MX2009011139A - Ligandos de receptor vainilloide novedosos y el uso de los mismos para la produccion de farmacos. - Google Patents

Ligandos de receptor vainilloide novedosos y el uso de los mismos para la produccion de farmacos.

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Publication number
MX2009011139A
MX2009011139A MX2009011139A MX2009011139A MX2009011139A MX 2009011139 A MX2009011139 A MX 2009011139A MX 2009011139 A MX2009011139 A MX 2009011139A MX 2009011139 A MX2009011139 A MX 2009011139A MX 2009011139 A MX2009011139 A MX 2009011139A
Authority
MX
Mexico
Prior art keywords
production
pharmaceuticals
receptor ligands
vanilloid receptor
novel vanilloid
Prior art date
Application number
MX2009011139A
Other languages
English (en)
Spanish (es)
Inventor
Bernd Sundermann
Derek Saunders
Klaus Schiene
Thomas Christoph
Jaewoo Lee
Robert Frank
Gregor Bahrenberg
Jean De Vry
Michael Przewosny
Original Assignee
Gruenenthal Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gruenenthal Gmbh filed Critical Gruenenthal Gmbh
Publication of MX2009011139A publication Critical patent/MX2009011139A/es

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    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72Nitrogen atoms
    • C07D213/74Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
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    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
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    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
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MX2009011139A 2007-04-16 2008-04-15 Ligandos de receptor vainilloide novedosos y el uso de los mismos para la produccion de farmacos. MX2009011139A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102007018151A DE102007018151A1 (de) 2007-04-16 2007-04-16 Neue Vanilloid-Rezeptor Liganden und ihre Verwendung zur Herstellung von Arzneimitteln
PCT/EP2008/002994 WO2008125337A2 (de) 2007-04-16 2008-04-15 Neue vanilloid-rezeptor liganden und ihre verwendung zur herstellung von arzneimitteln

Publications (1)

Publication Number Publication Date
MX2009011139A true MX2009011139A (es) 2009-10-30

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Application Number Title Priority Date Filing Date
MX2009011139A MX2009011139A (es) 2007-04-16 2008-04-15 Ligandos de receptor vainilloide novedosos y el uso de los mismos para la produccion de farmacos.

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Country Link
US (2) US8642775B2 (https=)
EP (1) EP2146962A2 (https=)
JP (1) JP5557734B2 (https=)
KR (1) KR101497357B1 (https=)
CN (1) CN101687799B (https=)
BR (1) BRPI0810031A2 (https=)
CA (1) CA2683910A1 (https=)
CO (1) CO6220938A2 (https=)
DE (1) DE102007018151A1 (https=)
EC (1) ECSP099693A (https=)
IL (1) IL201506A0 (https=)
MX (1) MX2009011139A (https=)
NZ (2) NZ599254A (https=)
RU (1) RU2487120C2 (https=)
WO (1) WO2008125337A2 (https=)
ZA (1) ZA200907096B (https=)

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AU2007313295A1 (en) * 2006-10-18 2008-04-24 Merck Sharp & Dohme Corp. 2-hydroxy-2-phenyl/thiophenyl propionamides as androgen receptor modulators
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US8791268B2 (en) 2014-07-29
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CA2683910A1 (en) 2008-04-16
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