MX342947B - Tratamiento de diabetes tipo 2. - Google Patents

Tratamiento de diabetes tipo 2.

Info

Publication number
MX342947B
MX342947B MX2012014334A MX2012014334A MX342947B MX 342947 B MX342947 B MX 342947B MX 2012014334 A MX2012014334 A MX 2012014334A MX 2012014334 A MX2012014334 A MX 2012014334A MX 342947 B MX342947 B MX 342947B
Authority
MX
Mexico
Prior art keywords
diabetes
treatment
type
triazine derivatives
formule
Prior art date
Application number
MX2012014334A
Other languages
English (en)
Other versions
MX2012014334A (es
Inventor
Cravo Daniel
Fouqueray Pascale
Hallakou-Bozec Sophie
Bolze Sébastien
Original Assignee
Poxel *
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Poxel * filed Critical Poxel *
Publication of MX2012014334A publication Critical patent/MX2012014334A/es
Publication of MX342947B publication Critical patent/MX342947B/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D251/00Heterocyclic compounds containing 1,3,5-triazine rings
    • C07D251/02Heterocyclic compounds containing 1,3,5-triazine rings not condensed with other rings
    • C07D251/10Heterocyclic compounds containing 1,3,5-triazine rings not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/53Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with three nitrogens as the only ring hetero atoms, e.g. chlorazanil, melamine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/2027Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Diabetes (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Endocrinology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Emergency Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Steroid Compounds (AREA)

Abstract

La presente invención se refiere a derivados de triazina para su uso en el tratamiento de diabetes tipo 2, y a composiciones que comprenden los derivados de triazina.
MX2012014334A 2010-06-09 2011-06-09 Tratamiento de diabetes tipo 2. MX342947B (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP10305612 2010-06-09
PCT/EP2011/059590 WO2011154497A1 (en) 2010-06-09 2011-06-09 Treatment of type 2 diabetes

Publications (2)

Publication Number Publication Date
MX2012014334A MX2012014334A (es) 2013-01-29
MX342947B true MX342947B (es) 2016-10-18

Family

ID=42938387

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2012014334A MX342947B (es) 2010-06-09 2011-06-09 Tratamiento de diabetes tipo 2.

Country Status (14)

Country Link
US (1) US20130131065A1 (es)
EP (2) EP2579880B1 (es)
JP (1) JP5707490B2 (es)
KR (1) KR101548217B1 (es)
CN (1) CN102933215A (es)
AU (1) AU2011263730B2 (es)
BR (1) BR112012030482A2 (es)
CA (1) CA2800428C (es)
EA (1) EA201201623A1 (es)
ES (1) ES2753976T3 (es)
IL (1) IL223289A (es)
MX (1) MX342947B (es)
TW (1) TWI436768B (es)
WO (1) WO2011154497A1 (es)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP5707489B2 (ja) * 2010-06-09 2015-04-30 ポクセル・エスアーエスPoxelsas 1型糖尿病の処置
US11759441B2 (en) 2011-01-07 2023-09-19 Anji Pharmaceuticals Inc. Biguanide compositions and methods of treating metabolic disorders
US11974971B2 (en) 2011-01-07 2024-05-07 Anji Pharmaceuticals Inc. Compositions and methods for treating metabolic disorders
US9211263B2 (en) 2012-01-06 2015-12-15 Elcelyx Therapeutics, Inc. Compositions and methods of treating metabolic disorders
LT2661266T (lt) 2011-01-07 2020-12-10 Anji Pharma (Us) Llc Gydimo būdai chemosensorinio receptoriaus ligando pagrindu
CN104254325A (zh) 2012-01-06 2014-12-31 埃尔舍利克斯治疗公司 双胍组合物和治疗代谢性病症的方法
CN110693867A (zh) * 2012-01-06 2020-01-17 埃尔舍利克斯治疗公司 用于治疗代谢性病症的组合物和方法
CN111163782A (zh) * 2017-10-02 2020-05-15 普克塞尔公司 治疗射血分数保留型心力衰竭的方法
SG11202007172YA (en) * 2018-06-06 2020-08-28 Metavant Sciences Gmbh Methods of treating subjects having diabetes with chronic kidney disease
CA3103324A1 (en) * 2018-06-14 2019-12-19 Poxel Film-coated tablet comprising a triazine derivative for use in the treatment of diabetes
KR20220113942A (ko) 2019-12-13 2022-08-17 스미토모 파마 가부시키가이샤 제조성 및 용출성이 우수한 소형 정제

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2804113B1 (fr) 2000-01-26 2004-06-18 Lipha Derives animes de dihydro-1,3,5-triazine et leurs applications en therapeutique
FR2853650B1 (fr) * 2003-04-10 2006-07-07 Merck Sante Sas Procede de dedoublement d'amines utiles pour le traitement de desordres associes au syndrome d'insulino-resistance
FR2896159B1 (fr) * 2006-01-13 2008-09-12 Merck Sante Soc Par Actions Si Combinaison de derives de triazine et d'agents sensibilisateurs a l'insuline.
KR101085157B1 (ko) * 2007-08-31 2011-11-18 한국화학연구원 1,3,5-트리아진-2,4,6-트리아민 화합물 또는 그의 약학적으로 허용 가능한 염, 및 이를 포함하는 약학적 조성물
DE102007054416A1 (de) * 2007-11-13 2009-05-14 Studiengesellschaft Kohle Mbh Verfahren zur Herstellung von 3,6-Dihydro-1,3,5- Triazin-Derivaten für die Behandlungen von Erkrankungen, die mit dem Insulinresistenz-Syndrom assoziiert sind
SG171986A1 (en) * 2008-12-12 2011-07-28 Merck Patent Gmbh Combination of insulin with triazine derivatives and its use for treating diabetes
JP5707489B2 (ja) * 2010-06-09 2015-04-30 ポクセル・エスアーエスPoxelsas 1型糖尿病の処置

Also Published As

Publication number Publication date
AU2011263730B2 (en) 2014-07-03
ES2753976T3 (es) 2020-04-15
IL223289A (en) 2017-07-31
KR20130083895A (ko) 2013-07-23
KR101548217B1 (ko) 2015-08-28
IL223289A0 (en) 2013-02-03
AU2011263730A1 (en) 2013-01-10
BR112012030482A2 (pt) 2016-08-09
MX2012014334A (es) 2013-01-29
TW201206443A (en) 2012-02-16
EA201201623A1 (ru) 2013-05-30
CN102933215A (zh) 2013-02-13
US20130131065A1 (en) 2013-05-23
EP2579880B1 (en) 2019-09-11
JP5707490B2 (ja) 2015-04-30
WO2011154497A1 (en) 2011-12-15
EP3597194A1 (en) 2020-01-22
CA2800428A1 (en) 2011-12-15
CA2800428C (en) 2014-08-26
JP2013531646A (ja) 2013-08-08
EP2579880A1 (en) 2013-04-17
TWI436768B (zh) 2014-05-11

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