IL217387A - Pyrazole alkylation processes - Google Patents
Pyrazole alkylation processesInfo
- Publication number
- IL217387A IL217387A IL217387A IL21738712A IL217387A IL 217387 A IL217387 A IL 217387A IL 217387 A IL217387 A IL 217387A IL 21738712 A IL21738712 A IL 21738712A IL 217387 A IL217387 A IL 217387A
- Authority
- IL
- Israel
- Prior art keywords
- pyrazoles
- alkylation
- processes
- Prior art date
Links
- 230000029936 alkylation Effects 0.000 title 1
- 238000005804 alkylation reaction Methods 0.000 title 1
- 238000000034 method Methods 0.000 title 1
- 150000003217 pyrazoles Chemical class 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Steroid Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US23013409P | 2009-07-31 | 2009-07-31 | |
| US36157010P | 2010-07-06 | 2010-07-06 | |
| PCT/EP2010/060884 WO2011012620A2 (en) | 2009-07-31 | 2010-07-27 | Processes for the alkylation of pyrazoles |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| IL217387A0 IL217387A0 (en) | 2012-02-29 |
| IL217387A true IL217387A (en) | 2016-02-29 |
Family
ID=42782270
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL217387A IL217387A (en) | 2009-07-31 | 2012-01-05 | Pyrazole alkylation processes |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US8563747B2 (enExample) |
| EP (1) | EP2459538B1 (enExample) |
| JP (1) | JP5956334B2 (enExample) |
| CN (1) | CN102471279A (enExample) |
| AR (1) | AR077332A1 (enExample) |
| BR (1) | BR112012008128B8 (enExample) |
| DK (1) | DK2459538T3 (enExample) |
| ES (1) | ES2525489T3 (enExample) |
| IL (1) | IL217387A (enExample) |
| MX (1) | MX2012001067A (enExample) |
| TW (1) | TW201107296A (enExample) |
| WO (1) | WO2011012620A2 (enExample) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN102471278B (zh) | 2009-07-28 | 2015-04-01 | 先正达参股股份有限公司 | 关于吡唑的烷基化方法 |
| CA2806436C (en) * | 2010-08-10 | 2019-09-10 | Syngenta Participations Ag | Process for the preparation of 3-haloalkylpyrazoles |
| JP5140776B1 (ja) * | 2012-09-05 | 2013-02-13 | タマ化学工業株式会社 | １−置換−３−フルオロアルキルピラゾール−４−カルボン酸エステルの製造方法 |
| ES2750353T3 (es) | 2014-08-19 | 2020-03-25 | Bayer Animal Health Gmbh | Procedimiento de preparación de 5-fluoro-1H-pirazoles partiendo de hexafluoropropeno |
| JP7885371B2 (ja) * | 2022-07-11 | 2026-07-06 | エルジー エナジー ソリューション リミテッド | リチウム二次電池用非水電解液及びこれを含むリチウム二次電池 |
| CN119823045B (zh) * | 2024-12-18 | 2025-10-17 | 湖南化工研究院有限公司 | 一种3-二氟甲基-1-甲基吡唑-4-甲酸乙酯的合成方法 |
Family Cites Families (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH0759560B2 (ja) * | 1987-10-19 | 1995-06-28 | 三井東圧化学株式会社 | １，３−ジアルキルピラゾール−４−カルボン酸エステルの製造法 |
| GB9405229D0 (en) * | 1994-03-17 | 1994-04-27 | Rhone Poulenc Agriculture | Compositions of matter |
| US5498624A (en) * | 1995-05-03 | 1996-03-12 | Monsanto Company | Selected pyrazolyl derivatives |
| JP2000044541A (ja) | 1998-08-03 | 2000-02-15 | Mitsui Chemicals Inc | １，３−ジアルキルピラゾール−４−カルボン酸エステルの製造法 |
| JP4568404B2 (ja) | 2000-05-17 | 2010-10-27 | 三井化学アグロ株式会社 | ピラゾールカルボン酸エステル誘導体の製造法 |
| HK1079785B (zh) | 2002-03-05 | 2007-08-10 | 辛根塔参与股份公司 | 邻环丙基-n-甲酰苯胺及其作为杀菌剂的用途 |
| GB0224316D0 (en) | 2002-10-18 | 2002-11-27 | Syngenta Participations Ag | Chemical compounds |
| JP2008502636A (ja) * | 2004-06-18 | 2008-01-31 | ビーエーエスエフ アクチェンゲゼルシャフト | Ｎ−（オルト−フェニル）−１−メチル−３−ジフルオロメチルピラゾール−４−カルボキシアニリドおよびそれらの殺菌剤としての使用 |
| EA010851B1 (ru) * | 2004-10-21 | 2008-12-30 | Зингента Партисипейшнс Аг | Способ получения пиразолов |
| US7863460B2 (en) * | 2005-02-25 | 2011-01-04 | Sagami Chemical Research Center | Process for producing 1-substituted-3-fluoroalkylpyrazole-4-carboxylate |
| ATE489372T1 (de) | 2005-10-25 | 2010-12-15 | Syngenta Participations Ag | Als mikrobiozide geeignete heterocyclische amidderivate |
| GB0526044D0 (en) * | 2005-12-21 | 2006-02-01 | Syngenta Ltd | Novel herbicides |
| WO2008053044A2 (de) * | 2006-11-03 | 2008-05-08 | Basf Se | Hetarylcarbonsäure-n-(biphen-2-yl)amid-verbindungen |
| US8580835B2 (en) | 2007-03-16 | 2013-11-12 | Syngenta Crop Protection, Llc | Solid forms of a microbiocide |
| BRPI0811446A2 (pt) * | 2007-05-11 | 2014-10-29 | Lilly Co Eli | " 2-[4-(pirazol-4-ilalquil)piperazin-1-il]-3-fenil pirazinas e piridinas e 3-[4-(pirazol-4-ilalquil)piperazin-1-il]-2-fenil piridinas como antagonistas de receptor 5-ht7" |
| WO2008145257A1 (en) | 2007-05-31 | 2008-12-04 | Syngenta Participations Ag | Process for the production of pyrazoles |
| KR20110004903A (ko) | 2008-05-08 | 2011-01-14 | 바스프 에스이 | 아릴카르복스아미드의 제조 방법 |
| GB0812028D0 (en) | 2008-07-01 | 2008-08-06 | Syngenta Participations Ag | Fungicidal compositions |
-
2010
- 2010-07-27 WO PCT/EP2010/060884 patent/WO2011012620A2/en not_active Ceased
- 2010-07-27 AR ARP100102714A patent/AR077332A1/es unknown
- 2010-07-27 BR BR112012008128A patent/BR112012008128B8/pt active IP Right Grant
- 2010-07-27 MX MX2012001067A patent/MX2012001067A/es not_active Application Discontinuation
- 2010-07-27 CN CN2010800339701A patent/CN102471279A/zh active Pending
- 2010-07-27 EP EP10736729.4A patent/EP2459538B1/en active Active
- 2010-07-27 JP JP2012522152A patent/JP5956334B2/ja active Active
- 2010-07-27 ES ES10736729.4T patent/ES2525489T3/es active Active
- 2010-07-27 TW TW099124617A patent/TW201107296A/zh unknown
- 2010-07-27 US US13/388,246 patent/US8563747B2/en active Active
- 2010-07-27 DK DK10736729.4T patent/DK2459538T3/en active
-
2012
- 2012-01-05 IL IL217387A patent/IL217387A/en active IP Right Grant
Also Published As
| Publication number | Publication date |
|---|---|
| JP2013500945A (ja) | 2013-01-10 |
| WO2011012620A3 (en) | 2011-06-09 |
| ES2525489T3 (es) | 2014-12-23 |
| TW201107296A (en) | 2011-03-01 |
| CN102471279A (zh) | 2012-05-23 |
| IL217387A0 (en) | 2012-02-29 |
| MX2012001067A (es) | 2012-03-16 |
| EP2459538A2 (en) | 2012-06-06 |
| US8563747B2 (en) | 2013-10-22 |
| WO2011012620A2 (en) | 2011-02-03 |
| BR112012008128B1 (pt) | 2017-10-31 |
| EP2459538B1 (en) | 2014-10-15 |
| DK2459538T3 (en) | 2015-01-05 |
| US20120130085A1 (en) | 2012-05-24 |
| AR077332A1 (es) | 2011-08-17 |
| BR112012008128B8 (pt) | 2019-07-16 |
| JP5956334B2 (ja) | 2016-07-27 |
| BR112012008128A2 (pt) | 2015-09-22 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| IL202664A0 (en) | Processes for the preparation of pyrazoles | |
| EP2435390A4 (en) | TRANSALCYLATION OF POLYCYCLOHEXYLBENZENES | |
| IL214184A0 (en) | Fungicidal pyrazoles | |
| ZA201202504B (en) | Process for the preparation of calcobutrol | |
| IL211701A0 (en) | Process for the preparation of bendamustine | |
| EP2464650A4 (en) | PROCESSES FOR PREPARING PEMETREXED | |
| IL215846A0 (en) | Method for the manufacture of degarelix | |
| PL2398808T3 (pl) | Sposób redukcyjnego alkilowania normorfinanów | |
| SI2516958T1 (sl) | Vžigalnik za ročno granato | |
| PL390042A1 (pl) | Sposób wytwarzania kwasu chlebowego | |
| ZA201202343B (en) | Process for the preparation of lenalidomide | |
| IL216942A0 (en) | Process for the manufacture of alkenones | |
| ZA201107111B (en) | Process for the preparation of layered silicates | |
| IL217387A0 (en) | Processes for the alkylation of pyrazoles | |
| ZA201104932B (en) | Phenylimidazole compounds | |
| GB0908435D0 (en) | Processes | |
| ZA201107435B (en) | Pyrazole copmpound | |
| IL221184A (en) | A process for preparing 1-alkylated tetrazole 5 is produced | |
| PL2443094T3 (pl) | Sposób wytwarzania telmisartanu | |
| PL2275467T3 (pl) | Prepolimery NCO ze związków zakończonych formamidem | |
| ZA201201657B (en) | Processes for the preparation of vardenafil | |
| IL217525A0 (en) | Processes relating to the alkylation of pyrazoles | |
| GB0919489D0 (en) | Pinsticks | |
| GB0904311D0 (en) | Processes for the preparation of compounds | |
| IL220160A (en) | A process for the preparation of defrasirox |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FF | Patent granted | ||
| KB | Patent renewed | ||
| KB | Patent renewed |