MX2008012791A - Terapia de combinacion de (2r,z)-2-amino-2-ciclohexil-n-(5-(1-meti l-1h-pirazol-4-il)-1-oxo-2,6-dihidro-1h-[1,2]diazepinos[4,5,6-cd[ indol-8-il)acetamida. - Google Patents
Terapia de combinacion de (2r,z)-2-amino-2-ciclohexil-n-(5-(1-meti l-1h-pirazol-4-il)-1-oxo-2,6-dihidro-1h-[1,2]diazepinos[4,5,6-cd[ indol-8-il)acetamida.Info
- Publication number
- MX2008012791A MX2008012791A MX2008012791A MX2008012791A MX2008012791A MX 2008012791 A MX2008012791 A MX 2008012791A MX 2008012791 A MX2008012791 A MX 2008012791A MX 2008012791 A MX2008012791 A MX 2008012791A MX 2008012791 A MX2008012791 A MX 2008012791A
- Authority
- MX
- Mexico
- Prior art keywords
- cancer
- oxo
- methyl
- cyclohexyl
- amino
- Prior art date
Links
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Landscapes
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US78927606P | 2006-04-04 | 2006-04-04 | |
| PCT/IB2007/000928 WO2007113671A1 (en) | 2006-04-04 | 2007-03-26 | Combination therapy of (2r,z)-2-amino-2-cyclohexyl-n-(5-(1-methyl-1h-pyrazol-4-yl)-1-oxo-2,6-dihydro-1h-[1,2]diazepino[4,5,6-cd]indol-8-yl)acetamide |
Publications (1)
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| MX2008012791A true MX2008012791A (es) | 2008-10-15 |
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| Application Number | Title | Priority Date | Filing Date |
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| MX2008012791A MX2008012791A (es) | 2006-04-04 | 2007-03-26 | Terapia de combinacion de (2r,z)-2-amino-2-ciclohexil-n-(5-(1-meti l-1h-pirazol-4-il)-1-oxo-2,6-dihidro-1h-[1,2]diazepinos[4,5,6-cd[ indol-8-il)acetamida. |
Country Status (14)
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| US (1) | US20090312280A1 (https=) |
| EP (1) | EP2007375A1 (https=) |
| JP (1) | JP2007277240A (https=) |
| KR (1) | KR20080100838A (https=) |
| CN (1) | CN101415417A (https=) |
| AR (1) | AR060284A1 (https=) |
| AU (1) | AU2007232279B2 (https=) |
| BR (1) | BRPI0709731A2 (https=) |
| CA (1) | CA2648371A1 (https=) |
| IL (1) | IL194340A0 (https=) |
| MX (1) | MX2008012791A (https=) |
| RU (1) | RU2409361C2 (https=) |
| TW (1) | TW200806301A (https=) |
| WO (1) | WO2007113671A1 (https=) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPWO2009113436A1 (ja) * | 2008-03-14 | 2011-07-21 | 国立大学法人 千葉大学 | Ｆｇｆｒ３遺伝子阻害剤の放射線照射併用による放射線の抗癌作用増強法および副作用軽減法 |
| KR20100131457A (ko) * | 2008-03-27 | 2010-12-15 | 다이호야쿠힌고교 가부시키가이샤 | 시티딘 유도체 및 카르보플라틴을 함유하는 항종양제 |
| US8481557B2 (en) | 2009-04-11 | 2013-07-09 | Array Biopharma Inc. | Method of treatment using checkpoint kinase 1 inhibitors |
| SG10201404012RA (en) * | 2009-04-11 | 2014-09-26 | Array Biopharma Inc | Checkpoint kinase 1 inhibitors for potentiating dna damaging agents |
| ES2621857T3 (es) | 2010-11-16 | 2017-07-05 | Array Biopharma, Inc. | Combinación de inhibidores de la cinasa 1 de punto de control e inhibidores de la cinasa WEE1 |
| IN2014DN06169A (https=) | 2011-12-31 | 2015-08-21 | Beigene Ltd | |
| MX2014008071A (es) | 2011-12-31 | 2015-07-06 | Beigene Ltd | Tetra o penta-piridoftalazinonas ciclicas fusionadas como inhibidores de poli(adenosin-difosfato-ribosa)polimerasas. |
| CN105764501A (zh) | 2013-07-26 | 2016-07-13 | 现代化制药公司 | 改善比生群治疗效益的组合物 |
| EP3461480A1 (en) | 2017-09-27 | 2019-04-03 | Onxeo | Combination of a dna damage response cell cycle checkpoint inhibitors and belinostat for treating cancer |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SE9704545D0 (sv) * | 1997-12-05 | 1997-12-05 | Astra Pharma Prod | Novel compounds |
| CA2512683C (en) * | 2003-01-09 | 2010-03-16 | Pfizer Inc. | Tricyclic compounds protein kinase inhibitors for enhancing the efficacy of anti-neoplastic agents and radiation therapy |
-
2007
- 2007-03-26 CN CNA2007800121818A patent/CN101415417A/zh active Pending
- 2007-03-26 AU AU2007232279A patent/AU2007232279B2/en not_active Ceased
- 2007-03-26 KR KR1020087024155A patent/KR20080100838A/ko not_active Ceased
- 2007-03-26 US US12/295,986 patent/US20090312280A1/en not_active Abandoned
- 2007-03-26 BR BRPI0709731-0A patent/BRPI0709731A2/pt not_active IP Right Cessation
- 2007-03-26 WO PCT/IB2007/000928 patent/WO2007113671A1/en not_active Ceased
- 2007-03-26 CA CA002648371A patent/CA2648371A1/en not_active Abandoned
- 2007-03-26 MX MX2008012791A patent/MX2008012791A/es unknown
- 2007-03-26 EP EP07734247A patent/EP2007375A1/en not_active Withdrawn
- 2007-03-26 RU RU2008139406/15A patent/RU2409361C2/ru not_active IP Right Cessation
- 2007-04-03 TW TW096111825A patent/TW200806301A/zh unknown
- 2007-04-03 AR ARP070101414A patent/AR060284A1/es not_active Application Discontinuation
- 2007-04-04 JP JP2007097995A patent/JP2007277240A/ja not_active Withdrawn
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2008
- 2008-09-25 IL IL194340A patent/IL194340A0/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| BRPI0709731A2 (pt) | 2011-07-26 |
| JP2007277240A (ja) | 2007-10-25 |
| AR060284A1 (es) | 2008-06-04 |
| CA2648371A1 (en) | 2007-10-11 |
| RU2409361C2 (ru) | 2011-01-20 |
| RU2008139406A (ru) | 2010-04-10 |
| AU2007232279A1 (en) | 2007-10-11 |
| AU2007232279B2 (en) | 2010-05-06 |
| IL194340A0 (en) | 2009-08-03 |
| WO2007113671A1 (en) | 2007-10-11 |
| CN101415417A (zh) | 2009-04-22 |
| EP2007375A1 (en) | 2008-12-31 |
| US20090312280A1 (en) | 2009-12-17 |
| KR20080100838A (ko) | 2008-11-19 |
| TW200806301A (en) | 2008-02-01 |
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