LT3028B - Benzodiazepine derivatives - Google Patents

Benzodiazepine derivatives Download PDF

Info

Publication number
LT3028B
LT3028B LTIP657A LTIP657A LT3028B LT 3028 B LT3028 B LT 3028B LT IP657 A LTIP657 A LT IP657A LT IP657 A LTIP657 A LT IP657A LT 3028 B LT3028 B LT 3028B
Authority
LT
Lithuania
Prior art keywords
compound
formula
hiv
compound according
thf
Prior art date
Application number
LTIP657A
Other languages
English (en)
Lithuanian (lt)
Inventor
Ming-Chu Hsu
Donna Mary Huryn
Steve Yik-Kai Tam
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of LTIP657A publication Critical patent/LTIP657A/xx
Publication of LT3028B publication Critical patent/LT3028B/lt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV

Landscapes

  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Virology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Communicable Diseases (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • AIDS & HIV (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
LTIP657A 1992-06-16 1993-06-15 Benzodiazepine derivatives LT3028B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US89919092A 1992-06-16 1992-06-16

Publications (2)

Publication Number Publication Date
LTIP657A LTIP657A (en) 1994-05-15
LT3028B true LT3028B (en) 1994-08-25

Family

ID=25410597

Family Applications (1)

Application Number Title Priority Date Filing Date
LTIP657A LT3028B (en) 1992-06-16 1993-06-15 Benzodiazepine derivatives

Country Status (21)

Country Link
EP (1) EP0574781A2 (xx)
JP (1) JPH0656825A (xx)
KR (1) KR940005612A (xx)
CN (1) CN1081442A (xx)
AU (1) AU4123093A (xx)
BG (1) BG97868A (xx)
BR (1) BR9302359A (xx)
CA (1) CA2098063A1 (xx)
CZ (1) CZ115893A3 (xx)
FI (1) FI932767A (xx)
HU (1) HUT64536A (xx)
IL (1) IL105977A0 (xx)
IS (1) IS4035A (xx)
LT (1) LT3028B (xx)
MX (1) MX9303422A (xx)
NO (1) NO932204L (xx)
PL (1) PL299312A1 (xx)
SI (1) SI9300288A (xx)
SK (1) SK61593A3 (xx)
UY (1) UY23600A1 (xx)
ZA (1) ZA934077B (xx)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6071895A (en) 1992-03-11 2000-06-06 Narhex Limited Polar-substituted hydrocarbons
DE69333270T2 (de) 1992-03-11 2004-08-05 Narhex Ltd. Aminderivate von oxo- und hydroxy- substituierten kohlenwasserstoffen
RU2126794C1 (ru) 1992-03-11 1999-02-27 Нархекс Лимитед Аминопроизводные оксо- или гидроксизамещенных гидразинов, способ их получения и фармацевтические композиции для ингибирования ретровирусной протеазы
US5888992A (en) 1992-03-11 1999-03-30 Narhex Limited Polar substituted hydrocarbons
IL110898A0 (en) * 1993-09-10 1994-11-28 Narhex Australia Pty Ltd Polar-substituted hydrocarbons
CN2504706Y (zh) * 2001-09-25 2002-08-07 闽祥实业有限公司 具有触摸控制功能的平板显示屏
WO2004103360A1 (ja) 2003-05-22 2004-12-02 Lead Chemical Co.,Ltd. 抗ウイルス作用を有する化合物および配合剤

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3398159A (en) 1961-06-20 1968-08-20 Hoffmann La Roche Aminophenyl heterocyclic ketones

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5141735A (en) * 1990-06-18 1992-08-25 Hoffman-La Roche, Inc. Substituted amino-benzodiazepines having anitviral activity
EP0475231A1 (en) * 1990-09-10 1992-03-18 F. Hoffmann-La Roche Ag Benzodiazepines
EP0491218A1 (en) * 1990-12-17 1992-06-24 F. Hoffmann-La Roche Ag Benzodiazepinones

Patent Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3398159A (en) 1961-06-20 1968-08-20 Hoffmann La Roche Aminophenyl heterocyclic ketones
US3400128A (en) 1961-06-20 1968-09-03 Hoffmann La Roche Heterocyclic intermediates
US3405122A (en) 1961-06-20 1968-10-08 Hoffmann La Roche Novel 3h-1, 4-benzodiazepin-2-(1h)-ones
US3407211A (en) 1961-06-20 1968-10-22 Hoffmann La Roche Acylaminophenyl heterocyclic ketones

Also Published As

Publication number Publication date
FI932767A (fi) 1993-12-17
NO932204L (no) 1993-12-17
EP0574781A2 (en) 1993-12-22
LTIP657A (en) 1994-05-15
HUT64536A (en) 1994-01-28
NO932204D0 (no) 1993-06-15
JPH0656825A (ja) 1994-03-01
BG97868A (en) 1994-05-27
SI9300288A (sl) 1993-12-31
HU9301704D0 (en) 1993-09-28
KR940005612A (ko) 1994-03-21
CA2098063A1 (en) 1993-12-17
EP0574781A3 (xx) 1994-04-06
IL105977A0 (en) 1993-10-20
FI932767A0 (fi) 1993-06-16
ZA934077B (en) 1993-12-16
PL299312A1 (en) 1994-01-10
UY23600A1 (es) 1993-12-09
CN1081442A (zh) 1994-02-02
CZ115893A3 (en) 1994-01-19
IS4035A (is) 1993-12-17
BR9302359A (pt) 1994-01-11
MX9303422A (es) 1994-06-30
AU4123093A (en) 1993-12-23
SK61593A3 (en) 1994-01-12

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MM9A Lapsed patents

Effective date: 19950615