MX2012001067A - Procesos para la alquilacion de pirazoles. - Google Patents
Procesos para la alquilacion de pirazoles.Info
- Publication number
- MX2012001067A MX2012001067A MX2012001067A MX2012001067A MX2012001067A MX 2012001067 A MX2012001067 A MX 2012001067A MX 2012001067 A MX2012001067 A MX 2012001067A MX 2012001067 A MX2012001067 A MX 2012001067A MX 2012001067 A MX2012001067 A MX 2012001067A
- Authority
- MX
- Mexico
- Prior art keywords
- sup
- pyrazoles
- alkylation
- processes
- optionally substituted
- Prior art date
Links
- 238000000034 method Methods 0.000 title abstract 2
- 230000029936 alkylation Effects 0.000 title 1
- 238000005804 alkylation reaction Methods 0.000 title 1
- 150000003217 pyrazoles Chemical class 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 2
- 125000004765 (C1-C4) haloalkyl group Chemical group 0.000 abstract 1
- 125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 abstract 1
- 125000001072 heteroaryl group Chemical group 0.000 abstract 1
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 abstract 1
- 125000000547 substituted alkyl group Chemical group 0.000 abstract 1
- 125000003107 substituted aryl group Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Steroid Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US23013409P | 2009-07-31 | 2009-07-31 | |
| US36157010P | 2010-07-06 | 2010-07-06 | |
| PCT/EP2010/060884 WO2011012620A2 (en) | 2009-07-31 | 2010-07-27 | Processes for the alkylation of pyrazoles |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX2012001067A true MX2012001067A (es) | 2012-03-16 |
Family
ID=42782270
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2012001067A MX2012001067A (es) | 2009-07-31 | 2010-07-27 | Procesos para la alquilacion de pirazoles. |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US8563747B2 (enExample) |
| EP (1) | EP2459538B1 (enExample) |
| JP (1) | JP5956334B2 (enExample) |
| CN (1) | CN102471279A (enExample) |
| AR (1) | AR077332A1 (enExample) |
| BR (1) | BR112012008128B8 (enExample) |
| DK (1) | DK2459538T3 (enExample) |
| ES (1) | ES2525489T3 (enExample) |
| IL (1) | IL217387A (enExample) |
| MX (1) | MX2012001067A (enExample) |
| TW (1) | TW201107296A (enExample) |
| WO (1) | WO2011012620A2 (enExample) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN102471278B (zh) | 2009-07-28 | 2015-04-01 | 先正达参股股份有限公司 | 关于吡唑的烷基化方法 |
| CA2806436C (en) * | 2010-08-10 | 2019-09-10 | Syngenta Participations Ag | Process for the preparation of 3-haloalkylpyrazoles |
| JP5140776B1 (ja) * | 2012-09-05 | 2013-02-13 | タマ化学工業株式会社 | １−置換−３−フルオロアルキルピラゾール−４−カルボン酸エステルの製造方法 |
| KR102540220B1 (ko) | 2014-08-19 | 2023-06-02 | 바이엘 애니멀 헬스 게엠베하 | 헥사플루오로프로펜으로부터 5-플루오로-1h-피라졸의 제조 방법 |
| CN119823045B (zh) * | 2024-12-18 | 2025-10-17 | 湖南化工研究院有限公司 | 一种3-二氟甲基-1-甲基吡唑-4-甲酸乙酯的合成方法 |
Family Cites Families (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH0759560B2 (ja) * | 1987-10-19 | 1995-06-28 | 三井東圧化学株式会社 | １，３−ジアルキルピラゾール−４−カルボン酸エステルの製造法 |
| GB9405229D0 (en) * | 1994-03-17 | 1994-04-27 | Rhone Poulenc Agriculture | Compositions of matter |
| US5498624A (en) * | 1995-05-03 | 1996-03-12 | Monsanto Company | Selected pyrazolyl derivatives |
| JP2000044541A (ja) * | 1998-08-03 | 2000-02-15 | Mitsui Chemicals Inc | １，３−ジアルキルピラゾール−４−カルボン酸エステルの製造法 |
| JP4568404B2 (ja) | 2000-05-17 | 2010-10-27 | 三井化学アグロ株式会社 | ピラゾールカルボン酸エステル誘導体の製造法 |
| EP1480955B1 (en) | 2002-03-05 | 2007-06-27 | Syngenta Participations AG | O-cyclopropyl-carboxanilides and their use as fungicides |
| GB0224316D0 (en) | 2002-10-18 | 2002-11-27 | Syngenta Participations Ag | Chemical compounds |
| BRPI0512118A (pt) | 2004-06-18 | 2008-02-06 | Basf Ag | composto, processo para combater fungos nocivos, e, agente fungicida |
| ES2399280T3 (es) * | 2004-10-21 | 2013-03-27 | Syngenta Participations Ag | Procedimiento para la preparación de pirazoles |
| US7863460B2 (en) * | 2005-02-25 | 2011-01-04 | Sagami Chemical Research Center | Process for producing 1-substituted-3-fluoroalkylpyrazole-4-carboxylate |
| EA014297B1 (ru) * | 2005-10-25 | 2010-10-29 | Зингента Партисипейшнс Аг | Гетероциклические амиды, применимые в качестве микробиоцидов |
| GB0526044D0 (en) * | 2005-12-21 | 2006-02-01 | Syngenta Ltd | Novel herbicides |
| WO2008053044A2 (de) * | 2006-11-03 | 2008-05-08 | Basf Se | Hetarylcarbonsäure-n-(biphen-2-yl)amid-verbindungen |
| JP5876209B2 (ja) | 2007-03-16 | 2016-03-02 | シンジェンタ リミテッド | 殺微生物剤の新規な固体形態 |
| ES2395872T3 (es) * | 2007-05-11 | 2013-02-15 | Eli Lilly And Company | 2-[4-(Pirazol-4-ilalquil)piperazin-1-il]-3-fenil pirazinas y piridinas y 3-[4-(pirazol-4-ilalquil)piperazin-1-il]-2-fenil piridinas como antagonistas del receptor de 5-HT7 |
| CA2687176C (en) * | 2007-05-31 | 2015-06-30 | Syngenta Limited | Process for the production of pyrazoles |
| PT2285779E (pt) | 2008-05-08 | 2013-05-22 | Basf Se | Processo para a produção de arilcarboxamidas |
| GB0812028D0 (en) | 2008-07-01 | 2008-08-06 | Syngenta Participations Ag | Fungicidal compositions |
-
2010
- 2010-07-27 MX MX2012001067A patent/MX2012001067A/es not_active Application Discontinuation
- 2010-07-27 AR ARP100102714A patent/AR077332A1/es unknown
- 2010-07-27 WO PCT/EP2010/060884 patent/WO2011012620A2/en not_active Ceased
- 2010-07-27 DK DK10736729.4T patent/DK2459538T3/en active
- 2010-07-27 EP EP10736729.4A patent/EP2459538B1/en active Active
- 2010-07-27 CN CN2010800339701A patent/CN102471279A/zh active Pending
- 2010-07-27 ES ES10736729.4T patent/ES2525489T3/es active Active
- 2010-07-27 BR BR112012008128A patent/BR112012008128B8/pt active IP Right Grant
- 2010-07-27 JP JP2012522152A patent/JP5956334B2/ja active Active
- 2010-07-27 TW TW099124617A patent/TW201107296A/zh unknown
- 2010-07-27 US US13/388,246 patent/US8563747B2/en active Active
-
2012
- 2012-01-05 IL IL217387A patent/IL217387A/en active IP Right Grant
Also Published As
| Publication number | Publication date |
|---|---|
| BR112012008128B8 (pt) | 2019-07-16 |
| CN102471279A (zh) | 2012-05-23 |
| US8563747B2 (en) | 2013-10-22 |
| DK2459538T3 (en) | 2015-01-05 |
| EP2459538B1 (en) | 2014-10-15 |
| IL217387A0 (en) | 2012-02-29 |
| AR077332A1 (es) | 2011-08-17 |
| WO2011012620A2 (en) | 2011-02-03 |
| US20120130085A1 (en) | 2012-05-24 |
| JP5956334B2 (ja) | 2016-07-27 |
| BR112012008128B1 (pt) | 2017-10-31 |
| EP2459538A2 (en) | 2012-06-06 |
| ES2525489T3 (es) | 2014-12-23 |
| WO2011012620A3 (en) | 2011-06-09 |
| JP2013500945A (ja) | 2013-01-10 |
| TW201107296A (en) | 2011-03-01 |
| IL217387A (en) | 2016-02-29 |
| BR112012008128A2 (pt) | 2015-09-22 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA | Abandonment or withdrawal |