LU85780A1 - Nouveaux esters enoliques precurseurs de medicaments et composition pharmaceutique les contenant - Google Patents

Nouveaux esters enoliques precurseurs de medicaments et composition pharmaceutique les contenant Download PDF

Info

Publication number
LU85780A1
LU85780A1 LU85780A LU85780A LU85780A1 LU 85780 A1 LU85780 A1 LU 85780A1 LU 85780 A LU85780 A LU 85780A LU 85780 A LU85780 A LU 85780A LU 85780 A1 LU85780 A1 LU 85780A1
Authority
LU
Luxembourg
Prior art keywords
methyl
carboxamide
dioxide
benzothiazine
pyridyl
Prior art date
Application number
LU85780A
Other languages
English (en)
French (fr)
Inventor
Joseph George Lombardino
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of LU85780A1 publication Critical patent/LU85780A1/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Rheumatology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Pain & Pain Management (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
LU85780A 1984-02-23 1985-02-20 Nouveaux esters enoliques precurseurs de medicaments et composition pharmaceutique les contenant LU85780A1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US58268484A 1984-02-23 1984-02-23
US58268484 1984-02-23

Publications (1)

Publication Number Publication Date
LU85780A1 true LU85780A1 (fr) 1985-12-11

Family

ID=24330094

Family Applications (1)

Application Number Title Priority Date Filing Date
LU85780A LU85780A1 (fr) 1984-02-23 1985-02-20 Nouveaux esters enoliques precurseurs de medicaments et composition pharmaceutique les contenant

Country Status (22)

Country Link
JP (1) JPS60184077A (xx)
KR (1) KR850006198A (xx)
AU (1) AU552478B2 (xx)
BE (1) BE901783A (xx)
DD (1) DD232045A5 (xx)
DE (1) DE3505576A1 (xx)
DK (1) DK81185A (xx)
ES (1) ES8606312A1 (xx)
FI (1) FI850742L (xx)
FR (1) FR2565980A1 (xx)
GB (1) GB2154585A (xx)
GR (1) GR850442B (xx)
HU (1) HUT37616A (xx)
IL (1) IL74407A0 (xx)
IT (1) IT1185514B (xx)
LU (1) LU85780A1 (xx)
NL (1) NL8500485A (xx)
NO (1) NO850725L (xx)
PL (1) PL252023A1 (xx)
PT (1) PT79988B (xx)
SE (1) SE8500889L (xx)
ZA (1) ZA851317B (xx)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4623486A (en) * 1985-05-29 1986-11-18 Pfizer Inc. [4-substituted benzoyloxy]-N-substituted-2H-1,2-benzothiazine-3-carboxamide 1,1-dioxides having anti-arthritic activity
US4610982A (en) * 1985-06-03 1986-09-09 Pfizer Inc. Anti-inflammatory benzo- and thieno-1,2-thiazine-3-carboxamide 1,1-dioxide derivatives, compositions, and method of use therefor
US20090221703A1 (en) 2006-07-09 2009-09-03 Chongxi Yu High penetration composition and uses thereof
US20090238763A1 (en) 2006-07-09 2009-09-24 Chongxi Yu High penetration compositions and uses thereof
CN101522692A (zh) * 2006-10-11 2009-09-02 于崇曦 具有快速皮肤穿透速度的带正电荷的水溶性的昔康及其相关化合物的前药
JP2010529101A (ja) 2007-06-04 2010-08-26 テックフィールズ インコーポレイテッド 非常に速い皮膚及び膜浸透速度を有するｎｓａｉａプロドラッグ及びその新規医薬使用
MX362949B (es) 2008-12-04 2019-02-27 Yu Chongxi Composiciones de alta penetracion y sus aplicaciones.

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3591574A (en) * 1968-05-29 1971-07-06 American Home Prod Tri-n-phenylglycyl derivatives of insulin
US3787324A (en) * 1971-03-01 1974-01-22 Warner Lambert Co 4-hydroxy-3-(3-isoxazolocarbamyl)-2h-1,2-benzothiazine 1,dioxides and process for their production
US3704298A (en) * 1971-06-22 1972-11-28 Warner Lambert Co 4-acyloxy-3-(2-isoxazolocarbamyl)-2h-1,2-benzothiazine 1,1-dioxides
AU518216B2 (en) * 1977-09-06 1981-09-17 Hafslund Nycomed Pharma Aktiengesellschaft Thienothiazine derivatives
JPS5714589A (en) * 1980-06-27 1982-01-25 Mitsui Toatsu Chem Inc Benzothiazine derivative, its preparation and drug composition
US4309427A (en) * 1981-01-15 1982-01-05 Pfizer Inc. Benzothiazine dioxide derivatives
IT8219486A0 (it) * 1982-02-05 1982-02-05 Chiesi Farma Spa Nuovi composti ad attivita'antiinfiammatoria, procedimento per la loro preparazione e relative composizioni farmaceutiche.
IT1206525B (it) * 1982-12-10 1989-04-27 Zionale S R L A Roma Preparato anti-infiammatorio nonsteroideo, per il trattamento delle affezioni artroreumatiche e metodo per la sua preparazione

Also Published As

Publication number Publication date
ZA851317B (en) 1986-10-29
BE901783A (fr) 1985-08-21
GB8504355D0 (en) 1985-03-20
FR2565980A1 (fr) 1985-12-20
GR850442B (xx) 1985-06-19
HUT37616A (en) 1986-01-23
NL8500485A (nl) 1985-09-16
DK81185D0 (da) 1985-02-22
FI850742A0 (fi) 1985-02-22
NO850725L (no) 1985-08-26
FI850742L (fi) 1985-08-24
DE3505576A1 (de) 1985-09-05
PT79988B (en) 1987-02-02
KR850006198A (ko) 1985-10-02
ES8606312A1 (es) 1986-04-16
AU3906685A (en) 1985-09-05
ES540590A0 (es) 1986-04-16
JPS60184077A (ja) 1985-09-19
DD232045A5 (de) 1986-01-15
SE8500889L (sv) 1985-08-24
IT8519585A0 (it) 1985-02-21
GB2154585A (en) 1985-09-11
IT1185514B (it) 1987-11-12
SE8500889D0 (sv) 1985-02-22
PT79988A (en) 1985-03-01
AU552478B2 (en) 1986-06-05
PL252023A1 (en) 1985-11-05
DK81185A (da) 1985-09-10
IL74407A0 (en) 1985-05-31

Similar Documents

Publication Publication Date Title
CA1194875A (fr) Procede pour la preparation de derive de la thieno [3,2-c] pyridine et les derives ainsi obtenus
EP0172096A1 (fr) Dérivés d'acylaminométhyl-3 imidazo[1,2-a]pyridines, leur préparation et leur application en thérapeutique
FR2645152A1 (fr) 3h-pteridinones-4, procedes de preparation et medicaments les contenant
EP0005689B1 (fr) Nouveaux acides lactame-N-acétiques et leurs amides, leurs procédés de préparation et compositions thérapeutiques
WO1997003987A1 (fr) Nouveaux derives de la galanthamine, leur procede de preparation, leur application comme medicaments et les compositions pharmaceutiques les renfermant
EP0151072B1 (fr) Dérivés de l'acide méthylènediphosphonique, procédé d'obtention et compositions pharmaceutiques antirhumatismales les contenant
FR2705095A1 (fr) Nouveaux indoles substitués, leur procédé de préparation et les compositions pharmaceutiques qui les contiennent.
EP0143123A2 (fr) Produits industriels nouveaux utilisés notamment comme intermédiaires dans la préparation de nouveaux dérivés du 4-hydroxy 3-quinoléine carboxamide substitués en 2 et la préparation desdits intermédiaires
LU85780A1 (fr) Nouveaux esters enoliques precurseurs de medicaments et composition pharmaceutique les contenant
EP0418933A1 (fr) Dérivés d'alcadiènes, leurs préparations, les médicaments les contenant et produits intermédiaires
EP0021940A1 (fr) Nouveaux dérivés aminés du benzothiazole, leur procédé de préparation et leur application en thérapeutique
EP0004494A1 (fr) Nouveaux dérivés de 1,3-dihydro 3-(1-(2-(2,3-dihydro 1,4-benzo-dioxin-2-yl)2-hydroxy éthyl)pipéridin-4-yl)2H-indol 2-one, leur procédé de préparation, leur application comme médicaments et les compositions pharmaceutiques les renfermant
EP0573318A1 (fr) Nouveaux dérivés de phényle carboxamide isoxazoles et leurs sels, leur procédé de préparation et les nouveaux intermédiaires de ce procédé, leur application comme médicaments et les compositions pharmaceutiques les renfermant
EP0459887A1 (fr) Dérivés N-pyrazolyl-ortho-dialkyl-benzamide doués d'activité anticonvulsivante, procédé de préparation et composition pharmaceutique
EP0463944A1 (fr) Acyl benzoxazolinones, leur procédé de préparation et les compositions pharmaceutiques qui les contiennent
BE861454A (fr) Derives d'acides thiazolidinecarboxyliques, leur preparation et leur utilisation
EP0196943B1 (fr) Nouveaux dérivés 8-thiotétrahydroquinoléines et leurs sels
CH633010A5 (fr) Derives de l'isoquinoleine, leur preparation et medicament qui les contient.
CA2010529A1 (fr) Derives de la 1-arylsulfonyl 2-piperidinone, leur procede et les intermediaires de preparation, leur application comme medicaments et les compositions les renfermant
EP0002635A1 (fr) Procédé de préparation de dérivés de thiéno (2,3-c) et (3,2-c) pyridines, nouveaux dérivés de la thiéno (2,3-c) pyridine obtenus et leur application thérapeutique
CA1266471A (fr) Derives du 4-morpholinyl 1h- indole et leurs sels, procede pour leur preparation et compositions pharmaceutiques les renfermant
EP0105881B1 (fr) Nouvelles cyanoguanidines, leur procede d'obtention et les compositions pharmaceutiques en renfermant
FR2585356A1 (fr) Nouveaux derives de l'acide 4-oh quinoleine carboxylique substitues en 2 par deux fonctions hydroxyle eventuellement etherifiees ou esterifiees, leurs procedes de preparation, les nouveaux intermediaires obtenus, leur application comme medicaments et les compositions les renfermant
EP0412014A1 (fr) Dérivés benzothiaziniques, leur préparation et leurs applications comme médicaments ou comme intermédiaires de synthèse de médicaments
LU85961A1 (fr) Nouveaux pro-medicaments heterocycliques d'oxicams anti-inflammatoires et leur procede de preparation