MX2009004259A - Proceso para la sulfinilacion de un derivado de pirazol. - Google Patents
Proceso para la sulfinilacion de un derivado de pirazol.Info
- Publication number
- MX2009004259A MX2009004259A MX2009004259A MX2009004259A MX2009004259A MX 2009004259 A MX2009004259 A MX 2009004259A MX 2009004259 A MX2009004259 A MX 2009004259A MX 2009004259 A MX2009004259 A MX 2009004259A MX 2009004259 A MX2009004259 A MX 2009004259A
- Authority
- MX
- Mexico
- Prior art keywords
- sulfinylation
- acid
- cf3s
- hydroxy group
- amine
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/44—Oxygen and nitrogen or sulfur and nitrogen atoms
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
- A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
- A01N47/02—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having no bond to a nitrogen atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
Landscapes
- Life Sciences & Earth Sciences (AREA)
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Environmental Sciences (AREA)
- Agronomy & Crop Science (AREA)
- Zoology (AREA)
- Wood Science & Technology (AREA)
- Dentistry (AREA)
- Engineering & Computer Science (AREA)
- Plant Pathology (AREA)
- Pest Control & Pesticides (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Tropical Medicine & Parasitology (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Epidemiology (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Catalysts (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
La presente invención se relaciona con un proceso para la sulfinilación de un derivado de pirazol, caracterizado porque se hace reaccionar 5-amino-1-[2,6-dicloro-4-(trifluorometil)fenil]-1H -pirazol-3-carbonitrilo (II) con un agente de sulfinilación S en presencia de al menos un complejo de amina ácida, en donde la(s) amina(s) es/son seleccionada(s) de amina(s) secundaria(s) y/o terciaria(s) y el/los ácido(s) es/son seleccionado(s) de ácido fluorhídrico, clorhídrico, bromhídrico y yodhídrico, y derivados del ácido sulfónico, y con la adición de un agente halogenante, en donde S es [CF3S(O)]2O; o CF3S(o)X en donde X significa flúor, cloro, bromo, yodo, un grupo hidroxi, o una sal de metal alcalino o alcalino térreo del grupo hidroxi; o sus mezclas, en donde la temperatura de la mezcla de la reacción en ningún momento excede los 39ºC.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US86517806P | 2006-11-10 | 2006-11-10 | |
US91364607P | 2007-04-24 | 2007-04-24 | |
PCT/EP2007/061894 WO2008055880A1 (en) | 2006-11-10 | 2007-11-05 | Process for the sulfinylation of a pyrazole derivative |
Publications (1)
Publication Number | Publication Date |
---|---|
MX2009004259A true MX2009004259A (es) | 2009-05-05 |
Family
ID=38983360
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MX2009004259A MX2009004259A (es) | 2006-11-10 | 2007-11-05 | Proceso para la sulfinilacion de un derivado de pirazol. |
Country Status (17)
Country | Link |
---|---|
US (1) | US20100004307A1 (es) |
EP (1) | EP2084137B1 (es) |
JP (1) | JP5450079B2 (es) |
KR (1) | KR20090081421A (es) |
AR (1) | AR063648A1 (es) |
AU (1) | AU2007316721B2 (es) |
BR (1) | BRPI0718758A2 (es) |
CA (1) | CA2667565A1 (es) |
DK (1) | DK2084137T3 (es) |
EA (1) | EA016304B1 (es) |
ES (1) | ES2422297T3 (es) |
IL (1) | IL198261A0 (es) |
MX (1) | MX2009004259A (es) |
NZ (1) | NZ576638A (es) |
PL (1) | PL2084137T3 (es) |
WO (1) | WO2008055880A1 (es) |
ZA (1) | ZA200903973B (es) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US8440709B2 (en) | 2005-12-14 | 2013-05-14 | Makhteshim Chemical Works Ltd. | Polymorphs and amorphous forms of 5-amino-1-[2,6-dichloro-4-(trifluoromethyl)phenyl]-4-[(trifluoromethyl)sulfinyl]-1H-pyrazole-3-carbonitrile |
DK2081908T3 (da) | 2006-11-10 | 2013-07-29 | Basf Agro B V Arnhem Nl Zuerich Branch | Fremgangsmåde til sulfinylering af et pyrazolderivat |
BRPI0718773A2 (pt) | 2006-11-10 | 2013-12-03 | Basf Se | " processo para a sulfinilação de um derivado de pirazol, composto, composição pesticida ou parasiticida, uso de um composto, métodos para controlar insetos, acarídeos ou nematódeos, para proteger plantas em crescimento e para tratar, controlar, prevenir ou proteger animais, e, processo para a preparação de uma composição." |
FR2925493B1 (fr) * | 2007-12-19 | 2011-09-30 | Vetoquinol | Procede de preparation du fipronil et d'analogues de celui-ci. |
DK2349987T3 (da) | 2008-10-02 | 2013-03-11 | Basf Se | Fremgangsmåde til fremstilling og oprensning af trifluormethansulfinsyre |
CN104926729B (zh) * | 2014-03-18 | 2018-01-19 | 上海泰禾国际贸易有限公司 | 一种合成氟虫腈的方法 |
Family Cites Families (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2716453B1 (fr) * | 1994-02-22 | 1996-03-29 | Rhone Poulenc Agrochimie | Procédé de sulfinylation de composés hétérocycliques. |
EP0165136B1 (fr) * | 1984-05-23 | 1989-03-01 | Rhone-Poulenc Chimie | Compositions détergentes comprenant des copolymères à base de polyoxyéthylène et de polyoxyalkylène utilisés comme agents antiredéposants , et leur procédé de preparation |
GB8713768D0 (en) * | 1987-06-12 | 1987-07-15 | May & Baker Ltd | Compositions of matter |
BR9710796A (pt) * | 1996-08-01 | 2000-01-11 | Rhodia Chimie Sa | Processo para enxertar um grupamento difluorometila substituìdo. |
JPH11246555A (ja) * | 1997-10-31 | 1999-09-14 | Sumitomo Chem Co Ltd | フッ素置換ベンゾヘテロ環化合物 |
JP2001220386A (ja) * | 1999-11-30 | 2001-08-14 | Takeda Chem Ind Ltd | オキサジアゾリン誘導体の製造方法 |
JP2002020364A (ja) * | 2000-07-06 | 2002-01-23 | Konica Corp | スルフィン酸ナトリウム、スルフィン酸カリウムの製造方法およびそれらを用いた写真用カプラーの製造方法 |
EP1331222A1 (en) * | 2002-01-28 | 2003-07-30 | Virbac S.A. | Environment friendly reagents and process for halogenoalkylsulfinylation of organic compounds |
CN1176078C (zh) * | 2002-03-27 | 2004-11-17 | 江苏省农药研究所 | 带三氟甲基亚磺酰基的吡唑类化合物的亚磺酰化方法 |
DK2349987T3 (da) * | 2008-10-02 | 2013-03-11 | Basf Se | Fremgangsmåde til fremstilling og oprensning af trifluormethansulfinsyre |
-
2007
- 2007-11-05 CA CA002667565A patent/CA2667565A1/en not_active Abandoned
- 2007-11-05 ES ES07822223T patent/ES2422297T3/es active Active
- 2007-11-05 KR KR1020097011873A patent/KR20090081421A/ko not_active Application Discontinuation
- 2007-11-05 DK DK07822223.9T patent/DK2084137T3/da active
- 2007-11-05 PL PL07822223T patent/PL2084137T3/pl unknown
- 2007-11-05 NZ NZ576638A patent/NZ576638A/en not_active IP Right Cessation
- 2007-11-05 BR BRPI0718758-0A patent/BRPI0718758A2/pt not_active Application Discontinuation
- 2007-11-05 EP EP07822223.9A patent/EP2084137B1/en active Active
- 2007-11-05 US US12/514,109 patent/US20100004307A1/en not_active Abandoned
- 2007-11-05 JP JP2009535704A patent/JP5450079B2/ja not_active Expired - Fee Related
- 2007-11-05 WO PCT/EP2007/061894 patent/WO2008055880A1/en active Application Filing
- 2007-11-05 MX MX2009004259A patent/MX2009004259A/es active IP Right Grant
- 2007-11-05 EA EA200900628A patent/EA016304B1/ru not_active IP Right Cessation
- 2007-11-05 AU AU2007316721A patent/AU2007316721B2/en active Active
- 2007-11-09 AR ARP070105014A patent/AR063648A1/es not_active Application Discontinuation
-
2009
- 2009-04-21 IL IL198261A patent/IL198261A0/en unknown
- 2009-06-08 ZA ZA2009/03973A patent/ZA200903973B/en unknown
Also Published As
Publication number | Publication date |
---|---|
NZ576638A (en) | 2011-12-22 |
US20100004307A1 (en) | 2010-01-07 |
WO2008055880A1 (en) | 2008-05-15 |
ES2422297T3 (es) | 2013-09-10 |
EP2084137B1 (en) | 2013-04-24 |
JP2010509273A (ja) | 2010-03-25 |
JP5450079B2 (ja) | 2014-03-26 |
KR20090081421A (ko) | 2009-07-28 |
AU2007316721A1 (en) | 2008-05-15 |
AR063648A1 (es) | 2009-02-04 |
EA016304B1 (ru) | 2012-04-30 |
PL2084137T3 (pl) | 2013-11-29 |
ZA200903973B (en) | 2012-02-29 |
IL198261A0 (en) | 2009-12-24 |
CA2667565A1 (en) | 2008-05-15 |
EP2084137A1 (en) | 2009-08-05 |
BRPI0718758A2 (pt) | 2013-12-03 |
EA200900628A1 (ru) | 2009-12-30 |
AU2007316721B2 (en) | 2013-05-09 |
DK2084137T3 (da) | 2013-07-22 |
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Legal Events
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FG | Grant or registration |