LTIP111A - Tam tikrų terapiškai aktyvių 4-pakeistų imidazolų panaudojimas perodinių farmacinių preparatų gamybai - Google Patents

Tam tikrų terapiškai aktyvių 4-pakeistų imidazolų panaudojimas perodinių farmacinių preparatų gamybai

Info

Publication number
LTIP111A
LTIP111A LTIP111A LTIP111A LTIP111A LT IP111 A LTIP111 A LT IP111A LT IP111 A LTIP111 A LT IP111A LT IP111 A LTIP111 A LT IP111A LT IP111 A LTIP111 A LT IP111A
Authority
LT
Lithuania
Prior art keywords
imidazoles
manufacture
pharmaceutical preparations
administered transdermally
certain therapeutically
Prior art date
Application number
LTIP111A
Other languages
English (en)
Inventor
Harry Jalonen
Arvo Sakari Risto Lammintausta
Original Assignee
Orion-Yhtymae Oy
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Orion-Yhtymae Oy filed Critical Orion-Yhtymae Oy
Publication of LTIP111A publication Critical patent/LTIP111A/lt
Publication of LT3005B publication Critical patent/LT3005B/lt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/70—Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
    • A61K9/7023—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
    • A61K9/703—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
    • A61K9/7038—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer
    • A61K9/7046—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds
    • A61K9/7069—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds obtained otherwise than by reactions only involving carbon to carbon unsaturated bonds, e.g. polysiloxane, polyesters, polyurethane, polyethylene oxide
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders

Landscapes

  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Dermatology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)

Abstract

Šis išradimas skirtas perodiniam preparatui, susidedančiam iš terapiškai aktyvaus junginio, apibrėžti formule@@@@@@ (I)@@@@@@@@arba@@@@@@@ (II)@@@@@@@@kurioje R1, R2 ir R3, gali būti vienodi arba skirtingi, yra H, CH3, C2H5 arba Cl; X yra CH=CH arba (CH2)n, kur n yra nuo 1 iki 3 arba X yra -C(OR5)H-, kur R5 yra metilas arba etilas; R4 yra vandenilis arba grynasis alkilas, turintis nuo 1 iki 4 anglies atomų. Perodinis junginių įvedimas gali būti atliekamas preparatais, paruoštais tepalo, emulsijos, pavilgo, tirpalo, kremo, drebučių arba perodinio tvarsčio pavidalo.
LTIP111A 1991-05-31 1992-05-29 Tam tikru terapiskai aktyviu 4-pakeistu imidazolu panaudojimas perodiniu farmaciniu preparatu gamybai LT3005B (lt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB9111773A GB2256135B (en) 1991-05-31 1991-05-31 Transdermal administration of 4-substituted imidazoles

Publications (2)

Publication Number Publication Date
LTIP111A true LTIP111A (lt) 1994-03-25
LT3005B LT3005B (lt) 1994-08-25

Family

ID=10695905

Family Applications (1)

Application Number Title Priority Date Filing Date
LTIP111A LT3005B (lt) 1991-05-31 1992-05-29 Tam tikru terapiskai aktyviu 4-pakeistu imidazolu panaudojimas perodiniu farmaciniu preparatu gamybai

Country Status (18)

Country Link
US (1) US5464628A (lt)
EP (1) EP0586467B1 (lt)
JP (1) JP3269822B2 (lt)
AT (1) ATE199317T1 (lt)
AU (1) AU1780892A (lt)
CA (1) CA2110162C (lt)
DE (1) DE69231709T2 (lt)
DK (1) DK0586467T3 (lt)
EE (1) EE02994B1 (lt)
ES (1) ES2154636T3 (lt)
FI (1) FI935350L (lt)
GB (1) GB2256135B (lt)
GR (1) GR3035499T3 (lt)
IE (1) IE66188B1 (lt)
LT (1) LT3005B (lt)
LV (1) LV10042B (lt)
NO (1) NO307365B1 (lt)
WO (1) WO1992021334A1 (lt)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU6821196A (en) * 1995-08-14 1997-03-12 Janssen Pharmaceutica N.V. Transdermal administration of vorozole
US5891461A (en) * 1995-09-14 1999-04-06 Cygnus, Inc. Transdermal administration of olanzapine
US5807570A (en) * 1995-09-29 1998-09-15 Cygnus, Inc. Transdermal administration of ropinirole and analogs thereof
GB9614098D0 (en) 1996-07-05 1996-09-04 Orion Yhtymae Oy Transdermal delivery of levosimendan
DE19820151A1 (de) * 1998-05-06 1999-11-11 Hexal Ag Transdermales therapeutisches System zur Anwendung von Candesartan
TW200306783A (en) 2002-04-29 2003-12-01 Fmc Corp Pesticidal heterocycles
FI20041425A0 (fi) * 2004-11-05 2004-11-05 Orion Corp Transmukosaalinen veterinäärinen koostumus
AU2004325626B2 (en) * 2004-12-15 2010-12-09 Drossapharm Ag External patches containing etofenamate
BRPI0706759A2 (pt) 2006-01-27 2011-04-05 Hofmann La Roche Ag F Uso de derivados de 4-imidazol para distúrbios do cns
ATE459251T1 (de) * 2006-08-08 2010-03-15 Intervet Int Bv Zusammensetzung für verstärkte antiparasitische wirksamkeit
US7795263B2 (en) * 2008-07-08 2010-09-14 Wildlife Laboratories, Inc. Pharmaceutical combination for and method of anesthetizing and immobilizing non-domesticated mammals
US20210323929A1 (en) * 2018-07-18 2021-10-21 Clexio Biosciences Ltd. Purified Detomidine, Process of Preparing and Methods of Use
CA3137267A1 (en) 2019-05-01 2020-11-05 Clexio Biosciences Ltd. Methods of treating pruritus
CN112220767B (zh) * 2020-09-25 2022-10-25 安徽省公众检验研究院有限公司 一种盐酸阿替美唑缓释片的制备方法

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU518569B2 (en) * 1979-08-07 1981-10-08 Farmos-Yhtyma Oy 4-benzyl- and 4-benzoyl imidazole derivatives
GB2069481B (en) * 1980-02-13 1983-07-27 Farmos Oy Substituted imidazole derivatives
GB2101114B (en) * 1981-07-10 1985-05-22 Farmos Group Ltd Substituted imidazole derivatives and their preparation and use
GB2167408B (en) 1984-11-23 1988-05-25 Farmos Oy Substituted imidazole derivatives and their preparation and use
US4672344A (en) 1985-04-19 1987-06-09 Siemens Aktiengesellschaft Polarized electromagnetic relay
FI864570A0 (fi) 1986-11-11 1986-11-11 Farmos Oy Terapeutiskt anvaendbar foerening.
US5124157A (en) * 1989-08-18 1992-06-23 Cygnus Therapeutic Systems Method and device for administering dexmedetomidine transdermally
FI894911A0 (fi) * 1989-10-17 1989-10-17 Farmos Oy En terapeutiskt vaerdefull foerening.
US5304569A (en) * 1989-11-13 1994-04-19 Orion-Yhtyma Oy Compositions and their use in lowering intraocular pressure

Also Published As

Publication number Publication date
LV10042A (lv) 1994-05-10
ATE199317T1 (de) 2001-03-15
EP0586467B1 (en) 2001-02-28
IE921938A1 (en) 1992-12-02
EE02994B1 (et) 1997-06-16
NO934261L (no) 1993-11-25
JP3269822B2 (ja) 2002-04-02
IE66188B1 (en) 1995-12-13
NO307365B1 (no) 2000-03-27
GB2256135B (en) 1995-01-18
GB9111773D0 (en) 1991-07-24
EP0586467A1 (en) 1994-03-16
LV10042B (en) 1995-02-20
CA2110162A1 (en) 1992-12-10
US5464628A (en) 1995-11-07
FI935350A7 (fi) 1993-11-30
ES2154636T3 (es) 2001-04-16
GB2256135A (en) 1992-12-02
GR3035499T3 (en) 2001-06-29
JPH06507618A (ja) 1994-09-01
WO1992021334A1 (en) 1992-12-10
NO934261D0 (no) 1993-11-25
DE69231709D1 (de) 2001-04-05
CA2110162C (en) 2002-11-12
FI935350A0 (fi) 1993-11-30
AU1780892A (en) 1993-01-08
LT3005B (lt) 1994-08-25
DK0586467T3 (da) 2001-03-26
DE69231709T2 (de) 2001-10-04
FI935350L (fi) 1993-11-30

Similar Documents

Publication Publication Date Title
LTIP111A (lt) Tam tikrų terapiškai aktyvių 4-pakeistų imidazolų panaudojimas perodinių farmacinių preparatų gamybai
KR900006318A (ko) 피페리디닐 벤즈이미다졸
CA2102454A1 (fr) Derives de l'erythromycine, leur procede de preparation, leur application comme medicaments
ES8107185A1 (es) Procedimiento para preparar piperidinas y pirrolidinas sus- tituidas
FR2452485A1 (fr) Nouveaux acides et esters 4-amino-3-quinoleinecarboxyliques, utiles notamment comme agents antisecretoires et anti-ulcere
KR910015562A (ko) 뇌부전 질환치료용 약제, 신규 2-(1-피페라지닐)-4-페닐시클로알카노 피리미딘 유도체, 및 그의 제법
RU94045799A (ru) СПОСОБ ПОЛУЧЕНИЯ β-ФЕНИЛИЗОСЕРИНА И ЕГО АНАЛОГОВ, СПОСОБ ПОЛУЧЕНИЯ ПРОИЗВОДНЫХ ТАКСАНА И ПРОМЕЖУТОЧНЫЕ СОЕДИНЕНИЯ СИНТЕЗА
KR960700213A (ko) 항-안드로겐성 일고리-및 이고리-알켄(Anti-androgenic cyclo and bicyclo alkenes)
KR890016017A (ko) 치환된 1-(1h-이미다졸-4-일)알킬-벤즈아미드
GB1062714A (en) -ß-(4'-acyloxy-4'-piperidyl)-ketones
FI104071B1 (fi) Analogiamenetelmä terapeuttisesti käyttökelpoisten 2,5-dihydro-2,5-diokso-1H-bents[b]atsepiinijohdannaisten valmistamiseksi
TNSN93107A1 (fr) Derives de piperidine, leur preparation et leur application en therapeutique
KR930019212A (ko) 피소스티그민 유도체와 이의 용도 및 이를 함유한 제약적 조제물
GB1421446A (en) Disalkylamino esters of benzopyranopyridines and compositions containing the same
ATE102051T1 (de) Arzneimittelzubereitungen.
AU687023B2 (en) Use of idazoxan and derivatives thereof in preparing a drug for treating parkinson's disease and its development
CA2116810A1 (fr) Utilisation de derives de la 6,6-dimethyl-2-acylcyclohex-4-en-1,3-diones dans le domaine cosmetique de la protection solaire, compositions les renfermant, nouveau derive et son procede de preparation
FR2360560A1 (fr) Derives du d-threo-1-phenyl-2-trifluoracetamido-1,3-propane-diol et leurs applications en tant qu'antibiotiques
KR900006287A (ko) 2-[4-(2-피페리디노-에톡시)-벤조일]-벤조산의 측쇄 알킬 에스테르, 이의 제조 방법 및 진경제로서의 이의 용도
JPS62201818A (ja) シクロペンテノン類を活性成分とするウイルス性皮膚疾患治療のための外用薬剤

Legal Events

Date Code Title Description
MM9A Lapsed patents

Effective date: 20060529