method for the preparation of Psilocybin and formulations of Psilocybin so produced
EP3733204A4 (en) 2017-12-27 2021-09-15 Takeda Pharmaceutical Company Limited THERAPEUTIC AGENT FOR URINARY INCONTINENCE OF STRESS AND FECAL INCONTINENCE
CA3089712A1 (en) 2018-01-30 2019-08-08 Apnimed, Inc. (Delaware) Methods and compositions for treating sleep apnea
EP3870292A4 (en) 2018-10-26 2022-11-09 The Research Foundation for The State University of New York COMBINATION OF SEROTONIN-SPECIFIC RESUPPUT INHIBITOR AND SEROTONIN 1A RECEPTOR PARTIAL AGONIST TO REDUCE L-DOPA-INDUCED DYSKINESIA
CA3129270A1 (en) * 2019-02-08 2020-08-13 The Brigham And Women's Hospital, Inc. Methods and compositions for treating sleep apnea
AU2020258086A1 (en) 2019-04-17 2021-11-11 Compass Pathfinder Limited Methods of treating neurocognitive disorders, chronic pain and reducing inflammation
US12205686B2 (en) * 2020-02-27 2025-01-21 The Cleveland Clinic Foundation Identifying patients for intensive hyperglycemia management
US20250073206A1 (en) * 2021-10-29 2025-03-06 Sensorium Therapeutics, Inc. Solid forms of mesembrine and therapeutic uses thereof
CN118679161A (zh) * 2021-12-10 2024-09-20 Gatc健康公司 治疗ptsd和神经障碍的方法
AU2023231581A1 (en) 2022-03-10 2024-09-26 Arena Pharmaceuticals, Inc. Methods of treatment
CN114965250B (zh) * 2022-05-19 2025-02-14 道生天合材料科技(上海)股份有限公司 胶粘剂储存期的预测方法
WO2023225773A1 (en) * 2022-05-23 2023-11-30 Sensorium Therapeutics, Inc. Solid forms of mesembrine and therapeutic uses thereof
AU2023406232A1 (en) * 2022-12-02 2025-05-22 Arena Pharmaceuticals, Inc. Methods of treatment
EP4665319A1 (en) * 2023-02-17 2025-12-24 Caamtech, Inc. 2-(2,5-diethoxy-4-(ethylthio)phenyl)ethane-1-aminium chloride
IL323075A (en) * 2023-03-02 2025-10-01 Alexander Shulgin Res Institute Inc Phenylalkylamine drugs
WO2025080932A1 (en) * 2023-10-11 2025-04-17 University Of Padova Methods of treatment with psilocybin and psilocin derivatives

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US3642822A (en) * 1969-11-03 1972-02-15 Upjohn Co Hexahydropyrrolobenzodiazepines
US4597961A (en) 1985-01-23 1986-07-01 Etscorn Frank T Transcutaneous application of nicotine
US4920989A (en) 1985-04-25 1990-05-01 Regents Of The University Of California Method and apparatus for aiding in the reduction of incidence of tobacco smoking
IL86170A (en) 1987-05-01 1992-12-01 Elan Transdermal Ltd Preparations and compositions comprising nicotine for percutaneous administration
US5004610A (en) 1988-06-14 1991-04-02 Alza Corporation Subsaturated nicotine transdermal therapeutic system
WO1992018005A1 (en) 1991-04-16 1992-10-29 National Institutes Of Health Method of treating trichotillomania and onychophagia
ATE280170T1 (de) * 2000-11-03 2004-11-15 Wyeth Corp Cyclopenta(b)(1,4) diazepino(6,7,1-hi)indole als 5ht2c antagonisten
AU2002227170A1 (en) * 2000-11-03 2002-05-15 Wyeth Cycloalkyl(b)(1,4)diazepino(6,7,1-hi)indoles and derivatives
WO2003086303A2 (en) 2002-04-12 2003-10-23 The University Of Chicago Farnesoid x-activated receptor agonists
TW200307540A (en) * 2002-04-25 2003-12-16 Wyeth Corp [1, 4]Diazocino[7, 8, 1-hi] indole derivatives as antipsychotic and antiobesity agents
CN1805939B (zh) * 2003-06-17 2010-10-13 艾尼纳制药公司 用于治疗5ht2c受体相关病症的苯并氮杂卓衍生物
MX2008012093A (es) * 2006-03-24 2008-10-03 Wyeth Corp Nuevas combinaciones terapeuticas para el tratamiento o la prevencion de trastornos psicoticos.
US9556200B2 (en) * 2012-03-06 2017-01-31 Takeda Pharmaceutical Company Limited Tricyclic compound
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WO2015066344A1 (en) * 2013-11-01 2015-05-07 Arena Pharmaceuticals, Inc. 5-ht2c receptor agonists and compositions and methods of use

Also Published As

Publication number Publication date
EP3288946A1 (en) 2018-03-07
HRP20192044T1 (hr) 2020-02-07
JP2018519251A (ja) 2018-07-19
PT3288946T (pt) 2019-11-27
KR102275505B1 (ko) 2021-07-08
MX2020005898A (es) 2020-08-13
AU2016255009A1 (en) 2017-12-14
IL255171A0 (en) 2017-12-31
HUE047169T2 (hu) 2020-04-28
EA034446B1 (ru) 2020-02-10
CN107873030B (zh) 2021-03-19
DK3288946T3 (da) 2019-11-25
US10392390B2 (en) 2019-08-27
CA3002544A1 (en) 2016-11-03
HK1244005B (en) 2020-04-17
EP3288946B1 (en) 2019-08-21
JP6675688B2 (ja) 2020-04-01
WO2016176177A1 (en) 2016-11-03
BR112017023088B1 (pt) 2023-10-03
MX2017013902A (es) 2018-03-16
EA201792356A1 (ru) 2018-05-31
ES2757922T3 (es) 2020-04-30
NZ737412A (en) 2021-06-25
KR20170140317A (ko) 2017-12-20
US20180186797A1 (en) 2018-07-05
BR112017023088A2 (pt) 2018-07-10
CA3002544C (en) 2024-03-05
CN107873030A (zh) 2018-04-03
AU2016255009B2 (en) 2020-10-08

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