KR910015570A - 시스 3-아미노-4-[2-(2-푸릴)에트-1-일]-1-메톡시카보닐메틸-아제티딘-2-온의 분해방법 - Google Patents

시스 3-아미노-4-[2-(2-푸릴)에트-1-일]-1-메톡시카보닐메틸-아제티딘-2-온의 분해방법 Download PDF

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Publication number
KR910015570A
KR910015570A KR1019910001905A KR910001905A KR910015570A KR 910015570 A KR910015570 A KR 910015570A KR 1019910001905 A KR1019910001905 A KR 1019910001905A KR 910001905 A KR910001905 A KR 910001905A KR 910015570 A KR910015570 A KR 910015570A
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KR
South Korea
Prior art keywords
methoxycarbonylmethyl
azetidin
eth
furyl
amino
Prior art date
Application number
KR1019910001905A
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English (en)
Inventor
알란 릭크 Ⅲ세 존
글래스비 라이트 이안
Original Assignee
리로이 휘테커
일라이 릴리 앤드 캄파니
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 리로이 휘테커, 일라이 릴리 앤드 캄파니 filed Critical 리로이 휘테커
Publication of KR910015570A publication Critical patent/KR910015570A/ko

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

내용 없음

Description

시스 3-아미노-4-[2-(2-푸릴)에트-1-일]-1-메톡시카보닐메틸-아제티딘-2-온의 분해방법
본 내용은 요부공개 건이므로 전문내용을 수록하지 않았음

Claims (4)

  1. (a) 용매중의 시스 /ββ-3-아미노-4-[2-(2-푸릴)에트-1-일]-1-메톡시카보닐메틸-아제티딘-2-온라세메이트 용액을 적어도 약 0.5 몰당량의 (-)-2, 3 : 4, 6-디-0-이소프로필리덴-2-케토-L-굴론산 수화물과 접촉시키고; (b) 상기에 의해 형성된,-이성체의 불용성 (-)-2, 3 : 4, 6-디-0-이소프로필리덴-2-케도-L-굴론산 수화물 염을 분리시키는 단계를 포함하는, 시스 /ββ-3-아미노-4-[2-(2-푸릴)에트-1-일]-1-메톡시카보닐메틸-아제티딘-2-온을 그의 구성 에난티오머로 분해시키는 방법.
  2. 제1항에 있어서, 사용된 극성 유기 용매가 이소프로판올인 방법.
  3. 제1항에 있어서, 사용된 극성 유기 용매가 햅탄과 이소프로판올의 혼합물인 방법.
  4. 시스 -3-아미노-4-[2-(2-푸릴)에트-1-일]-1-메톡시카보닐메틸-아제티딘-2-온의 (-)-2, 3 : 4, 6-디-0-이소프로필리덴-2-케톤-L-굴론산 수화물 염.
    ※ 참고사항 : 최초출원 내용에 의하여 공개하는 것임.
KR1019910001905A 1990-02-06 1991-02-04 시스 3-아미노-4-[2-(2-푸릴)에트-1-일]-1-메톡시카보닐메틸-아제티딘-2-온의 분해방법 KR910015570A (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US07/475,515 1990-02-06
US07/475,515 US5030725A (en) 1990-02-06 1990-02-06 Method of resolving cis 3-amino-4-[2-(2-furyl)eth-1-yl]-1-methoxycarbonylmethyl-azetidin-2-one using (-)-DAG

Publications (1)

Publication Number Publication Date
KR910015570A true KR910015570A (ko) 1991-09-30

Family

ID=23887896

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019910001905A KR910015570A (ko) 1990-02-06 1991-02-04 시스 3-아미노-4-[2-(2-푸릴)에트-1-일]-1-메톡시카보닐메틸-아제티딘-2-온의 분해방법

Country Status (18)

Country Link
US (1) US5030725A (ko)
EP (1) EP0441543A1 (ko)
JP (1) JPH04211079A (ko)
KR (1) KR910015570A (ko)
CN (1) CN1023703C (ko)
AU (1) AU628708B2 (ko)
CA (1) CA2035550A1 (ko)
FI (1) FI910553A (ko)
HU (1) HUT60705A (ko)
IE (1) IE910382A1 (ko)
IL (1) IL97139A0 (ko)
MX (1) MX166218B (ko)
NO (1) NO910426L (ko)
NZ (1) NZ237002A (ko)
PT (1) PT96662A (ko)
RU (1) RU1797611C (ko)
YU (1) YU19591A (ko)
ZA (1) ZA91778B (ko)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2751811B1 (fr) * 1996-07-24 1998-10-09 Matra Communication Procede de demodulation numerique
DE19710862A1 (de) 1997-03-15 1998-09-17 Itt Mfg Enterprises Inc Hydraulische, mit Fremdkraft betätigbare Bremsanlage
WO2009147430A1 (en) 2008-06-02 2009-12-10 Generics [Uk] Limited A process for the preparation of enantiomerically pure amines
AR110150A1 (es) * 2016-11-09 2019-02-27 Roivant Sciences Gmbh Procesos para la preparación de inhibidores de tph1

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3904632A (en) * 1972-05-08 1975-09-09 Hoffmann La Roche (')-di-o-isopropylidene-2-keto-l-gulonates
US4167581A (en) * 1972-12-15 1979-09-11 Imperial Chemical Industries Limited Alkanolamine derivatives and pharmaceutical compositions and uses thereof
US4711887A (en) * 1982-04-23 1987-12-08 Imperial Chemical Industries Plc Hydrazinopyridazine compounds
US4665171A (en) * 1985-07-17 1987-05-12 Harvard University Process and intermediates for β-lactam antibiotics
US4931556A (en) * 1988-10-17 1990-06-05 Eli Lilly And Company Method of resolving cis 3-amino-4-(2-(2-furyl)eth-1-yl)-methoxycarbonylmethyl-azetidin-2-one and malic acid salts thereof
US4931557A (en) * 1988-10-17 1990-06-05 Eli Lilly And Company Method of resolving cis 3-amino-4-(2-furyl)vinyl)-1-methoxycarbonylmethyl-azetidin-2-one and di-p-toluoyl-tartaric acid salts thereof
US4923983A (en) * 1989-07-31 1990-05-08 Eli Lilly And Company Method of resolving cis 3-amino-4-[2-(2-furyl)eth-1-yl]-1-methoxycarbonylmethyl-azetidin-2-one
US4983983A (en) * 1989-12-05 1991-01-08 The United States Of America As Represented By The Secretary Of The Navy Semi-automatic direction finding set

Also Published As

Publication number Publication date
HUT60705A (en) 1992-10-28
NO910426L (no) 1991-08-07
PT96662A (pt) 1991-10-31
HU910392D0 (en) 1991-08-28
US5030725A (en) 1991-07-09
NZ237002A (en) 1992-06-25
IE910382A1 (en) 1991-08-14
AU7024191A (en) 1991-08-08
MX166218B (es) 1992-12-23
FI910553A0 (fi) 1991-02-05
FI910553A (fi) 1991-08-07
NO910426D0 (no) 1991-02-04
CN1053920A (zh) 1991-08-21
YU19591A (sh) 1994-01-20
JPH04211079A (ja) 1992-08-03
ZA91778B (en) 1992-10-28
IL97139A0 (en) 1992-05-25
CA2035550A1 (en) 1991-08-07
EP0441543A1 (en) 1991-08-14
CN1023703C (zh) 1994-02-09
AU628708B2 (en) 1992-09-17
RU1797611C (ru) 1993-02-23

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