MX2008012791A - Terapia de combinacion de (2r,z)-2-amino-2-ciclohexil-n-(5-(1-meti l-1h-pirazol-4-il)-1-oxo-2,6-dihidro-1h-[1,2]diazepinos[4,5,6-cd[ indol-8-il)acetamida. - Google Patents
Terapia de combinacion de (2r,z)-2-amino-2-ciclohexil-n-(5-(1-meti l-1h-pirazol-4-il)-1-oxo-2,6-dihidro-1h-[1,2]diazepinos[4,5,6-cd[ indol-8-il)acetamida.Info
- Publication number
- MX2008012791A MX2008012791A MX2008012791A MX2008012791A MX2008012791A MX 2008012791 A MX2008012791 A MX 2008012791A MX 2008012791 A MX2008012791 A MX 2008012791A MX 2008012791 A MX2008012791 A MX 2008012791A MX 2008012791 A MX2008012791 A MX 2008012791A
- Authority
- MX
- Mexico
- Prior art keywords
- cancer
- oxo
- methyl
- cyclohexyl
- amino
- Prior art date
Links
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- A61K31/4738—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems
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Landscapes
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US78927606P | 2006-04-04 | 2006-04-04 | |
| PCT/IB2007/000928 WO2007113671A1 (en) | 2006-04-04 | 2007-03-26 | Combination therapy of (2r,z)-2-amino-2-cyclohexyl-n-(5-(1-methyl-1h-pyrazol-4-yl)-1-oxo-2,6-dihydro-1h-[1,2]diazepino[4,5,6-cd]indol-8-yl)acetamide |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX2008012791A true MX2008012791A (es) | 2008-10-15 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2008012791A MX2008012791A (es) | 2006-04-04 | 2007-03-26 | Terapia de combinacion de (2r,z)-2-amino-2-ciclohexil-n-(5-(1-meti l-1h-pirazol-4-il)-1-oxo-2,6-dihidro-1h-[1,2]diazepinos[4,5,6-cd[ indol-8-il)acetamida. |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US20090312280A1 (enExample) |
| EP (1) | EP2007375A1 (enExample) |
| JP (1) | JP2007277240A (enExample) |
| KR (1) | KR20080100838A (enExample) |
| CN (1) | CN101415417A (enExample) |
| AR (1) | AR060284A1 (enExample) |
| AU (1) | AU2007232279B2 (enExample) |
| BR (1) | BRPI0709731A2 (enExample) |
| CA (1) | CA2648371A1 (enExample) |
| IL (1) | IL194340A0 (enExample) |
| MX (1) | MX2008012791A (enExample) |
| RU (1) | RU2409361C2 (enExample) |
| TW (1) | TW200806301A (enExample) |
| WO (1) | WO2007113671A1 (enExample) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2009113436A1 (ja) * | 2008-03-14 | 2009-09-17 | 国立大学法人千葉大学 | Ｆｇｆｒ３遺伝子阻害剤の放射線照射併用による放射線の抗癌作用増強法および副作用軽減法 |
| SG189699A1 (en) * | 2008-03-27 | 2013-05-31 | Taiho Pharmaceutical Co Ltd | Anti-tumor agent comprising cytidine derivative and carboplatin |
| EP2416773B1 (en) * | 2009-04-11 | 2016-09-28 | Array Biopharma, Inc. | Checkpoint kinase 1 inhibitors for potentiating dna damaging agents |
| US8481557B2 (en) | 2009-04-11 | 2013-07-09 | Array Biopharma Inc. | Method of treatment using checkpoint kinase 1 inhibitors |
| EP2640386B1 (en) | 2010-11-16 | 2017-01-18 | Array Biopharma Inc. | Combination of checkpoint kinase 1 inhibitors and wee 1 kinase inhibitors |
| EP2797919B1 (en) | 2011-12-31 | 2017-03-29 | BeiGene, Ltd. | Fused tetra or penta-cyclic pyridophthalazinones as parp inhibitors |
| MX353578B (es) | 2011-12-31 | 2018-01-19 | Beigene Ltd | Dihidrodiazpinocarbazolonas tetra o penta-ciclicas fusionadas como inhibidores de poli (adp-ribosa) polimerasa (parp). |
| CA2928568A1 (en) | 2013-07-26 | 2015-01-29 | Update Pharma Inc. | Combinatorial methods to improve the therapeutic benefit of bisantrene |
| EP3461480A1 (en) | 2017-09-27 | 2019-04-03 | Onxeo | Combination of a dna damage response cell cycle checkpoint inhibitors and belinostat for treating cancer |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SE9704545D0 (sv) * | 1997-12-05 | 1997-12-05 | Astra Pharma Prod | Novel compounds |
| SI1585749T1 (sl) * | 2003-01-09 | 2008-10-31 | Pfizer | Derivati diazepinoindola kot inhibitorji kinaze |
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2007
- 2007-03-26 MX MX2008012791A patent/MX2008012791A/es unknown
- 2007-03-26 BR BRPI0709731-0A patent/BRPI0709731A2/pt not_active IP Right Cessation
- 2007-03-26 CA CA002648371A patent/CA2648371A1/en not_active Abandoned
- 2007-03-26 AU AU2007232279A patent/AU2007232279B2/en not_active Ceased
- 2007-03-26 EP EP07734247A patent/EP2007375A1/en not_active Withdrawn
- 2007-03-26 US US12/295,986 patent/US20090312280A1/en not_active Abandoned
- 2007-03-26 RU RU2008139406/15A patent/RU2409361C2/ru not_active IP Right Cessation
- 2007-03-26 KR KR1020087024155A patent/KR20080100838A/ko not_active Ceased
- 2007-03-26 WO PCT/IB2007/000928 patent/WO2007113671A1/en not_active Ceased
- 2007-03-26 CN CNA2007800121818A patent/CN101415417A/zh active Pending
- 2007-04-03 TW TW096111825A patent/TW200806301A/zh unknown
- 2007-04-03 AR ARP070101414A patent/AR060284A1/es not_active Application Discontinuation
- 2007-04-04 JP JP2007097995A patent/JP2007277240A/ja not_active Withdrawn
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2008
- 2008-09-25 IL IL194340A patent/IL194340A0/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| JP2007277240A (ja) | 2007-10-25 |
| AU2007232279B2 (en) | 2010-05-06 |
| KR20080100838A (ko) | 2008-11-19 |
| CA2648371A1 (en) | 2007-10-11 |
| CN101415417A (zh) | 2009-04-22 |
| US20090312280A1 (en) | 2009-12-17 |
| RU2008139406A (ru) | 2010-04-10 |
| IL194340A0 (en) | 2009-08-03 |
| EP2007375A1 (en) | 2008-12-31 |
| WO2007113671A1 (en) | 2007-10-11 |
| TW200806301A (en) | 2008-02-01 |
| AU2007232279A1 (en) | 2007-10-11 |
| AR060284A1 (es) | 2008-06-04 |
| RU2409361C2 (ru) | 2011-01-20 |
| BRPI0709731A2 (pt) | 2011-07-26 |
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