EE200000499A - Angiotensiin II antagonistliku toimega toimeainetprolongeeritult vabastav preparaat, selle valmistamise meetod ja kasutamine - Google Patents

Angiotensiin II antagonistliku toimega toimeainetprolongeeritult vabastav preparaat, selle valmistamise meetod ja kasutamine

Info

Publication number
EE200000499A
EE200000499A EEP200000499A EEP200000499A EE200000499A EE 200000499 A EE200000499 A EE 200000499A EE P200000499 A EEP200000499 A EE P200000499A EE P200000499 A EEP200000499 A EE P200000499A EE 200000499 A EE200000499 A EE 200000499A
Authority
EE
Estonia
Prior art keywords
preparation
angiotensin
prolonged
antagonist activity
release preparation
Prior art date
Application number
EEP200000499A
Other languages
English (en)
Inventor
Igari Yasutaka
Saikawa Akira
Inada Yoshiyuki
Kamei Shigeru
Original Assignee
Takeda Chemical Industries, Ltd.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Takeda Chemical Industries, Ltd. filed Critical Takeda Chemical Industries, Ltd.
Publication of EE200000499A publication Critical patent/EE200000499A/et

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4178—1,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4184—1,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1611—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1629—Organic macromolecular compounds
    • A61K9/1641—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, poloxamers
    • A61K9/1647—Polyesters, e.g. poly(lactide-co-glycolide)
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
EEP200000499A 1998-03-04 1999-03-03 Angiotensiin II antagonistliku toimega toimeainetprolongeeritult vabastav preparaat, selle valmistamise meetod ja kasutamine EE200000499A (et)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP5236698 1998-03-04
PCT/JP1999/001011 WO1999044590A1 (en) 1998-03-04 1999-03-03 Sustained-release preparation for aii antagonist, production and use thereof

Publications (1)

Publication Number Publication Date
EE200000499A true EE200000499A (et) 2002-02-15

Family

ID=12912818

Family Applications (1)

Application Number Title Priority Date Filing Date
EEP200000499A EE200000499A (et) 1998-03-04 1999-03-03 Angiotensiin II antagonistliku toimega toimeainetprolongeeritult vabastav preparaat, selle valmistamise meetod ja kasutamine

Country Status (21)

Country Link
US (2) US6589547B1 (et)
EP (1) EP1058541B1 (et)
KR (1) KR20010086245A (et)
CN (1) CN1291888A (et)
AT (1) ATE258430T1 (et)
AU (1) AU2745199A (et)
BR (1) BR9908474A (et)
CA (1) CA2318446C (et)
DE (1) DE69914460T2 (et)
EE (1) EE200000499A (et)
ES (1) ES2214013T3 (et)
HU (1) HUP0101439A3 (et)
ID (1) ID25640A (et)
IL (1) IL137979A0 (et)
LT (1) LT4800B (et)
LV (1) LV12585B (et)
NO (1) NO20004350L (et)
PL (1) PL342684A1 (et)
SK (1) SK11902000A3 (et)
WO (1) WO1999044590A1 (et)
ZA (1) ZA991706B (et)

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EP1413315A4 (en) * 2001-08-03 2006-08-16 Takeda Pharmaceutical DRUGS WITH CONTINUOUS RELEASE
BRPI0105509B8 (pt) * 2001-11-05 2021-05-25 Univ Minas Gerais formulações do peptídeo angiotensina-(1-7) usando as ciclodextrinas, lipossomas e o polímero plga
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CN101052402A (zh) * 2004-10-29 2007-10-10 兴和株式会社 肾小球疾病治疗剂
WO2006087394A1 (fr) * 2005-02-21 2006-08-24 Flamel Technologies Forme pharmaceutique orale de losartan
KR20070116648A (ko) * 2005-03-30 2007-12-10 다케다 야쿠힌 고교 가부시키가이샤 벤즈이미다졸 유도체 및 안지오텐신 ⅱ 길항제로서의 용도
KR20080039510A (ko) * 2005-08-22 2008-05-07 알렘빅 리미티드 발사르탄 제조 방법
GEP20125420B (en) * 2006-08-10 2012-03-26 Takeda Pharmaceutical Solid pharmaceutical composition comprising benzimidazole compound
EP1897537A1 (en) * 2006-09-04 2008-03-12 Novartis AG Composition comprising an angiotensin II receptor antagonist
PE20081364A1 (es) * 2006-09-04 2008-12-04 Novartis Ag Composicion farmaceutica que comprende valsartan
EP1908469A1 (en) 2006-10-06 2008-04-09 Boehringer Ingelheim Vetmedica Gmbh Angiotensin II receptor antagonist for the treatment of systemic diseases in cats
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Also Published As

Publication number Publication date
US7294344B2 (en) 2007-11-13
US20030198676A1 (en) 2003-10-23
DE69914460T2 (de) 2004-10-28
AU2745199A (en) 1999-09-20
ES2214013T3 (es) 2004-09-01
WO1999044590A1 (en) 1999-09-10
HUP0101439A2 (hu) 2001-10-28
CA2318446C (en) 2008-09-23
KR20010086245A (ko) 2001-09-10
LT2000082A (en) 2001-03-26
BR9908474A (pt) 2000-12-05
EP1058541B1 (en) 2004-01-28
NO20004350D0 (no) 2000-09-01
LV12585A (en) 2000-12-20
ATE258430T1 (de) 2004-02-15
SK11902000A3 (sk) 2001-02-12
CN1291888A (zh) 2001-04-18
PL342684A1 (en) 2001-07-02
DE69914460D1 (de) 2004-03-04
IL137979A0 (en) 2001-10-31
EP1058541A1 (en) 2000-12-13
ID25640A (id) 2000-10-19
ZA991706B (en) 2000-10-03
CA2318446A1 (en) 1999-09-10
NO20004350L (no) 2000-10-03
HUP0101439A3 (en) 2002-09-30
LT4800B (lt) 2001-06-25
US6589547B1 (en) 2003-07-08
LV12585B (en) 2001-03-20

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