MX2022007436A - Inhibidores de la autotaxina y sus usos. - Google Patents

Inhibidores de la autotaxina y sus usos.

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Publication number
MX2022007436A
MX2022007436A MX2022007436A MX2022007436A MX2022007436A MX 2022007436 A MX2022007436 A MX 2022007436A MX 2022007436 A MX2022007436 A MX 2022007436A MX 2022007436 A MX2022007436 A MX 2022007436A MX 2022007436 A MX2022007436 A MX 2022007436A
Authority
MX
Mexico
Prior art keywords
autotaxin inhibitors
autotaxin
methods
compositions
inhibitors
Prior art date
Application number
MX2022007436A
Other languages
English (en)
Inventor
John Howard Hutchinson
David Lonergan
Gretchen Bain
Jillian Frances Evans
Original Assignee
Sabre Therapeutics Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sabre Therapeutics Llc filed Critical Sabre Therapeutics Llc
Publication of MX2022007436A publication Critical patent/MX2022007436A/es

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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
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    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings

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  • Urology & Nephrology (AREA)
  • Heart & Thoracic Surgery (AREA)
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  • Hematology (AREA)
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  • Ophthalmology & Optometry (AREA)
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Abstract

Aquí se describen métodos y composiciones para el tratamiento de afecciones, enfermedades o trastornos asociados con la actividad de la autotaxina. Los métodos y composiciones descritos en este documento incluyen el uso de al menos un compuesto inhibidor de autotaxina.
MX2022007436A 2015-05-27 2017-11-27 Inhibidores de la autotaxina y sus usos. MX2022007436A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201562167216P 2015-05-27 2015-05-27

Publications (1)

Publication Number Publication Date
MX2022007436A true MX2022007436A (es) 2022-07-19

Family

ID=57393709

Family Applications (2)

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MX2017015225A MX2017015225A (es) 2015-05-27 2016-05-24 Inhibidores de la autotaxina y sus usos.
MX2022007436A MX2022007436A (es) 2015-05-27 2017-11-27 Inhibidores de la autotaxina y sus usos.

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MX2017015225A MX2017015225A (es) 2015-05-27 2016-05-24 Inhibidores de la autotaxina y sus usos.

Country Status (15)

Country Link
US (2) US10632104B2 (es)
EP (2) EP3302490B1 (es)
JP (2) JP6873919B2 (es)
KR (2) KR20240060887A (es)
CN (2) CN107921048A (es)
AU (3) AU2016268250B2 (es)
BR (1) BR122023011445B1 (es)
CA (1) CA2986759A1 (es)
EA (2) EA036337B1 (es)
ES (1) ES2915267T3 (es)
HK (1) HK1253587A1 (es)
IL (2) IL280863B1 (es)
MX (2) MX2017015225A (es)
SG (1) SG10201911204WA (es)
WO (1) WO2016191427A1 (es)

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US10632104B2 (en) 2015-05-27 2020-04-28 Sabre Therapeutics Llc Autotaxin inhibitors and uses thereof
CN107021915A (zh) * 2017-04-27 2017-08-08 李亚庆 一种治疗妇科炎症的化合物及制备方法和应用
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WO2020061114A1 (en) * 2018-09-18 2020-03-26 Metacrine, Inc. Farnesoid x receptor agonists for the treatment of disease
CN112190708B (zh) * 2019-07-08 2023-09-05 上海交通大学医学院附属瑞金医院 趋化因子受体ccr6抑制剂在预防银屑病复发中的新应用
CN114767863B (zh) * 2022-04-29 2024-01-30 西北工业大学 一种enpp2基因或蛋白在调控结直肠癌细胞中的应用
WO2023215196A1 (en) * 2022-05-03 2023-11-09 Sabre Therapeutics Llc Polymorphic and salt forms of the autotaxin inhibitor cudetaxestat
WO2023215684A1 (en) * 2022-05-05 2023-11-09 The Trustees Of Indiana University Therapeutic strategies to manage facial contractures post injury
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