LV12585B - LONG-TERM CONTINUOUS ACTIVITY (PROLONGED ACTIVITY) PREPARATION FOR HEAD ANTAGONIST, ITS ACQUISITION AND APPLICATION - Google Patents

LONG-TERM CONTINUOUS ACTIVITY (PROLONGED ACTIVITY) PREPARATION FOR HEAD ANTAGONIST, ITS ACQUISITION AND APPLICATION Download PDF

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Publication number
LV12585B
LV12585B LVP-00-110A LV000110A LV12585B LV 12585 B LV12585 B LV 12585B LV 000110 A LV000110 A LV 000110A LV 12585 B LV12585 B LV 12585B
Authority
LV
Latvia
Prior art keywords
compound
group
sustained
acid
angiotensin
Prior art date
Application number
LVP-00-110A
Other languages
English (en)
Latvian (lv)
Other versions
LV12585A (en
Inventor
Yasutaka Igari
Akira Saikawa
Yoshiyuki Inada
Shigeru Kamei
Original Assignee
Takeda Chemical Industries, Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Takeda Chemical Industries, Ltd filed Critical Takeda Chemical Industries, Ltd
Publication of LV12585A publication Critical patent/LV12585A/xx
Publication of LV12585B publication Critical patent/LV12585B/en

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • A61K31/41781,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • A61K31/41841,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1611Inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1629Organic macromolecular compounds
    • A61K9/1641Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, poloxamers
    • A61K9/1647Polyesters, e.g. poly(lactide-co-glycolide)
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Inorganic Chemistry (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicinal Preparation (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
LVP-00-110A 1998-03-04 2000-08-16 LONG-TERM CONTINUOUS ACTIVITY (PROLONGED ACTIVITY) PREPARATION FOR HEAD ANTAGONIST, ITS ACQUISITION AND APPLICATION LV12585B (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP5236698 1998-03-04
PCT/JP1999/001011 WO1999044590A1 (en) 1998-03-04 1999-03-03 Sustained-release preparation for aii antagonist, production and use thereof

Publications (2)

Publication Number Publication Date
LV12585A LV12585A (en) 2000-12-20
LV12585B true LV12585B (en) 2001-03-20

Family

ID=12912818

Family Applications (1)

Application Number Title Priority Date Filing Date
LVP-00-110A LV12585B (en) 1998-03-04 2000-08-16 LONG-TERM CONTINUOUS ACTIVITY (PROLONGED ACTIVITY) PREPARATION FOR HEAD ANTAGONIST, ITS ACQUISITION AND APPLICATION

Country Status (21)

Country Link
US (2) US6589547B1 (es)
EP (1) EP1058541B1 (es)
KR (1) KR20010086245A (es)
CN (1) CN1291888A (es)
AT (1) ATE258430T1 (es)
AU (1) AU2745199A (es)
BR (1) BR9908474A (es)
CA (1) CA2318446C (es)
DE (1) DE69914460T2 (es)
EE (1) EE200000499A (es)
ES (1) ES2214013T3 (es)
HU (1) HUP0101439A3 (es)
ID (1) ID25640A (es)
IL (1) IL137979A0 (es)
LT (1) LT4800B (es)
LV (1) LV12585B (es)
NO (1) NO20004350L (es)
PL (1) PL342684A1 (es)
SK (1) SK11902000A3 (es)
WO (1) WO1999044590A1 (es)
ZA (1) ZA991706B (es)

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AU2001232348A1 (en) * 2000-02-21 2001-08-27 Takeda Chemical Industries Ltd. Sustained release preparations of physiologically active compound hardly solublein water and production process and use of the same
WO2002015935A1 (fr) * 2000-08-25 2002-02-28 Takeda Chemical Industries, Ltd. Agents de reduction du fibrinogene
US20040102502A1 (en) * 2000-10-25 2004-05-27 Toshifumi Watanabe Preventing/remedies for portal hypertension
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US20040219208A1 (en) * 2001-08-03 2004-11-04 Ryu Kawamura Sustained-release medicines
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CN101011393B (zh) * 2007-02-16 2010-10-06 广州柏赛罗药业有限公司 厄贝沙坦胃内滞留型缓释药物组合物
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Also Published As

Publication number Publication date
BR9908474A (pt) 2000-12-05
LT4800B (lt) 2001-06-25
SK11902000A3 (sk) 2001-02-12
NO20004350L (no) 2000-10-03
EP1058541B1 (en) 2004-01-28
ZA991706B (en) 2000-10-03
CA2318446A1 (en) 1999-09-10
US7294344B2 (en) 2007-11-13
EE200000499A (et) 2002-02-15
EP1058541A1 (en) 2000-12-13
US6589547B1 (en) 2003-07-08
ATE258430T1 (de) 2004-02-15
CA2318446C (en) 2008-09-23
HUP0101439A3 (en) 2002-09-30
US20030198676A1 (en) 2003-10-23
CN1291888A (zh) 2001-04-18
AU2745199A (en) 1999-09-20
NO20004350D0 (no) 2000-09-01
DE69914460T2 (de) 2004-10-28
PL342684A1 (en) 2001-07-02
WO1999044590A1 (en) 1999-09-10
DE69914460D1 (de) 2004-03-04
KR20010086245A (ko) 2001-09-10
LV12585A (en) 2000-12-20
IL137979A0 (en) 2001-10-31
HUP0101439A2 (hu) 2001-10-28
ES2214013T3 (es) 2004-09-01
LT2000082A (en) 2001-03-26
ID25640A (id) 2000-10-19

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