JP5956334B2 - ピラゾールのアルキル化のためのプロセス - Google Patents
ピラゾールのアルキル化のためのプロセス Download PDFInfo
- Publication number
- JP5956334B2 JP5956334B2 JP2012522152A JP2012522152A JP5956334B2 JP 5956334 B2 JP5956334 B2 JP 5956334B2 JP 2012522152 A JP2012522152 A JP 2012522152A JP 2012522152 A JP2012522152 A JP 2012522152A JP 5956334 B2 JP5956334 B2 JP 5956334B2
- Authority
- JP
- Japan
- Prior art keywords
- formula
- compound
- optionally substituted
- alkyl
- methyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Active
Links
- 0 Cc1n[n]cc1C(O*)=O Chemical compound Cc1n[n]cc1C(O*)=O 0.000 description 2
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Steroid Compounds (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US23013409P | 2009-07-31 | 2009-07-31 | |
| US36157010P | 2010-07-06 | 2010-07-06 | |
| US61/361,570 | 2010-07-06 | ||
| US61/230,134 | 2010-07-06 | ||
| PCT/EP2010/060884 WO2011012620A2 (en) | 2009-07-31 | 2010-07-27 | Processes for the alkylation of pyrazoles |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2013500945A JP2013500945A (ja) | 2013-01-10 |
| JP2013500945A5 JP2013500945A5 (enExample) | 2015-12-17 |
| JP5956334B2 true JP5956334B2 (ja) | 2016-07-27 |
Family
ID=42782270
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2012522152A Active JP5956334B2 (ja) | 2009-07-31 | 2010-07-27 | ピラゾールのアルキル化のためのプロセス |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US8563747B2 (enExample) |
| EP (1) | EP2459538B1 (enExample) |
| JP (1) | JP5956334B2 (enExample) |
| CN (1) | CN102471279A (enExample) |
| AR (1) | AR077332A1 (enExample) |
| BR (1) | BR112012008128B8 (enExample) |
| DK (1) | DK2459538T3 (enExample) |
| ES (1) | ES2525489T3 (enExample) |
| IL (1) | IL217387A (enExample) |
| MX (1) | MX2012001067A (enExample) |
| TW (1) | TW201107296A (enExample) |
| WO (1) | WO2011012620A2 (enExample) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP5763634B2 (ja) | 2009-07-28 | 2015-08-12 | シンジェンタ パーティシペーションズ アクチェンゲゼルシャフト | ピラゾールのアルキル化に関する方法 |
| PT2603494T (pt) * | 2010-08-10 | 2017-02-03 | Syngenta Participations Ag | Processo para a preparação de 3-haloalquilopirazóis |
| JP5140776B1 (ja) * | 2012-09-05 | 2013-02-13 | タマ化学工業株式会社 | １−置換−３−フルオロアルキルピラゾール−４−カルボン酸エステルの製造方法 |
| KR102540220B1 (ko) * | 2014-08-19 | 2023-06-02 | 바이엘 애니멀 헬스 게엠베하 | 헥사플루오로프로펜으로부터 5-플루오로-1h-피라졸의 제조 방법 |
| CN119823045B (zh) * | 2024-12-18 | 2025-10-17 | 湖南化工研究院有限公司 | 一种3-二氟甲基-1-甲基吡唑-4-甲酸乙酯的合成方法 |
Family Cites Families (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH0759560B2 (ja) * | 1987-10-19 | 1995-06-28 | 三井東圧化学株式会社 | １，３−ジアルキルピラゾール−４−カルボン酸エステルの製造法 |
| GB9405229D0 (en) * | 1994-03-17 | 1994-04-27 | Rhone Poulenc Agriculture | Compositions of matter |
| US5498624A (en) * | 1995-05-03 | 1996-03-12 | Monsanto Company | Selected pyrazolyl derivatives |
| JP2000044541A (ja) * | 1998-08-03 | 2000-02-15 | Mitsui Chemicals Inc | １，３−ジアルキルピラゾール−４−カルボン酸エステルの製造法 |
| JP4568404B2 (ja) | 2000-05-17 | 2010-10-27 | 三井化学アグロ株式会社 | ピラゾールカルボン酸エステル誘導体の製造法 |
| DK1480955T3 (da) | 2002-03-05 | 2007-10-29 | Syngenta Participations Ag | O-cyclopropyl-carboxanilider og deres anvendelse som fungicider |
| GB0224316D0 (en) | 2002-10-18 | 2002-11-27 | Syngenta Participations Ag | Chemical compounds |
| BRPI0512118A (pt) * | 2004-06-18 | 2008-02-06 | Basf Ag | composto, processo para combater fungos nocivos, e, agente fungicida |
| TWI357898B (en) * | 2004-10-21 | 2012-02-11 | Syngenta Participations Ag | Process for the preparation of pyrazoles |
| US7863460B2 (en) * | 2005-02-25 | 2011-01-04 | Sagami Chemical Research Center | Process for producing 1-substituted-3-fluoroalkylpyrazole-4-carboxylate |
| GEP20115161B (en) | 2005-10-25 | 2011-02-10 | Syngenta Participations Ag | Heterocyclic amide derivatives useful as microbiocides |
| GB0526044D0 (en) | 2005-12-21 | 2006-02-01 | Syngenta Ltd | Novel herbicides |
| WO2008053044A2 (de) * | 2006-11-03 | 2008-05-08 | Basf Se | Hetarylcarbonsäure-n-(biphen-2-yl)amid-verbindungen |
| DK2120577T3 (en) | 2007-03-16 | 2014-12-15 | Syngenta Ltd | NOVEL SOLID FORM OF A microbicide |
| WO2008141020A1 (en) | 2007-05-11 | 2008-11-20 | Eli Lilly And Company | 2-[4-(pyrazol-4-ylalkyl)piperazin-1-yl]-3-phenyl pyrazines and pyridines and 3-[4-(pyrazol-4-ylalkyl)piperazin-1-yl]-2-phenyl pyridines as 5-ht7 receptor antagonists |
| RU2459807C2 (ru) * | 2007-05-31 | 2012-08-27 | Зингента Партисипейшнс Аг | Способ получения пиразолов |
| KR20110004903A (ko) | 2008-05-08 | 2011-01-14 | 바스프 에스이 | 아릴카르복스아미드의 제조 방법 |
| GB0812028D0 (en) | 2008-07-01 | 2008-08-06 | Syngenta Participations Ag | Fungicidal compositions |
-
2010
- 2010-07-27 CN CN2010800339701A patent/CN102471279A/zh active Pending
- 2010-07-27 US US13/388,246 patent/US8563747B2/en active Active
- 2010-07-27 DK DK10736729.4T patent/DK2459538T3/en active
- 2010-07-27 MX MX2012001067A patent/MX2012001067A/es not_active Application Discontinuation
- 2010-07-27 ES ES10736729.4T patent/ES2525489T3/es active Active
- 2010-07-27 AR ARP100102714A patent/AR077332A1/es unknown
- 2010-07-27 JP JP2012522152A patent/JP5956334B2/ja active Active
- 2010-07-27 TW TW099124617A patent/TW201107296A/zh unknown
- 2010-07-27 BR BR112012008128A patent/BR112012008128B8/pt active IP Right Grant
- 2010-07-27 EP EP10736729.4A patent/EP2459538B1/en active Active
- 2010-07-27 WO PCT/EP2010/060884 patent/WO2011012620A2/en not_active Ceased
-
2012
- 2012-01-05 IL IL217387A patent/IL217387A/en active IP Right Grant
Also Published As
| Publication number | Publication date |
|---|---|
| TW201107296A (en) | 2011-03-01 |
| ES2525489T3 (es) | 2014-12-23 |
| WO2011012620A2 (en) | 2011-02-03 |
| JP2013500945A (ja) | 2013-01-10 |
| US8563747B2 (en) | 2013-10-22 |
| CN102471279A (zh) | 2012-05-23 |
| BR112012008128B8 (pt) | 2019-07-16 |
| DK2459538T3 (en) | 2015-01-05 |
| EP2459538B1 (en) | 2014-10-15 |
| IL217387A0 (en) | 2012-02-29 |
| BR112012008128A2 (pt) | 2015-09-22 |
| US20120130085A1 (en) | 2012-05-24 |
| EP2459538A2 (en) | 2012-06-06 |
| IL217387A (en) | 2016-02-29 |
| MX2012001067A (es) | 2012-03-16 |
| WO2011012620A3 (en) | 2011-06-09 |
| AR077332A1 (es) | 2011-08-17 |
| BR112012008128B1 (pt) | 2017-10-31 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| JP5956334B2 (ja) | ピラゾールのアルキル化のためのプロセス | |
| US20180208559A1 (en) | Process for the preparation of 3-haloalkylpyrazoles | |
| AU703688B2 (en) | Process for producing 3,5-diaryl pyrazolene | |
| JP5763634B2 (ja) | ピラゾールのアルキル化に関する方法 | |
| BR112013004066B1 (pt) | Processo para a preparação de 3-haloalquilapirazóis |
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