TW200639167A - Pharmaceutical compounds - Google Patents

Pharmaceutical compounds

Info

Publication number
TW200639167A
TW200639167A TW095101703A TW95101703A TW200639167A TW 200639167 A TW200639167 A TW 200639167A TW 095101703 A TW095101703 A TW 095101703A TW 95101703 A TW95101703 A TW 95101703A TW 200639167 A TW200639167 A TW 200639167A
Authority
TW
Taiwan
Prior art keywords
ylamide
benzoylamino
pyrazole
dichloro
acid
Prior art date
Application number
TW095101703A
Other languages
Chinese (zh)
Other versions
TWI455932B (en
Inventor
David Charles Rees
Gary Trewartha
Mladen Vinkovic
Paul Graham Wyatt
Original Assignee
Astex Therapeutics Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astex Therapeutics Ltd filed Critical Astex Therapeutics Ltd
Publication of TW200639167A publication Critical patent/TW200639167A/en
Application granted granted Critical
Publication of TWI455932B publication Critical patent/TWI455932B/en

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  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

The invention provides an acid addition salt of 4-(2,6-dichloro-benzoylamino)-1H-pyrazole-3-carboxylic acid piperidin-4-ylamide and crystals thereof, the salt being formed with an acid selected from methanesulphonic acid and acetic acid and mixtures thereof. Also provided are the novel uses of salts of 4-(2,6-dichloro-benzoylamino)-1H-pyrazole-3-carboxylic acid piperidin-4-ylamide, processes for the preparation of 4-(2,6-dichloro-benzoylamino)-1H-pyrazole-3-carboxylic acid piperidin-4-ylamide and its salts and novel chemical intermediates.
TW095101703A 2005-01-21 2006-01-17 Acid addition salts of, processes for preparing, and uses of 4-(2,6-dichloro-benzoylamino)-1H-pyrazole-3-carboxylic acid piperidin-4-ylamide TWI455932B (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US64597305P 2005-01-21 2005-01-21
GB0501475A GB0501475D0 (en) 2005-01-22 2005-01-22 Pharmaceutical compounds

Publications (2)

Publication Number Publication Date
TW200639167A true TW200639167A (en) 2006-11-16
TWI455932B TWI455932B (en) 2014-10-11

Family

ID=34259610

Family Applications (1)

Application Number Title Priority Date Filing Date
TW095101703A TWI455932B (en) 2005-01-21 2006-01-17 Acid addition salts of, processes for preparing, and uses of 4-(2,6-dichloro-benzoylamino)-1H-pyrazole-3-carboxylic acid piperidin-4-ylamide

Country Status (4)

Country Link
GB (1) GB0501475D0 (en)
GT (1) GT200600012A (en)
MY (1) MY148886A (en)
TW (1) TWI455932B (en)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN116283779A (en) * 2023-03-29 2023-06-23 河南大学 Carboxylic acid schiff base, its preparation method and its application as metal and alloy corrosion inhibitor

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9872445B2 (en) 2010-09-30 2018-01-23 The Toro Company Turf management

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0102687D0 (en) * 2001-02-02 2001-03-21 Pharmacia & Upjohn Spa Oxazolyl-pyrazole derivatives active as kinase inhibitors,process for their preparation and pharmaceutical compositions comprising them

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN116283779A (en) * 2023-03-29 2023-06-23 河南大学 Carboxylic acid schiff base, its preparation method and its application as metal and alloy corrosion inhibitor

Also Published As

Publication number Publication date
TWI455932B (en) 2014-10-11
MY148886A (en) 2013-06-14
GT200600012A (en) 2006-08-09
GB0501475D0 (en) 2005-03-02

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Legal Events

Date Code Title Description
MM4A Annulment or lapse of patent due to non-payment of fees