MA52348A - Composés hétéroaromatiques ayant une activité contre vrs - Google Patents
Composés hétéroaromatiques ayant une activité contre vrsInfo
- Publication number
- MA52348A MA52348A MA052348A MA52348A MA52348A MA 52348 A MA52348 A MA 52348A MA 052348 A MA052348 A MA 052348A MA 52348 A MA52348 A MA 52348A MA 52348 A MA52348 A MA 52348A
- Authority
- MA
- Morocco
- Prior art keywords
- activity against
- heteroaromatic compounds
- against rsv
- rsv
- heteroaromatic
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/472—Non-condensed isoquinolines, e.g. papaverine
- A61K31/4725—Non-condensed isoquinolines, e.g. papaverine containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/16—Antivirals for RNA viruses for influenza or rhinoviruses
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP18168671 | 2018-04-23 |
Publications (1)
Publication Number | Publication Date |
---|---|
MA52348A true MA52348A (fr) | 2021-03-03 |
Family
ID=62046706
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MA052348A MA52348A (fr) | 2018-04-23 | 2019-04-19 | Composés hétéroaromatiques ayant une activité contre vrs |
Country Status (13)
Country | Link |
---|---|
US (1) | US11708369B2 (fr) |
EP (1) | EP3784667B1 (fr) |
JP (1) | JP2021522222A (fr) |
KR (1) | KR20210005569A (fr) |
CN (1) | CN112004815A (fr) |
AU (1) | AU2019260109B2 (fr) |
CA (1) | CA3095277A1 (fr) |
EA (1) | EA202092439A1 (fr) |
ES (1) | ES2957316T3 (fr) |
MA (1) | MA52348A (fr) |
MX (1) | MX2020011200A (fr) |
SG (1) | SG11202010323QA (fr) |
WO (1) | WO2019206828A1 (fr) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA3087926A1 (fr) | 2018-01-31 | 2019-08-08 | Janssen Sciences Ireland Unlimited Company | Pyrazolopyrimidines substituees par cycloalkyle ayant une activite contre le vrs |
KR20210005569A (ko) * | 2018-04-23 | 2021-01-14 | 얀센 사이언시즈 아일랜드 언리미티드 컴퍼니 | Rsv에 대한 활성을 갖는 헤테로방향족 화합물 |
EP4171547A1 (fr) | 2020-05-27 | 2023-05-03 | Axial Therapeutics, Inc. | Composés modulateurs de tlr2, compositions pharmaceutiques et leurs utilisations |
Family Cites Families (51)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU4250596A (en) | 1994-12-22 | 1996-07-10 | Biochem Pharma Inc. | Low molecular weight bicyclic thrombin inhibitors |
WO1997001275A1 (fr) | 1995-06-29 | 1997-01-16 | Merck & Co., Inc. | Combinaisons d'inhibiteurs de farnesyl-proteine transferase |
ZA9610738B (en) | 1995-12-22 | 1997-06-24 | Warner Lambert Co | Subtype selective nmda receptor ligands and the use thereof |
US5972966A (en) | 1996-12-05 | 1999-10-26 | Merck & Co., Inc. | Inhibitors of farnesyl-protein transferase |
US5977134A (en) | 1996-12-05 | 1999-11-02 | Merck & Co., Inc. | Inhibitors of farnesyl-protein transferase |
US6177443B1 (en) | 1997-03-07 | 2001-01-23 | Novo Nordisk A/S | 4,5,6,7-tetrahydro-thieno[3, 2-C]pyridine derivatives, their preparation and use |
CA2375909A1 (fr) | 1999-07-19 | 2001-01-25 | Shionogi & Co., Ltd. | Composes tricycliques porteurs de pendants acyloxymethoxycarbonyle |
EP1113007A1 (fr) | 1999-12-24 | 2001-07-04 | Pfizer Inc. | Composés de tétrahydroisoquinoline comme agonistes/antagonistes d'oestrogène |
WO2003016274A2 (fr) | 2001-08-21 | 2003-02-27 | Sepracor, Inc. | Piperidines 2-substitue, ligands pour des recepteurs et des transporteurs de monoamines |
CA2483306A1 (fr) | 2002-04-23 | 2003-11-06 | Shionogi & Co., Ltd. | Derive de pyrazolo[1,5-a]pyrimidine et inhibiteur de la nad(p)h oxydase contenant ledit derive |
CA2499523C (fr) | 2002-09-20 | 2011-04-19 | Medisyn Technologies, Inc. | Agents therapeutiques et traitements correspondants |
EP1546132A1 (fr) | 2002-09-26 | 2005-06-29 | Pfizer Limited | Derives de pyrazole utilises en tant qu'inhibiteurs de la transcriptase inverse |
WO2004037817A1 (fr) | 2002-10-25 | 2004-05-06 | Mitsubishi Pharma Corporation | Composes de n-oxyde |
AR043633A1 (es) | 2003-03-20 | 2005-08-03 | Schering Corp | Ligandos de receptores de canabinoides |
EP2258365B1 (fr) | 2003-03-28 | 2013-05-29 | Novartis Vaccines and Diagnostics, Inc. | Utilisation de composés organiques pour potentialiser l'immunité |
FR2856596B1 (fr) | 2003-06-27 | 2007-04-27 | Bioprojet Soc Civ | Nouvelle association medicamenteuse psychiatrique et utilisation d'une antagoniste ou agoniste inverse du recepteur h3 de l'histamine pour preparer un medicament prevenant des effets indesirables de psychotropes. |
EP1671962A1 (fr) | 2003-10-10 | 2006-06-21 | Ono Pharmaceutical Co., Ltd. | Nouveau compose heterocyclique fondu et utilisation correspondante |
CA2541618C (fr) | 2003-10-30 | 2011-12-13 | Boehringer Ingelheim (Canada) Ltd. | Inhibiteurs polymerase rsv |
AR046959A1 (es) | 2003-12-18 | 2006-01-04 | Tibotec Pharm Ltd | Morfolinilo que contiene bencimidazoles como inhibidores de la replicacion del virus sincitial respiratorio |
KR20060127909A (ko) | 2003-12-24 | 2006-12-13 | 비오타 사이언티픽 매니지먼트 피티와이 엘티디 | 호흡기 다핵체 바이러스 감염 치료용 다환 물질 |
CN101775013A (zh) | 2004-09-13 | 2010-07-14 | 小野药品工业株式会社 | 含氮杂环衍生物及含有其作为活性成分的药物 |
EP2316458A1 (fr) | 2004-09-20 | 2011-05-04 | Xenon Pharmaceuticals Inc. | Derives de pyridazine destines a l'inhibition du desaturase-coa-stearoyl de l'humain |
WO2007044085A2 (fr) | 2005-05-19 | 2007-04-19 | Xenon Pharmaceuticals Inc. | Composes heteroaryle et leurs utilisations en tant qu'agents therapeutiques |
CA2612263C (fr) | 2005-06-20 | 2015-04-14 | Tibotec Pharmaceuticals Ltd. | 1-(2-amino-3-(alkyl substitue)-3h-benzimidazolylmethyl)-(3-subtitue)-1,3-dihydrobenzoimidazol-2-ones ayant une activite sur le virus syncyntial respiratoire |
US7507842B2 (en) | 2005-08-12 | 2009-03-24 | Radiorx, Inc. | Cyclic nitro compounds, pharmaceutical compositions thereof and uses thereof |
US20090111828A1 (en) | 2005-11-23 | 2009-04-30 | Astrazeneca Ab | L-alanine derivatives |
US20080176870A1 (en) | 2006-11-20 | 2008-07-24 | Bert Nolte | Heterobicyclic metalloprotease inhibitors |
AU2008287421A1 (en) | 2007-08-10 | 2009-02-19 | Glaxosmithkline Llc | Nitrogen containing bicyclic chemical entities for treating viral infections |
KR20100094554A (ko) | 2007-12-06 | 2010-08-26 | 쉐링 코포레이션 | 감마 세크레타제 조절인자 |
US20100063047A1 (en) | 2008-09-10 | 2010-03-11 | Kalypsys, Inc. | Aminopyrimidine inhibitors of histamine receptors for the treatment of disease |
CA2738453C (fr) | 2008-10-23 | 2017-07-04 | Boehringer Ingelheim International Gmbh | Derivees d'uree de nortropanes substitues, medicaments contenant de tels composes et leur utilisation |
US20100204265A1 (en) | 2009-02-09 | 2010-08-12 | Genelabs Technologies, Inc. | Certain Nitrogen Containing Bicyclic Chemical Entities for Treating Viral Infections |
WO2010104307A2 (fr) | 2009-03-07 | 2010-09-16 | 주식회사 메디젠텍 | Compositions pharmaceutiques pour traiter ou prévenir des maladies causées par la translocation de gsk3 du noyau cellulaire au cytoplasme, contenant des composés inhibant la translocation de gsk3 du noyau cellulaire au cytoplasme |
US9238647B2 (en) | 2009-03-23 | 2016-01-19 | Merck Sharp & Dohme Corp. | P2X3 receptor antagonists for treatment of pain |
JP5530514B2 (ja) | 2009-06-11 | 2014-06-25 | アッヴィ・バハマズ・リミテッド | Hcv感染を治療するための抗ウィルス化合物 |
US8937150B2 (en) | 2009-06-11 | 2015-01-20 | Abbvie Inc. | Anti-viral compounds |
EA201591390A1 (ru) * | 2010-06-24 | 2016-06-30 | Джилид Сайэнс, Инк. | Пиразол[1,5-a]пиримидины для противовирусного лечения |
EP2794611B1 (fr) | 2011-12-22 | 2017-10-11 | Gilead Sciences, Inc. | Pyrazolo[1,5]pyrimidines en tant qu'agents antiviraux |
CN106986869A (zh) * | 2012-04-17 | 2017-07-28 | 吉利德科学公司 | 用于抗病毒治疗的化合物和方法 |
JP6564380B2 (ja) | 2013-09-20 | 2019-08-21 | ユニバーシティ オブ ピッツバーグ − オブ ザ コモンウェルス システム オブ ハイヤー エデュケイション | 前立腺癌を治療するための化合物 |
JP6510539B2 (ja) | 2014-01-09 | 2019-05-08 | ザ ジェイ. デヴィッド グラッドストーン インスティテューツ, ア テスタメンタリー トラスト エスタブリッシュド アンダー ザ ウィル オブ ジェイ. デヴィッド グラッドストーン | 置換ベンゾオキサジン及び関連化合物 |
KR101551313B1 (ko) | 2014-07-28 | 2015-09-09 | 충남대학교산학협력단 | 신규한 인덴 유도체, 이의 제조방법 및 이를 유효성분으로 함유하는 망막 질환의 예방 또는 치료용 약학적 조성물 |
WO2016071293A2 (fr) | 2014-11-03 | 2016-05-12 | Iomet Pharma Ltd | Composé pharmaceutique |
EA032081B1 (ru) | 2014-12-08 | 2019-04-30 | Янссен Сайенсиз Айрлэнд Юси | ЗАМЕЩЕННЫЕ ПИПЕРИДИНОМ ПРОИЗВОДНЫЕ ПИРАЗОЛО[1,5-a]ПИРИМИДИНА С ИНГИБИРУЮЩЕЙ АКТИВНОСТЬЮ В ОТНОШЕНИИ РЕПЛИКАЦИИ РЕСПИРАТОРНО-СИНЦИТИАЛЬНОГО ВИРУСА (RSV) |
CN105777632A (zh) | 2015-01-09 | 2016-07-20 | 成都贝斯凯瑞生物科技有限公司 | 芳环并氮杂环衍生物及其应用 |
JO3637B1 (ar) | 2015-04-28 | 2020-08-27 | Janssen Sciences Ireland Uc | مركبات بيرازولو- وترايازولو- بيريميدين مضادة للفيروسات rsv |
TW201932470A (zh) | 2017-11-29 | 2019-08-16 | 愛爾蘭商健生科學愛爾蘭無限公司 | 具有抗rsv活性之吡唑并嘧啶 |
CA3087926A1 (fr) | 2018-01-31 | 2019-08-08 | Janssen Sciences Ireland Unlimited Company | Pyrazolopyrimidines substituees par cycloalkyle ayant une activite contre le vrs |
KR20210005569A (ko) | 2018-04-23 | 2021-01-14 | 얀센 사이언시즈 아일랜드 언리미티드 컴퍼니 | Rsv에 대한 활성을 갖는 헤테로방향족 화합물 |
JP2022507779A (ja) | 2018-11-26 | 2022-01-18 | ヤンセン・サイエンシズ・アイルランド・アンリミテッド・カンパニー | Rsvに対する活性を有するさらなるヘテロ芳香族化合物 |
WO2020234333A1 (fr) | 2019-05-23 | 2020-11-26 | Janssen Sciences Ireland Unlimited Company | Autres composés hétéroaromatiques ayant une activité contre le vrs |
-
2019
- 2019-04-19 KR KR1020207029130A patent/KR20210005569A/ko not_active Application Discontinuation
- 2019-04-19 ES ES19718707T patent/ES2957316T3/es active Active
- 2019-04-19 US US17/050,419 patent/US11708369B2/en active Active
- 2019-04-19 MA MA052348A patent/MA52348A/fr unknown
- 2019-04-19 WO PCT/EP2019/060216 patent/WO2019206828A1/fr active Application Filing
- 2019-04-19 EP EP19718707.3A patent/EP3784667B1/fr active Active
- 2019-04-19 CA CA3095277A patent/CA3095277A1/fr active Pending
- 2019-04-19 CN CN201980027482.0A patent/CN112004815A/zh active Pending
- 2019-04-19 EA EA202092439A patent/EA202092439A1/ru unknown
- 2019-04-19 AU AU2019260109A patent/AU2019260109B2/en active Active
- 2019-04-19 SG SG11202010323QA patent/SG11202010323QA/en unknown
- 2019-04-19 MX MX2020011200A patent/MX2020011200A/es unknown
- 2019-04-19 JP JP2020558603A patent/JP2021522222A/ja active Pending
Also Published As
Publication number | Publication date |
---|---|
ES2957316T3 (es) | 2024-01-17 |
AU2019260109B2 (en) | 2023-07-13 |
EP3784667A1 (fr) | 2021-03-03 |
MX2020011200A (es) | 2020-11-13 |
EP3784667B1 (fr) | 2023-08-16 |
CA3095277A1 (fr) | 2019-10-31 |
US20210094958A1 (en) | 2021-04-01 |
EA202092439A1 (ru) | 2021-03-05 |
WO2019206828A1 (fr) | 2019-10-31 |
CN112004815A (zh) | 2020-11-27 |
AU2019260109A1 (en) | 2020-09-17 |
KR20210005569A (ko) | 2021-01-14 |
SG11202010323QA (en) | 2020-11-27 |
US11708369B2 (en) | 2023-07-25 |
EP3784667C0 (fr) | 2023-08-16 |
JP2021522222A (ja) | 2021-08-30 |
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