MX2011008885A - Composiciones, sintesis y metodos para usar derivados de arilpiperazina. - Google Patents

Composiciones, sintesis y metodos para usar derivados de arilpiperazina.

Info

Publication number
MX2011008885A
MX2011008885A MX2011008885A MX2011008885A MX2011008885A MX 2011008885 A MX2011008885 A MX 2011008885A MX 2011008885 A MX2011008885 A MX 2011008885A MX 2011008885 A MX2011008885 A MX 2011008885A MX 2011008885 A MX2011008885 A MX 2011008885A
Authority
MX
Mexico
Prior art keywords
methods
arylpiperazine derivatives
synthesis
compositions
polypeptides
Prior art date
Application number
MX2011008885A
Other languages
English (en)
Inventor
Prabhu Prasad Mohapatra
Laxminarayan Bhat
Kouacou Adiey
Original Assignee
Reviva Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Reviva Pharmaceuticals Inc filed Critical Reviva Pharmaceuticals Inc
Publication of MX2011008885A publication Critical patent/MX2011008885A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/28—1,4-Oxazines; Hydrogenated 1,4-oxazines
    • C07D265/34—1,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings
    • C07D265/36—1,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings condensed with one six-membered ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4965—Non-condensed pyrazines
    • A61K31/497—Non-condensed pyrazines containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/538—1,4-Oxazines, e.g. morpholine ortho- or peri-condensed with carbocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Immobilizing And Processing Of Enzymes And Microorganisms (AREA)
  • Enzymes And Modification Thereof (AREA)

Abstract

La presente invención provee derivados de arilpiperazina que pueden usarse ventajosamente para tratar esquizofrenia y psicosis relacionada tal corno trastorno maniaco agudo, trastorne bipolar, trastorno autista y depresión.
MX2011008885A 2009-02-26 2010-02-26 Composiciones, sintesis y metodos para usar derivados de arilpiperazina. MX2011008885A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US15579109P 2009-02-26 2009-02-26
PCT/US2010/025687 WO2010099502A1 (en) 2009-02-26 2010-02-26 Compositions, synthesis, and methods of utilizing arylpiperazine derivatives

Publications (1)

Publication Number Publication Date
MX2011008885A true MX2011008885A (es) 2011-09-29

Family

ID=42631516

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2011008885A MX2011008885A (es) 2009-02-26 2010-02-26 Composiciones, sintesis y metodos para usar derivados de arilpiperazina.

Country Status (25)

Country Link
US (9) US8575185B2 (es)
EP (1) EP2400968B1 (es)
JP (1) JP5337259B2 (es)
KR (1) KR101705727B1 (es)
CN (2) CN106045936A (es)
AU (1) AU2010217772B2 (es)
BR (1) BRPI1009757B1 (es)
CA (1) CA2753599C (es)
CO (1) CO6430428A2 (es)
DK (1) DK2400968T3 (es)
ES (1) ES2605232T3 (es)
HK (1) HK1167240A1 (es)
HU (1) HUE031053T2 (es)
IL (1) IL214754A (es)
MX (1) MX2011008885A (es)
MY (1) MY161473A (es)
NZ (1) NZ595263A (es)
PH (1) PH12011501669B1 (es)
PL (1) PL2400968T3 (es)
PT (1) PT2400968T (es)
RU (1) RU2506262C2 (es)
SG (1) SG173842A1 (es)
UA (1) UA102730C2 (es)
WO (2) WO2010099502A1 (es)
ZA (1) ZA201106805B (es)

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* Cited by examiner, † Cited by third party
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WO2010099502A1 (en) 2009-02-26 2010-09-02 Reviva Pharmaceuticals, Inc. Compositions, synthesis, and methods of utilizing arylpiperazine derivatives
KR101571670B1 (ko) * 2012-08-08 2015-11-25 주식회사 씨엠지제약 아리피프라졸을 포함하는 경구용 속용 필름 제제
WO2015157451A1 (en) 2014-04-08 2015-10-15 Reviva Pharmaceuticals, Inc. Methods for treating attention deficit hyperactivity disorder
CN107206007B (zh) * 2015-01-12 2021-08-10 雷维瓦药品公司 用于治疗肺高血压的方法
WO2016115150A1 (en) * 2015-01-12 2016-07-21 Reviva Pharmaceuticals Inc. Methods for treating psychosis associated with parkinson's disease
WO2016115144A1 (en) 2015-01-12 2016-07-21 Reviva Pharmaceuticals Inc. Methods for treating alzheimer's disease
GB201508864D0 (en) * 2015-05-22 2015-07-01 Glaxosmithkline Ip Dev Ltd Compounds
WO2017042837A2 (en) * 2015-09-11 2017-03-16 Sun Pharmaceutical Industries Limited Stable crystalline form of regadenoson
CN113912586B (zh) 2016-08-31 2023-04-07 江苏恒瑞医药股份有限公司 氧代吡啶酰胺类衍生物、其制备方法及其在医药上的应用
CN112618580A (zh) * 2020-12-30 2021-04-09 北京科拓恒通生物技术股份有限公司 鼠李糖乳杆菌Probio-M9及其制品用于制备治疗自闭症药物的用途

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Also Published As

Publication number Publication date
NZ595263A (en) 2013-06-28
US20150005298A1 (en) 2015-01-01
US8431570B2 (en) 2013-04-30
US20100216783A1 (en) 2010-08-26
US20160229821A1 (en) 2016-08-11
US8188076B2 (en) 2012-05-29
EP2400968B1 (en) 2016-09-28
BRPI1009757A2 (pt) 2016-03-15
EP2400968A1 (en) 2012-01-04
EP2400968A4 (en) 2012-08-01
US8461154B2 (en) 2013-06-11
US8575185B2 (en) 2013-11-05
ES2605232T3 (es) 2017-03-13
AU2010217772A1 (en) 2011-10-20
US20150166493A1 (en) 2015-06-18
US8859552B2 (en) 2014-10-14
PT2400968T (pt) 2016-12-09
RU2506262C2 (ru) 2014-02-10
IL214754A0 (en) 2011-11-30
US9975862B2 (en) 2018-05-22
IL214754A (en) 2014-05-28
BRPI1009757B1 (pt) 2020-01-14
HUE031053T2 (en) 2017-06-28
US20100222359A1 (en) 2010-09-02
JP5337259B2 (ja) 2013-11-06
CN102413830A (zh) 2012-04-11
DK2400968T3 (da) 2017-01-02
PH12011501669B1 (en) 2014-02-13
HK1167240A1 (zh) 2012-11-23
KR20120013306A (ko) 2012-02-14
CA2753599C (en) 2017-03-14
KR101705727B1 (ko) 2017-02-10
AU2010217772B2 (en) 2014-10-23
CA2753599A1 (en) 2010-09-02
JP2012519182A (ja) 2012-08-23
WO2010099503A1 (en) 2010-09-02
US20120220574A1 (en) 2012-08-30
US9604944B2 (en) 2017-03-28
US8980883B2 (en) 2015-03-17
WO2010099502A1 (en) 2010-09-02
US20140155392A1 (en) 2014-06-05
MY161473A (en) 2017-04-14
US20120220579A1 (en) 2012-08-30
RU2011139154A (ru) 2013-04-10
ZA201106805B (en) 2013-02-27
UA102730C2 (uk) 2013-08-12
PL2400968T3 (pl) 2017-04-28
CN106045936A (zh) 2016-10-26
SG173842A1 (en) 2011-09-29
US20170327477A1 (en) 2017-11-16
CO6430428A2 (es) 2012-04-30
US9255076B2 (en) 2016-02-09

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