LV13281B - Citalopram for the treatment of elevated blood pressure - Google Patents
Citalopram for the treatment of elevated blood pressure Download PDFInfo
- Publication number
- LV13281B LV13281B LVP-04-124A LV040124A LV13281B LV 13281 B LV13281 B LV 13281B LV 040124 A LV040124 A LV 040124A LV 13281 B LV13281 B LV 13281B
- Authority
- LV
- Latvia
- Prior art keywords
- citalopram
- blood pressure
- treatment
- use according
- patients
- Prior art date
Links
- 229960001653 citalopram Drugs 0.000 title claims abstract description 65
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- 230000036772 blood pressure Effects 0.000 title claims abstract description 61
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- WSEQXVZVJXJVFP-FQEVSTJZSA-N escitalopram Chemical compound C1([C@]2(C3=CC=C(C=C3CO2)C#N)CCCN(C)C)=CC=C(F)C=C1 WSEQXVZVJXJVFP-FQEVSTJZSA-N 0.000 claims description 29
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Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
- A61K31/343—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide condensed with a carbocyclic ring, e.g. coumaran, bufuralol, befunolol, clobenfurol, amiodarone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- External Artificial Organs (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
- Dental Preparations (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicinal Preparation (AREA)
Claims (10)
- LV 13281 IZGUDROJUMA FORMULA 1. Citaloprama vai tā farmaceitiski pieņemama sāļa izmantošana farmaceitiskas kompozīcijas pagatavošanai, kas ir derīga paaugstināta (augsta) asinsspiediena ārstēšanai, asins spiediena normalizēšanai vai asinsspiediena pazemināšanai un/vai paaugstināta asinsspiediena profilaksei. 10
- 2. Izmantošana saskaņā ar 1. punktu farmaceitiskas kompozīcijas pagatavošanai, kas ir derīga nestabila paaugstināta asinsspiediena ārstēšanai un/vai profilaksei.
- 3. Izmantošana saskaņā ar 1. vai 2. punktu farmaceitiskas kompozīcijas pagatavošanai, kas ir derīga paaugstināta asinsspiediena, kas rodas pacientiem ar traucējumiem panikas stāvoklī, ārstēšanai un/vai profilaksei.
- 4. Izmantošana saskaņā ar 1. punktu farmaceitiskas kompozīcijas pagatavošanai, kas ir derīga būtiski paaugstināta asinsspiediena ārstēšanai un/vai profilaksei.
- 5. Izmantošana saskaņā ar 1. punktu farmaceitiskas kompozīcijas 25 pagatavošanai, kas ir derīga insulta profilaksei un/vai ārstēšanai.
- 6. Izmantošana saskaņā ar jebkuru punktu no 1. līdz 5. punktam, kur tiek izmantots racēmisks citaloprams.
- 7. Izmantošana saskaņā ar jebkuru punktu no 1. līdz 5. punktam, kur tiek izmantots (S)-citaloprams.
- 8. Izmantošana saskaņā ar jebkuru punktu no 1. līdz 7. punktam, kur citaloprams vai tā farmaceitiski pieņemamais sāls tiek izmantots 35 kopā ar papildus antihipertensīvu līdzekli. 2
- 9. Izmantošana saskaņā ar 8. punktu, kur tiek izmatots vismaz viens no šādiem antihipertensīviem līdzekļiem: centrālās darbības antihipertensīvs līdzeklis, labāk metildopa, klonidīns, guanfacīns, 5 guanabenzs; β-blokators, labāk acebutolols, atenolols, betaksolols, bisoprolols, karteolols, propranolols, metoprolols, nadolols, penbutolols, pindolols, timolols, bucindolols, labetalols, karvedilols, nebivolols; α-blokators, labāk prazosīns, terazosīns, doksazosīns, trimazosīns, fenoksibenzamīds, fentolamīns; tiešās darbības 10 vazodilators, labāk hidralazīns, minoksidils, diazoksīds, fenoldopāms; kalcija kanālu blokators, labāk verapamils, diltiazems, nifedipīns, nimodipīns, felodipīns, nikardipīns, isradipīns, amlodipīns, nisoldipīns, lacidipīns; AKE inhibitors, labāk kaptoprils, enalaprils, lisinoprils, kvinaprils, ramiprils, benazeprils, fosinoprils, 15 moeksiprils, perindoprils, trandolaprils; angiotenzīna II receptoru antagonists, labāk losartāns, kandesartāns, irbesartāns, valsartāns, telmisartāns, eprosartāns; imidazolīna receptoru agonists, labāk moksonidīns, rilmenidīns.
- 10. Izmantošana saskaņā ar jebkuru punktu no 1. līdz 9. punktam, kur tiek pagatavotas farmaceitiskās kompozīcijas, kas satur vismaz vienu farmaceitiski pieņemamu inertu nesēju un/vai palīgvielu.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| HU0200980A HU0200980D0 (lv) | 2002-03-14 | 2002-03-14 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| LV13281B true LV13281B (en) | 2005-09-20 |
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ID=89980266
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| LVP-04-124A LV13281B (en) | 2002-03-14 | 2004-10-14 | Citalopram for the treatment of elevated blood pressure |
Country Status (35)
| Country | Link |
|---|---|
| US (1) | US7141604B2 (lv) |
| EP (1) | EP1490049B1 (lv) |
| JP (1) | JP2005519945A (lv) |
| KR (1) | KR100718368B1 (lv) |
| CN (1) | CN1259912C (lv) |
| AT (1) | ATE324887T1 (lv) |
| AU (1) | AU2003211195B2 (lv) |
| BG (1) | BG108904A (lv) |
| BR (1) | BR0303384A (lv) |
| CA (1) | CA2459834A1 (lv) |
| CY (1) | CY1106129T1 (lv) |
| CZ (1) | CZ2004661A3 (lv) |
| DE (1) | DE60305018T2 (lv) |
| DK (1) | DK1490049T3 (lv) |
| EA (1) | EA008350B1 (lv) |
| EE (1) | EE200400069A (lv) |
| ES (2) | ES2263009T3 (lv) |
| HK (1) | HK1075390A1 (lv) |
| HR (1) | HRP20040165B1 (lv) |
| HU (1) | HU0200980D0 (lv) |
| IL (2) | IL160486A0 (lv) |
| IS (1) | IS2392B (lv) |
| LT (1) | LT5255B (lv) |
| LV (1) | LV13281B (lv) |
| MX (1) | MXPA04008919A (lv) |
| NO (1) | NO20034998D0 (lv) |
| PL (1) | PL368902A1 (lv) |
| PT (1) | PT1490049E (lv) |
| SI (1) | SI1490049T1 (lv) |
| SK (1) | SK2222004A3 (lv) |
| TR (1) | TR200401036T1 (lv) |
| UA (1) | UA77506C2 (lv) |
| WO (1) | WO2003075914A1 (lv) |
| YU (1) | YU91203A (lv) |
| ZA (1) | ZA200408056B (lv) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ZA200601804B (en) * | 2003-10-10 | 2007-05-30 | Solvay Pharm Gmbh | Pharmaceutcal composition comprising a selective II imidazoline receptor agonist and an angiotensin II receptor blocker |
| DE102004002638A1 (de) * | 2004-01-19 | 2005-08-18 | Merck Patent Gmbh | Kombinationen von Serotonin-Wiederaufnahme-Hemmern und Imidazolin-I2-Agonisten |
| EP2008653A1 (de) * | 2007-06-28 | 2008-12-31 | Charité-Universitätsmedizin Berlin | Serotonerge Verbindungen zur Behandlung neuronaler Krankheiten |
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|---|---|---|---|---|
| GB1552012A (en) | 1975-12-16 | 1979-09-05 | Du Pont Canada | Process for the treatment of comminuted oats |
| PT1015416E (pt) * | 1997-07-08 | 2002-03-28 | Lundbeck & Co As H | Metodo para a producao de citalopram |
| JP3813820B2 (ja) * | 1997-11-11 | 2006-08-23 | ハー・ルンドベック・アクチエゼルスカベット | シタロプラムの製造方法 |
| US6333357B1 (en) * | 1999-11-05 | 2001-12-25 | Be Able, Llc | Behavior chemotherapy |
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2002
- 2002-03-14 HU HU0200980A patent/HU0200980D0/hu unknown
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2003
- 2003-03-13 CN CNB038012936A patent/CN1259912C/zh not_active Expired - Fee Related
- 2003-03-13 JP JP2003574189A patent/JP2005519945A/ja active Pending
- 2003-03-13 DK DK03743933T patent/DK1490049T3/da active
- 2003-03-13 MX MXPA04008919A patent/MXPA04008919A/es active IP Right Grant
- 2003-03-13 EP EP03743933A patent/EP1490049B1/en not_active Expired - Lifetime
- 2003-03-13 TR TR2004/01036T patent/TR200401036T1/xx unknown
- 2003-03-13 UA UA20041008333A patent/UA77506C2/uk unknown
- 2003-03-13 YU YU91203A patent/YU91203A/sh unknown
- 2003-03-13 CZ CZ2004661A patent/CZ2004661A3/cs unknown
- 2003-03-13 AU AU2003211195A patent/AU2003211195B2/en not_active Ceased
- 2003-03-13 SI SI200330354T patent/SI1490049T1/sl unknown
- 2003-03-13 IL IL16048603A patent/IL160486A0/xx not_active IP Right Cessation
- 2003-03-13 ES ES03743933T patent/ES2263009T3/es not_active Expired - Lifetime
- 2003-03-13 EA EA200401147A patent/EA008350B1/ru not_active IP Right Cessation
- 2003-03-13 DE DE60305018T patent/DE60305018T2/de not_active Expired - Fee Related
- 2003-03-13 AT AT03743933T patent/ATE324887T1/de not_active IP Right Cessation
- 2003-03-13 BR BR0303384-8A patent/BR0303384A/pt not_active IP Right Cessation
- 2003-03-13 KR KR1020047005264A patent/KR100718368B1/ko not_active IP Right Cessation
- 2003-03-13 PL PL03368902A patent/PL368902A1/xx not_active Application Discontinuation
- 2003-03-13 SK SK222-2004A patent/SK2222004A3/sk unknown
- 2003-03-13 WO PCT/HU2003/000021 patent/WO2003075914A1/en not_active IP Right Cessation
- 2003-03-13 EE EEP200400069A patent/EE200400069A/xx unknown
- 2003-03-13 ES ES200450048A patent/ES2238939B2/es not_active Expired - Fee Related
- 2003-03-13 CA CA002459834A patent/CA2459834A1/en not_active Abandoned
- 2003-03-13 PT PT03743933T patent/PT1490049E/pt unknown
- 2003-03-13 US US10/489,179 patent/US7141604B2/en not_active Expired - Lifetime
- 2003-11-10 NO NO20034998A patent/NO20034998D0/no not_active Application Discontinuation
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2004
- 2004-02-19 HR HR20040165A patent/HRP20040165B1/xx not_active IP Right Cessation
- 2004-02-19 IL IL160486A patent/IL160486A/en unknown
- 2004-05-12 LT LT2004049A patent/LT5255B/lt not_active IP Right Cessation
- 2004-08-20 IS IS7418A patent/IS2392B/is unknown
- 2004-10-06 ZA ZA200408056A patent/ZA200408056B/en unknown
- 2004-10-14 BG BG108904A patent/BG108904A/en unknown
- 2004-10-14 LV LVP-04-124A patent/LV13281B/en unknown
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2005
- 2005-06-29 HK HK05105529A patent/HK1075390A1/xx not_active IP Right Cessation
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2006
- 2006-07-20 CY CY20061101010T patent/CY1106129T1/el unknown
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