MX2007002248A - Triazolobenzodiazepinas y su uso como antagonistas de vasopresina. - Google Patents
Triazolobenzodiazepinas y su uso como antagonistas de vasopresina.Info
- Publication number
- MX2007002248A MX2007002248A MX2007002248A MX2007002248A MX2007002248A MX 2007002248 A MX2007002248 A MX 2007002248A MX 2007002248 A MX2007002248 A MX 2007002248A MX 2007002248 A MX2007002248 A MX 2007002248A MX 2007002248 A MX2007002248 A MX 2007002248A
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Links
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- XJDNKRIXUMDJCW-UHFFFAOYSA-J titanium tetrachloride Chemical compound Cl[Ti](Cl)(Cl)Cl XJDNKRIXUMDJCW-UHFFFAOYSA-J 0.000 description 1
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Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
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- A—HUMAN NECESSITIES
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- A61P15/06—Antiabortive agents; Labour repressants
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- A—HUMAN NECESSITIES
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- A61P15/12—Drugs for genital or sexual disorders; Contraceptives for climacteric disorders
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- A—HUMAN NECESSITIES
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Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Hospice & Palliative Care (AREA)
- Neurosurgery (AREA)
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- Rheumatology (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Urology & Nephrology (AREA)
- Hematology (AREA)
- Vascular Medicine (AREA)
- Gynecology & Obstetrics (AREA)
- Pregnancy & Childbirth (AREA)
- Otolaryngology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB0418980A GB0418980D0 (en) | 2004-08-25 | 2004-08-25 | Triazole compounds useful in therapy |
| US61660104P | 2004-10-05 | 2004-10-05 | |
| PCT/IB2005/002711 WO2006021882A1 (en) | 2004-08-25 | 2005-08-12 | Triazolobenzodiazepines and their use as vasopressin antagonists |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX2007002248A true MX2007002248A (es) | 2008-10-02 |
Family
ID=35355092
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2007002248A MX2007002248A (es) | 2004-08-25 | 2005-08-12 | Triazolobenzodiazepinas y su uso como antagonistas de vasopresina. |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US7456170B2 (https=) |
| EP (1) | EP1784408A1 (https=) |
| JP (1) | JP2008510789A (https=) |
| BR (1) | BRPI0514458A (https=) |
| CA (1) | CA2578370A1 (https=) |
| MX (1) | MX2007002248A (https=) |
| WO (1) | WO2006021882A1 (https=) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SI2356123T1 (sl) | 2008-11-13 | 2013-01-31 | F. Hoffmann-La Roche Ag | Piro-5,6-dihidro-4h-2,3,5,10b-tetraaza-benzo(e)azuleni |
| KR101385433B1 (ko) | 2008-11-18 | 2014-04-14 | 에프. 호프만-라 로슈 아게 | 다이하이드로테트라아자벤조아줄렌의 알킬사이클로헥실에터 |
| HRP20131067T1 (hr) * | 2008-11-28 | 2013-12-06 | F. Hoffmann - La Roche Ag | Arilcikloheksileteri od dihidrotetraazabenzoazulena za primjenu kao antagonista receptora vazopresina v1a |
| US8420633B2 (en) * | 2010-03-31 | 2013-04-16 | Hoffmann-La Roche Inc. | Aryl-cyclohexyl-tetraazabenzo[e]azulenes |
| US8461151B2 (en) | 2010-04-13 | 2013-06-11 | Hoffmann-La Roche Inc. | Aryl-/heteroaryl-cyclohexenyl-tetraazabenzo[e]azulenes |
| US8492376B2 (en) * | 2010-04-21 | 2013-07-23 | Hoffmann-La Roche Inc. | Heteroaryl-cyclohexyl-tetraazabenzo[e]azulenes |
| US8481528B2 (en) * | 2010-04-26 | 2013-07-09 | Hoffmann-La Roche Inc. | Heterobiaryl-cyclohexyl-tetraazabenzo[e]azulenes |
| US8513238B2 (en) * | 2010-05-10 | 2013-08-20 | Hoffmann-La Roche Inc. | Heteroaryl-cyclohexyl-tetraazabenzo[E]azulenes |
| US8828989B2 (en) * | 2011-09-26 | 2014-09-09 | Hoffmann-La Roche Inc. | Oxy-cyclohexyl-4H,6H-5-oxa-2,3,10b-triaza-benzo[E]azulenes as V1A antagonists |
| HUE034118T2 (en) | 2012-03-06 | 2018-01-29 | Pfizer | Macrocyclic derivatives for the treatment of proliferative diseases |
| CA2919738A1 (en) * | 2013-08-19 | 2015-02-26 | F. Hoffmann-La Roche Ag | V1a antagonists to treat phase shift sleep disorders |
| NZ720340A (en) | 2013-12-05 | 2020-03-27 | Hoffmann La Roche | Synthesis of trans-8-chloro-5-methyl-1 -[4-(pyridin-2-yloxy)-cyclohexyl]-5,6-dihydro-4h-2,3,5,10b-tetraaza-benzo[e]azulene and crystalline forms thereof |
| HU231206B1 (hu) | 2017-12-15 | 2021-10-28 | Richter Gedeon Nyrt. | Triazolobenzazepinek |
| TW201938171A (zh) | 2017-12-15 | 2019-10-01 | 匈牙利商羅特格登公司 | 作為血管升壓素V1a受體拮抗劑之三環化合物 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE69826487T2 (de) | 1997-07-30 | 2005-12-01 | Wyeth | Trizyclische vasopressin-agonisten |
| CN100379723C (zh) * | 2002-02-19 | 2008-04-09 | 特瓦制药工业有限公司 | 阿托伐他汀半钙脱溶剂的方法和基本上不含有机溶剂的阿托伐他汀半钙 |
| GB0303852D0 (en) * | 2003-02-19 | 2003-03-26 | Pfizer Ltd | Triazole compounds useful in therapy |
| US7119088B2 (en) * | 2003-02-19 | 2006-10-10 | Pfizer Inc. | Triazole compounds useful in therapy |
-
2005
- 2005-08-12 WO PCT/IB2005/002711 patent/WO2006021882A1/en not_active Ceased
- 2005-08-12 MX MX2007002248A patent/MX2007002248A/es unknown
- 2005-08-12 BR BRPI0514458-2A patent/BRPI0514458A/pt not_active IP Right Cessation
- 2005-08-12 EP EP05781153A patent/EP1784408A1/en not_active Withdrawn
- 2005-08-12 JP JP2007529032A patent/JP2008510789A/ja not_active Withdrawn
- 2005-08-12 US US11/570,694 patent/US7456170B2/en not_active Expired - Fee Related
- 2005-08-12 CA CA002578370A patent/CA2578370A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| BRPI0514458A (pt) | 2008-06-10 |
| JP2008510789A (ja) | 2008-04-10 |
| EP1784408A1 (en) | 2007-05-16 |
| CA2578370A1 (en) | 2006-03-02 |
| US20070249585A1 (en) | 2007-10-25 |
| WO2006021882A1 (en) | 2006-03-02 |
| US7456170B2 (en) | 2008-11-25 |
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