MX2009004401A - Proceso para la sulfinilacion de un derivado de pirazol. - Google Patents

Proceso para la sulfinilacion de un derivado de pirazol.

Info

Publication number
MX2009004401A
MX2009004401A MX2009004401A MX2009004401A MX2009004401A MX 2009004401 A MX2009004401 A MX 2009004401A MX 2009004401 A MX2009004401 A MX 2009004401A MX 2009004401 A MX2009004401 A MX 2009004401A MX 2009004401 A MX2009004401 A MX 2009004401A
Authority
MX
Mexico
Prior art keywords
sulfinylation
pyrazole derivative
cf3s
hydroxy group
amine
Prior art date
Application number
MX2009004401A
Other languages
English (en)
Inventor
Michael Keil
Oliver Kuhn
Martin Sukopp
Carsten Groening
Jon J Longlet
Original Assignee
Basf Se
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Basf Se filed Critical Basf Se
Publication of MX2009004401A publication Critical patent/MX2009004401A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/44—Oxygen and nitrogen or sulfur and nitrogen atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Agronomy & Crop Science (AREA)
  • Wood Science & Technology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Epidemiology (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

Un proceso para la sulfinilación de un derivado de pirazol, caracterizado porque 5-amino-1 -[2,6-dicloro-4-(trifluorometil)fen il]-1 H-pirazol-3-carbonitrilo (II) reacciona con un agente S de sulfinilación en presencia de al menos un complejo de amina ácida, en donde la(s) amina(s) se selecciona(n) de aminas secundarias cíclicas y el(los) ácido(s) se selecciona(n) de derivados de ácido sulfónico y con la adición de un agente halogenante, en donde S es [CF3S(O)]2O; o CF3S(O)X en donde X significa fluoro, cloro, bromo, yodo, un grupo hidroxi, o una sal de metal alcalino o alcalinotérreo del grupo hidroxi; o las mezclas de éstos.
MX2009004401A 2006-11-10 2007-11-05 Proceso para la sulfinilacion de un derivado de pirazol. MX2009004401A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US86517806P 2006-11-10 2006-11-10
US91363807P 2007-04-24 2007-04-24
PCT/EP2007/061893 WO2008055879A1 (en) 2006-11-10 2007-11-05 Process for the sulfinylation of a pyrazole derivative

Publications (1)

Publication Number Publication Date
MX2009004401A true MX2009004401A (es) 2009-05-08

Family

ID=39167218

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2009004401A MX2009004401A (es) 2006-11-10 2007-11-05 Proceso para la sulfinilacion de un derivado de pirazol.

Country Status (16)

Country Link
US (1) US8629287B2 (es)
EP (1) EP2081909B8 (es)
JP (1) JP5450078B2 (es)
KR (1) KR20090083454A (es)
CN (1) CN102746234A (es)
AR (1) AR063647A1 (es)
AU (1) AU2007316720B2 (es)
BR (1) BRPI0718773A2 (es)
CA (1) CA2667562A1 (es)
EA (1) EA018047B1 (es)
ES (1) ES2398595T3 (es)
IL (1) IL198260A0 (es)
MX (1) MX2009004401A (es)
NZ (1) NZ576593A (es)
WO (1) WO2008055879A1 (es)
ZA (1) ZA200903969B (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2630849C (en) 2005-12-14 2013-05-14 Makhteshim Chemical Works Ltd. Polymorphs and amorphous forms of 5-amino-1-[2,6-dichloro-4-(trifluoromethyl)phenyl]-4-[(trifluoromethyl)sulfinyl]-1h-pyrazole-3-carbonitrile
ES2422296T3 (es) 2006-11-10 2013-09-10 Basf Se Proceso para la sulfinilación de un derivado pirazol
AU2009299905B2 (en) 2008-10-02 2013-10-10 Boehringer Ingelheim Animal Health USA Inc. Method for producing and purifying trifluoromethanesulfinic acid

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2716453B1 (fr) * 1994-02-22 1996-03-29 Rhone Poulenc Agrochimie Procédé de sulfinylation de composés hétérocycliques.
EP0165136B1 (fr) 1984-05-23 1989-03-01 Rhone-Poulenc Chimie Compositions détergentes comprenant des copolymères à base de polyoxyéthylène et de polyoxyalkylène utilisés comme agents antiredéposants , et leur procédé de preparation
GB8713768D0 (en) * 1987-06-12 1987-07-15 May & Baker Ltd Compositions of matter
BR9710796A (pt) * 1996-08-01 2000-01-11 Rhodia Chimie Sa Processo para enxertar um grupamento difluorometila substituìdo.
JPH11246555A (ja) * 1997-10-31 1999-09-14 Sumitomo Chem Co Ltd フッ素置換ベンゾヘテロ環化合物
DE69720082T2 (de) 1997-12-22 2003-12-11 Minnesota Mining & Mfg Verfahren zur herstellung von fluorierten sulfinaten
DE19853560A1 (de) 1998-11-20 2000-05-25 Bayer Ag Verfahren zur Herstellung von 5-Amino-3-(thio)carbamoylpyrazolen
ES2222743T3 (es) 1999-10-22 2005-02-01 Bayer Cropscience S.A. Procedimiento para preparar un derivado 4-trifluorometilsulfinilpirazol.
JP2001220386A (ja) * 1999-11-30 2001-08-14 Takeda Chem Ind Ltd オキサジアゾリン誘導体の製造方法
JP2002020364A (ja) * 2000-07-06 2002-01-23 Konica Corp スルフィン酸ナトリウム、スルフィン酸カリウムの製造方法およびそれらを用いた写真用カプラーの製造方法
EP1331222A1 (en) * 2002-01-28 2003-07-30 Virbac S.A. Environment friendly reagents and process for halogenoalkylsulfinylation of organic compounds
CN1176078C (zh) * 2002-03-27 2004-11-17 江苏省农药研究所 带三氟甲基亚磺酰基的吡唑类化合物的亚磺酰化方法
BRPI0718758A2 (pt) 2006-11-10 2013-12-03 Basf Se " processo para a sulfinilação de um derivado de pirazol, composto, composição pesticida ou parasiticida, uso de um composto, métodos para o controle de insetos, acarídeos ou nematódeos, para proteger plantas em crescimento, e para tratar, controlar, prevenir ou proteger animais, e, processo para a preparação de uma composição."
ES2422296T3 (es) 2006-11-10 2013-09-10 Basf Se Proceso para la sulfinilación de un derivado pirazol
FR2924115B1 (fr) 2007-11-27 2010-02-26 Rhodia Operations Procede de preparation d'un acide trifluoromethanesulfinique
AU2009299905B2 (en) * 2008-10-02 2013-10-10 Boehringer Ingelheim Animal Health USA Inc. Method for producing and purifying trifluoromethanesulfinic acid

Also Published As

Publication number Publication date
WO2008055879A1 (en) 2008-05-15
JP2010509272A (ja) 2010-03-25
ES2398595T3 (es) 2013-03-20
EP2081909B1 (en) 2013-01-09
JP5450078B2 (ja) 2014-03-26
KR20090083454A (ko) 2009-08-03
US8629287B2 (en) 2014-01-14
ZA200903969B (en) 2012-02-29
AU2007316720A1 (en) 2008-05-15
BRPI0718773A2 (pt) 2013-12-03
EA018047B1 (ru) 2013-05-30
CN102746234A (zh) 2012-10-24
EP2081909B8 (en) 2013-02-20
IL198260A0 (en) 2009-12-24
EA200900627A1 (ru) 2009-10-30
EP2081909A1 (en) 2009-07-29
CA2667562A1 (en) 2008-05-15
NZ576593A (en) 2011-12-22
US20100093822A1 (en) 2010-04-15
AU2007316720B2 (en) 2013-05-09
AR063647A1 (es) 2009-02-04

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