MX2021004710A - Compuestos polimorficos y usos de los mismos. - Google Patents
Compuestos polimorficos y usos de los mismos.Info
- Publication number
- MX2021004710A MX2021004710A MX2021004710A MX2021004710A MX2021004710A MX 2021004710 A MX2021004710 A MX 2021004710A MX 2021004710 A MX2021004710 A MX 2021004710A MX 2021004710 A MX2021004710 A MX 2021004710A MX 2021004710 A MX2021004710 A MX 2021004710A
- Authority
- MX
- Mexico
- Prior art keywords
- polymorphic compounds
- compounds
- polymorphic
- relates
- present
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C225/00—Compounds containing amino groups and doubly—bound oxygen atoms bound to the same carbon skeleton, at least one of the doubly—bound oxygen atoms not being part of a —CHO group, e.g. amino ketones
- C07C225/02—Compounds containing amino groups and doubly—bound oxygen atoms bound to the same carbon skeleton, at least one of the doubly—bound oxygen atoms not being part of a —CHO group, e.g. amino ketones having amino groups bound to acyclic carbon atoms of the carbon skeleton
- C07C225/04—Compounds containing amino groups and doubly—bound oxygen atoms bound to the same carbon skeleton, at least one of the doubly—bound oxygen atoms not being part of a —CHO group, e.g. amino ketones having amino groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being saturated
- C07C225/06—Compounds containing amino groups and doubly—bound oxygen atoms bound to the same carbon skeleton, at least one of the doubly—bound oxygen atoms not being part of a —CHO group, e.g. amino ketones having amino groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being saturated and acyclic
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
- C07C229/02—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
- C07C229/04—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated
- C07C229/06—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one amino and one carboxyl group bound to the carbon skeleton
- C07C229/08—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one amino and one carboxyl group bound to the carbon skeleton the nitrogen atom of the amino group being further bound to hydrogen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K33/00—Medicinal preparations containing inorganic active ingredients
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/13—Crystalline forms, e.g. polymorphs
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Inorganic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Steroid Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201862749922P | 2018-10-24 | 2018-10-24 | |
| PCT/US2019/057815 WO2020086816A1 (en) | 2018-10-24 | 2019-10-24 | Polymorphic compounds and uses thereof |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX2021004710A true MX2021004710A (es) | 2021-06-04 |
Family
ID=70328246
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2021004710A MX2021004710A (es) | 2018-10-24 | 2019-10-24 | Compuestos polimorficos y usos de los mismos. |
| MX2025010903A MX2025010903A (es) | 2018-10-24 | 2021-04-23 | Compuestos polimorficos y usos de los mismos |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2025010903A MX2025010903A (es) | 2018-10-24 | 2021-04-23 | Compuestos polimorficos y usos de los mismos |
Country Status (8)
| Country | Link |
|---|---|
| US (4) | US11345654B2 (https=) |
| EP (1) | EP3870158A4 (https=) |
| JP (2) | JP7644002B2 (https=) |
| CN (1) | CN113164414A (https=) |
| AU (2) | AU2019364542B2 (https=) |
| CA (1) | CA3117336A1 (https=) |
| MX (2) | MX2021004710A (https=) |
| WO (1) | WO2020086816A1 (https=) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2016342027B2 (en) | 2015-10-23 | 2021-05-13 | Navitor Pharmaceuticals, Inc. | Modulators of Sestrin-GATOR2 interaction and uses thereof |
| PL3615019T3 (pl) | 2017-04-26 | 2026-01-19 | Navitor Pharmaceuticals, Inc. | Modulator interakcji sestryna-gator2 do zastosowania w leczeniu depresji opornej na leczenie |
| EP3870158A4 (en) | 2018-10-24 | 2022-08-10 | Navitor Pharmaceuticals, Inc. | Polymorphic compounds and uses thereof |
| US11723890B2 (en) | 2019-11-01 | 2023-08-15 | Navitor Pharmaceuticals, Inc. | Methods of treatment using an mTORC1 modulator |
| CN115927459A (zh) * | 2022-07-19 | 2023-04-07 | 华南农业大学 | 猪ctns基因在促进动物骨骼肌生长中的应用 |
| AU2023374029A1 (en) * | 2022-11-01 | 2025-05-08 | Navitor Pharmaceuticals, Inc. | MODULATORS OF mTORC1 ACTIVITY AND USES THEREOF |
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| RS50352B (sr) | 1999-06-10 | 2009-11-10 | Warner-Lambert Company Llc., | Monosupstituisane 3-propil gama-aminobuterne kiseline |
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| TWI329105B (en) | 2002-02-01 | 2010-08-21 | Rigel Pharmaceuticals Inc | 2,4-pyrimidinediamine compounds and their uses |
| PT1536827E (pt) | 2002-08-14 | 2009-03-20 | Silence Therapeutics Ag | Utilização de proteína cinase n beta |
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| EP1692153A4 (en) | 2003-07-03 | 2007-03-21 | Univ Pennsylvania | INHIBITION OF EXPRESSION OF SYK-KINASE |
| WO2005113556A1 (en) | 2004-05-13 | 2005-12-01 | Icos Corporation | Quinazolinones as inhibitors of human phosphatidylinositol 3-kinase delta |
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| JP2017501113A (ja) * | 2013-10-23 | 2017-01-12 | ホワイトヘッド・インスティテュート・フォー・バイオメディカル・リサーチ | アミノ酸によるｍＴＯＲＣ１の調節およびその使用 |
| CA2976106A1 (en) * | 2015-02-12 | 2016-08-18 | The Arizona Board Of Regents On Behalf Of The University Of Arizona | Methods for treating neuroblastoma |
| AU2016342027B2 (en) | 2015-10-23 | 2021-05-13 | Navitor Pharmaceuticals, Inc. | Modulators of Sestrin-GATOR2 interaction and uses thereof |
| US20180327364A1 (en) | 2015-11-13 | 2018-11-15 | Brandeis University | Mtor inhibitors and methods of use thereof |
| EP3445451B1 (en) * | 2016-04-21 | 2021-08-18 | Baylor College of Medicine | Compositions and methods for the treatment of lysosomal storage disorders and disorders characterized by lysosomal dysfunction |
| JP6872768B2 (ja) * | 2016-10-21 | 2021-05-19 | 国立大学法人山口大学 | ｍＴＯＲＣ１活性化抑制剤 |
| PL3615019T3 (pl) | 2017-04-26 | 2026-01-19 | Navitor Pharmaceuticals, Inc. | Modulator interakcji sestryna-gator2 do zastosowania w leczeniu depresji opornej na leczenie |
| KR20250167147A (ko) | 2018-02-08 | 2025-11-28 | 오비드 테라퓨틱스 인크. | 이명, 급성 감각신경성 난청, 메니에르병, 투렛 증후군, 주의력 결핍 과잉행동 장애 및 중독의 치료에 있어서 (1s,3s)-3-아미노-4-(디플루오로메틸리덴) 시클로펜탄-1-카르복시산 및 (s)-3-아미노-4-(디플루오로메틸리덴)시클로펜트-1-엔-1-카르복시산의 용도 |
| EP3870158A4 (en) | 2018-10-24 | 2022-08-10 | Navitor Pharmaceuticals, Inc. | Polymorphic compounds and uses thereof |
| US10926803B2 (en) | 2019-07-17 | 2021-02-23 | GM Global Technology Operations LLC | Four rail front crush structure with load dissemination into eight element support structure |
| US11723890B2 (en) | 2019-11-01 | 2023-08-15 | Navitor Pharmaceuticals, Inc. | Methods of treatment using an mTORC1 modulator |
-
2019
- 2019-10-24 EP EP19874934.3A patent/EP3870158A4/en active Pending
- 2019-10-24 AU AU2019364542A patent/AU2019364542B2/en active Active
- 2019-10-24 US US16/662,517 patent/US11345654B2/en active Active
- 2019-10-24 CN CN201980077762.2A patent/CN113164414A/zh active Pending
- 2019-10-24 WO PCT/US2019/057815 patent/WO2020086816A1/en not_active Ceased
- 2019-10-24 CA CA3117336A patent/CA3117336A1/en active Pending
- 2019-10-24 JP JP2021522528A patent/JP7644002B2/ja active Active
- 2019-10-24 MX MX2021004710A patent/MX2021004710A/es unknown
-
2021
- 2021-04-23 MX MX2025010903A patent/MX2025010903A/es unknown
-
2022
- 2022-05-05 US US17/737,478 patent/US11697633B2/en active Active
-
2023
- 2023-05-30 US US18/203,341 patent/US12252456B2/en active Active
-
2024
- 2024-10-03 JP JP2024174435A patent/JP2025000975A/ja active Pending
-
2025
- 2025-02-14 US US19/053,599 patent/US20250188017A1/en active Pending
- 2025-11-28 AU AU2025271494A patent/AU2025271494A1/en active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| US11697633B2 (en) | 2023-07-11 |
| AU2019364542B2 (en) | 2025-08-28 |
| MX2025010903A (es) | 2025-10-01 |
| US11345654B2 (en) | 2022-05-31 |
| JP2022505849A (ja) | 2022-01-14 |
| US20250188017A1 (en) | 2025-06-12 |
| WO2020086816A1 (en) | 2020-04-30 |
| JP7644002B2 (ja) | 2025-03-11 |
| AU2019364542A1 (en) | 2021-06-10 |
| EP3870158A4 (en) | 2022-08-10 |
| CN113164414A (zh) | 2021-07-23 |
| JP2025000975A (ja) | 2025-01-07 |
| CA3117336A1 (en) | 2020-04-30 |
| AU2025271494A1 (en) | 2026-01-08 |
| US20240018091A1 (en) | 2024-01-18 |
| EP3870158A1 (en) | 2021-09-01 |
| US20200131114A1 (en) | 2020-04-30 |
| US12252456B2 (en) | 2025-03-18 |
| US20220371985A1 (en) | 2022-11-24 |
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