MX2012001290A - Composiciones y metodos para el tratamiento de la enfermedad de parkinson. - Google Patents
Composiciones y metodos para el tratamiento de la enfermedad de parkinson.Info
- Publication number
- MX2012001290A MX2012001290A MX2012001290A MX2012001290A MX2012001290A MX 2012001290 A MX2012001290 A MX 2012001290A MX 2012001290 A MX2012001290 A MX 2012001290A MX 2012001290 A MX2012001290 A MX 2012001290A MX 2012001290 A MX2012001290 A MX 2012001290A
- Authority
- MX
- Mexico
- Prior art keywords
- dopamine
- days
- receptor
- disease
- parkinson
- Prior art date
Links
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4515—Non condensed piperidines, e.g. piperocaine having a butyrophenone group in position 1, e.g. haloperidol
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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- A—HUMAN NECESSITIES
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Landscapes
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- Nutrition Science (AREA)
- Physiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
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| US23026409P | 2009-07-31 | 2009-07-31 | |
| PCT/CA2010/001185 WO2011011886A1 (en) | 2009-07-31 | 2010-07-30 | Compositions and methods for treating parkinson's disease |
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| MX2012001290A true MX2012001290A (es) | 2012-06-12 |
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| Publication number | Priority date | Publication date | Assignee | Title |
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| CA3178035A1 (en) | 2012-12-24 | 2014-07-03 | Neurogastrx, Inc. | Methods for treating gi tract disorders |
| JP6371716B2 (ja) * | 2014-04-01 | 2018-08-08 | 東京エレクトロン株式会社 | 基板液処理装置及び基板液処理方法並びに基板液処理プログラムを記録したコンピュータ読み取り可能な記録媒体 |
| WO2015200369A1 (en) | 2014-06-24 | 2015-12-30 | Neurogastrx, Inc. | Prodrugs of metopimazine |
| US10836757B1 (en) | 2020-04-02 | 2020-11-17 | Neurogastrx, Inc. | Polymorphic forms of metopimazine |
| CN114601928B (zh) * | 2022-04-02 | 2023-03-17 | 首都医科大学 | 一种钙超载介导神经元死亡的标志物及应用 |
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| IT1219667B (it) * | 1988-06-21 | 1990-05-24 | Polifarma Spa | Impiego di uridina nel trattamento farmacologico di disturbi dovuti ad alterato equilibrio dopaminergico |
| RU2057529C1 (ru) * | 1994-05-30 | 1996-04-10 | Алексей Михайлович Коршунов | Способ лечения синдрома паркинсонизма |
| US20010056101A1 (en) * | 1998-06-29 | 2001-12-27 | Carol A. Tamminga | Use of dopamine receptor antagonists in combination with partial dopamine agonist to prevent tolerance in treating nervous disorders related to dopamine dysfunction |
| DE10111486A1 (de) * | 2001-03-09 | 2002-10-02 | Ralph R Dawirs | Verwendung einer oder mehrerer neuroaktiver Substanzen zur Behandlung der Parkinsonschen Krankheit |
| ES2286453T3 (es) * | 2002-09-17 | 2007-12-01 | Motac Neuroscience Limited | Tratamiento de la discinesia. |
| CN1802153A (zh) * | 2002-10-22 | 2006-07-12 | 药物滥用科学研究公司 | 用选择性多巴胺d1受体激动剂治疗认知损害 |
| CA2628298A1 (en) * | 2004-11-03 | 2006-05-11 | Clera Inc. | Method to detect dopamine receptors in the functional d2high state |
| AU2009212065B2 (en) * | 2008-02-05 | 2014-03-20 | Clera Inc. | Compositions and methods for alleviating depression or improving cognition |
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- 2010-07-30 CA CA2769149A patent/CA2769149A1/en not_active Abandoned
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| CA2769149A1 (en) | 2011-02-03 |
| US9192605B2 (en) | 2015-11-24 |
| EP2459194A4 (en) | 2012-12-19 |
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| IL217149A0 (en) | 2012-02-29 |
| AU2010278645A1 (en) | 2012-03-08 |
| CN102548555A (zh) | 2012-07-04 |
| US20120115910A1 (en) | 2012-05-10 |
| JP5756105B2 (ja) | 2015-07-29 |
| BR112012008193A2 (pt) | 2016-03-01 |
| NZ598247A (en) | 2014-01-31 |
| WO2011011886A1 (en) | 2011-02-03 |
| EP2459194A1 (en) | 2012-06-06 |
| KR20120103557A (ko) | 2012-09-19 |
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