IL217387A - Pyrazole alkylation processes - Google Patents
Pyrazole alkylation processesInfo
- Publication number
- IL217387A IL217387A IL217387A IL21738712A IL217387A IL 217387 A IL217387 A IL 217387A IL 217387 A IL217387 A IL 217387A IL 21738712 A IL21738712 A IL 21738712A IL 217387 A IL217387 A IL 217387A
- Authority
- IL
- Israel
- Prior art keywords
- pyrazoles
- alkylation
- processes
- Prior art date
Links
- 230000029936 alkylation Effects 0.000 title 1
- 238000005804 alkylation reaction Methods 0.000 title 1
- 238000000034 method Methods 0.000 title 1
- 150000003217 pyrazoles Chemical class 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Steroid Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US23013409P | 2009-07-31 | 2009-07-31 | |
| US36157010P | 2010-07-06 | 2010-07-06 | |
| PCT/EP2010/060884 WO2011012620A2 (en) | 2009-07-31 | 2010-07-27 | Processes for the alkylation of pyrazoles |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| IL217387A0 IL217387A0 (en) | 2012-02-29 |
| IL217387A true IL217387A (en) | 2016-02-29 |
Family
ID=42782270
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL217387A IL217387A (en) | 2009-07-31 | 2012-01-05 | Pyrazole alkylation processes |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US8563747B2 (enExample) |
| EP (1) | EP2459538B1 (enExample) |
| JP (1) | JP5956334B2 (enExample) |
| CN (1) | CN102471279A (enExample) |
| AR (1) | AR077332A1 (enExample) |
| BR (1) | BR112012008128B8 (enExample) |
| DK (1) | DK2459538T3 (enExample) |
| ES (1) | ES2525489T3 (enExample) |
| IL (1) | IL217387A (enExample) |
| MX (1) | MX2012001067A (enExample) |
| TW (1) | TW201107296A (enExample) |
| WO (1) | WO2011012620A2 (enExample) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MX2012001059A (es) * | 2009-07-28 | 2012-03-14 | Syngenta Participations Ag | Procesos relacionados con la alquilacion de pirazoles. |
| JP5869570B2 (ja) * | 2010-08-10 | 2016-02-24 | シンジェンタ パーティシペーションズ アクチェンゲゼルシャフト | ３−ハロアルキルピラゾールの調製方法 |
| JP5140776B1 (ja) * | 2012-09-05 | 2013-02-13 | タマ化学工業株式会社 | １−置換−３−フルオロアルキルピラゾール−４−カルボン酸エステルの製造方法 |
| JP6676038B2 (ja) * | 2014-08-19 | 2020-04-08 | バイエル・アニマル・ヘルス・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツングＢａｙｅｒ Ａｎｉｍａｌ Ｈｅａｌｔｈ Ｇｍｂｈ | ヘキサフルオロプロペンから出発する５−フルオロ−１ｈ−ピラゾール類の調製のための方法 |
| JP2025523564A (ja) * | 2022-07-11 | 2025-07-23 | エルジー エナジー ソリューション リミテッド | リチウム二次電池用非水電解液及びこれを含むリチウム二次電池 |
| CN119823045B (zh) * | 2024-12-18 | 2025-10-17 | 湖南化工研究院有限公司 | 一种3-二氟甲基-1-甲基吡唑-4-甲酸乙酯的合成方法 |
Family Cites Families (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH0759560B2 (ja) * | 1987-10-19 | 1995-06-28 | 三井東圧化学株式会社 | １，３−ジアルキルピラゾール−４−カルボン酸エステルの製造法 |
| GB9405229D0 (en) * | 1994-03-17 | 1994-04-27 | Rhone Poulenc Agriculture | Compositions of matter |
| US5498624A (en) * | 1995-05-03 | 1996-03-12 | Monsanto Company | Selected pyrazolyl derivatives |
| JP2000044541A (ja) * | 1998-08-03 | 2000-02-15 | Mitsui Chemicals Inc | １，３−ジアルキルピラゾール−４−カルボン酸エステルの製造法 |
| JP4568404B2 (ja) | 2000-05-17 | 2010-10-27 | 三井化学アグロ株式会社 | ピラゾールカルボン酸エステル誘導体の製造法 |
| DK1480955T3 (da) | 2002-03-05 | 2007-10-29 | Syngenta Participations Ag | O-cyclopropyl-carboxanilider og deres anvendelse som fungicider |
| GB0224316D0 (en) | 2002-10-18 | 2002-11-27 | Syngenta Participations Ag | Chemical compounds |
| CN1968934A (zh) * | 2004-06-18 | 2007-05-23 | 巴斯福股份公司 | N－(邻苯基)－1－甲基－3－二氟甲基吡唑－4－甲酰苯胺及其作为杀真菌剂的用途 |
| WO2006045504A1 (en) * | 2004-10-21 | 2006-05-04 | Syngenta Participations Ag | Process for the preparation of pyrazoles |
| JP4114754B2 (ja) * | 2005-02-25 | 2008-07-09 | 財団法人相模中央化学研究所 | １−置換−３−フルオロアルキルピラゾール−４−カルボン酸エステルの製造方法 |
| ES2354374T3 (es) | 2005-10-25 | 2011-03-14 | Syngenta Participations Ag | Derivados de amidas heterocíclicas útiles como microbiocidas. |
| GB0526044D0 (en) | 2005-12-21 | 2006-02-01 | Syngenta Ltd | Novel herbicides |
| WO2008053044A2 (de) * | 2006-11-03 | 2008-05-08 | Basf Se | Hetarylcarbonsäure-n-(biphen-2-yl)amid-verbindungen |
| PT2120577E (pt) | 2007-03-16 | 2014-12-22 | Syngenta Ltd | Nova forma sólida de um microbiocida |
| DK2155717T3 (da) * | 2007-05-11 | 2012-11-19 | Lilly Co Eli | 2-[4-(pyrazol-4-ylalkyl)piperazin-1-yl]-3-phenyl-pyraziner og -pyridiner og 3-[4-(pyrazol-4-ylalkyl)piperazin-1-yl]-2-phenyl-pyridiner som 5-ht7-receptorantagonister |
| CN101679281B (zh) * | 2007-05-31 | 2013-09-11 | 先正达参股股份有限公司 | 吡唑的制备方法 |
| AU2009245791B2 (en) | 2008-05-08 | 2013-05-16 | Basf Se | Method for manufacturing aryl carboxamides |
| GB0812028D0 (en) | 2008-07-01 | 2008-08-06 | Syngenta Participations Ag | Fungicidal compositions |
-
2010
- 2010-07-27 MX MX2012001067A patent/MX2012001067A/es not_active Application Discontinuation
- 2010-07-27 AR ARP100102714A patent/AR077332A1/es unknown
- 2010-07-27 TW TW099124617A patent/TW201107296A/zh unknown
- 2010-07-27 DK DK10736729.4T patent/DK2459538T3/en active
- 2010-07-27 CN CN2010800339701A patent/CN102471279A/zh active Pending
- 2010-07-27 ES ES10736729.4T patent/ES2525489T3/es active Active
- 2010-07-27 WO PCT/EP2010/060884 patent/WO2011012620A2/en not_active Ceased
- 2010-07-27 EP EP10736729.4A patent/EP2459538B1/en active Active
- 2010-07-27 BR BR112012008128A patent/BR112012008128B8/pt active IP Right Grant
- 2010-07-27 US US13/388,246 patent/US8563747B2/en active Active
- 2010-07-27 JP JP2012522152A patent/JP5956334B2/ja active Active
-
2012
- 2012-01-05 IL IL217387A patent/IL217387A/en active IP Right Grant
Also Published As
| Publication number | Publication date |
|---|---|
| EP2459538A2 (en) | 2012-06-06 |
| US20120130085A1 (en) | 2012-05-24 |
| MX2012001067A (es) | 2012-03-16 |
| TW201107296A (en) | 2011-03-01 |
| ES2525489T3 (es) | 2014-12-23 |
| JP5956334B2 (ja) | 2016-07-27 |
| JP2013500945A (ja) | 2013-01-10 |
| WO2011012620A2 (en) | 2011-02-03 |
| BR112012008128B8 (pt) | 2019-07-16 |
| BR112012008128B1 (pt) | 2017-10-31 |
| BR112012008128A2 (pt) | 2015-09-22 |
| CN102471279A (zh) | 2012-05-23 |
| IL217387A0 (en) | 2012-02-29 |
| AR077332A1 (es) | 2011-08-17 |
| EP2459538B1 (en) | 2014-10-15 |
| US8563747B2 (en) | 2013-10-22 |
| DK2459538T3 (en) | 2015-01-05 |
| WO2011012620A3 (en) | 2011-06-09 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FF | Patent granted | ||
| KB | Patent renewed | ||
| KB | Patent renewed |