KR900006323A - 시스 3-아미노-4-[2-(2-푸릴)에트-1-일]-1-메톡시카보닐메틸-아제티딘-2-온의 분할방법 및 그의 말산염. - Google Patents
시스 3-아미노-4-[2-(2-푸릴)에트-1-일]-1-메톡시카보닐메틸-아제티딘-2-온의 분할방법 및 그의 말산염. Download PDFInfo
- Publication number
- KR900006323A KR900006323A KR1019890014916A KR890014916A KR900006323A KR 900006323 A KR900006323 A KR 900006323A KR 1019890014916 A KR1019890014916 A KR 1019890014916A KR 890014916 A KR890014916 A KR 890014916A KR 900006323 A KR900006323 A KR 900006323A
- Authority
- KR
- South Korea
- Prior art keywords
- malic acid
- cis
- azetidin
- eth
- furyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
내용 없음
Description
본 내용은 요부공개 건이므로 전문내용을 수록하지 않았음
Claims (6)
- (a)시스 αα/ββ 라세메이트의 극성 유기 용액을 광학적 활성인 말산 적어도 약 0.5몰-당량을 접촉시키고 ; (b) 이에 의해 생성된 불용성 염을 분리시키는 단계들을 포함하는, 시스 αα/ββ-3-아미노-4-[2-(2-푸릴)에트-1-일]-1-메톡시카보닐메틸-아제티딘-2-온을 그의 성분 에난티오머들로 분할하는 방법.
- 제 1 항에 있어서, 상기 이용된 극성 유기 용매나 테트라하이드로 푸란인 방법.
- 제 2 항에 있어서, 분할제로서 S(-)-말산이 이용되는 방법.
- 제 2 항에 있어서, 분할제로서 R(+)-말산이 이용되는 방법.
- 시스 ββ-3-아미노-4-[2-(2-푸릴)에트-1-일]-1-메톡시카보닐메틸-아제티딘-2-온의 S(-)-말산 염.
- 시스 αα-3-아미노-4-[2-(2-푸릴)에트-1-일]-1-메톡시 카보닐메틸-아제티딘-2-온의 R(+)-말산 염.※ 참고사항 : 최초출원 내용에 의하여 공개하는 것임.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US07/258,919 US4931556A (en) | 1988-10-17 | 1988-10-17 | Method of resolving cis 3-amino-4-(2-(2-furyl)eth-1-yl)-methoxycarbonylmethyl-azetidin-2-one and malic acid salts thereof |
US258,919 | 1999-03-01 |
Publications (1)
Publication Number | Publication Date |
---|---|
KR900006323A true KR900006323A (ko) | 1990-05-07 |
Family
ID=22982693
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
KR1019890014916A KR900006323A (ko) | 1988-10-17 | 1989-10-17 | 시스 3-아미노-4-[2-(2-푸릴)에트-1-일]-1-메톡시카보닐메틸-아제티딘-2-온의 분할방법 및 그의 말산염. |
Country Status (11)
Country | Link |
---|---|
US (1) | US4931556A (ko) |
EP (1) | EP0365212B1 (ko) |
JP (1) | JPH02169589A (ko) |
KR (1) | KR900006323A (ko) |
AT (1) | ATE116313T1 (ko) |
DE (1) | DE68920264T2 (ko) |
ES (1) | ES2065395T3 (ko) |
GR (1) | GR3015506T3 (ko) |
HU (1) | HU207312B (ko) |
IE (1) | IE65410B1 (ko) |
IL (1) | IL91959A0 (ko) |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6587567B1 (en) | 1997-01-06 | 2003-07-01 | Murata Manufacturing Co., Ltd. | Piezoelectric electroacoustic transducer |
Families Citing this family (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5030725A (en) * | 1990-02-06 | 1991-07-09 | Eli Lilly And Company | Method of resolving cis 3-amino-4-[2-(2-furyl)eth-1-yl]-1-methoxycarbonylmethyl-azetidin-2-one using (-)-DAG |
US5057607A (en) * | 1990-06-08 | 1991-10-15 | Eli Lilly And Company | Enantiomerically selective biocatalyzed acylation |
US5159073A (en) * | 1990-09-13 | 1992-10-27 | Eli Lilly And Company | Intermediates to 1-carbacephalosporins and process for preparation thereof |
EP0479431B1 (en) * | 1990-09-13 | 1999-12-08 | Eli Lilly And Company | Intermediates to 1-carbacephalosporins and process for preparation thereof |
US5225553A (en) * | 1990-09-13 | 1993-07-06 | Eli Lilly And Company | Intermediates to 1-carbacephalosporins and process for preparation thereof |
US5142038A (en) * | 1991-07-23 | 1992-08-25 | Eli Lilly And Company | Process of enantiomeric separation of carbacephem intermediates |
TW372244B (en) * | 1993-07-29 | 1999-10-21 | Ciba Sc Holding Ag | Process for producing novel finely divided highly transparent diketopyrrolopyrrole pigments |
DE59409750D1 (de) * | 1993-07-29 | 2001-06-21 | Ciba Sc Holding Ag | Neue feinteilige cyansubstituierte Diketopyrrolopyrrolpigmente und Herstellung derselben |
US6617451B1 (en) | 1999-07-23 | 2003-09-09 | Eli Lilly And Company | Enantioselective acylation of cis racemic azetidinones |
NZ583970A (en) | 2007-10-11 | 2011-04-29 | Univ California | Compositions and methods of inhibiting n-acylethanolamine-hydrolyzing acid amidase |
WO2014144836A2 (en) | 2013-03-15 | 2014-09-18 | The Regents Of The University Of California | Carbamate derivatives of lactam based n-acylethanolamine acid amidase (naaa) inhibitors |
WO2014144547A2 (en) | 2013-03-15 | 2014-09-18 | The Regents Of The University Of California | Amide derivatives of lactam based n-acylethanolamine acid amidase (naaa) inhibitors |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS4834736B1 (ko) * | 1969-05-14 | 1973-10-23 | ||
FR2229401A1 (en) * | 1973-05-17 | 1974-12-13 | Medimac Sa | Optical resolution of rotoxamine - using dextro-maleic acid and direct pptn. of the laevo-rotoxamine-dextro-maleate salt useful as an antihistamine |
JPS5310974B2 (ko) * | 1974-06-10 | 1978-04-18 | ||
US4727146A (en) * | 1980-07-03 | 1988-02-23 | The United States Of America As Represented By The Department Of Health And Human Services | Synthesis of chiral 1-benzyl-1,2,3,4-tetra-hydroisoquinolines by asymmetric reduction |
US4665171A (en) * | 1985-07-17 | 1987-05-12 | Harvard University | Process and intermediates for β-lactam antibiotics |
-
1988
- 1988-10-17 US US07/258,919 patent/US4931556A/en not_active Expired - Fee Related
-
1989
- 1989-10-12 IL IL91959A patent/IL91959A0/xx not_active IP Right Cessation
- 1989-10-12 EP EP89310446A patent/EP0365212B1/en not_active Expired - Lifetime
- 1989-10-12 AT AT89310446T patent/ATE116313T1/de not_active IP Right Cessation
- 1989-10-12 DE DE68920264T patent/DE68920264T2/de not_active Expired - Fee Related
- 1989-10-12 ES ES89310446T patent/ES2065395T3/es not_active Expired - Lifetime
- 1989-10-16 IE IE332289A patent/IE65410B1/en not_active IP Right Cessation
- 1989-10-16 HU HU895327A patent/HU207312B/hu not_active IP Right Cessation
- 1989-10-16 JP JP1270146A patent/JPH02169589A/ja active Pending
- 1989-10-17 KR KR1019890014916A patent/KR900006323A/ko not_active Application Discontinuation
-
1995
- 1995-03-20 GR GR950400637T patent/GR3015506T3/el unknown
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6587567B1 (en) | 1997-01-06 | 2003-07-01 | Murata Manufacturing Co., Ltd. | Piezoelectric electroacoustic transducer |
Also Published As
Publication number | Publication date |
---|---|
HU895327D0 (ko) | 1990-01-28 |
IL91959A0 (en) | 1990-07-12 |
GR3015506T3 (en) | 1995-06-30 |
EP0365212A2 (en) | 1990-04-25 |
IE65410B1 (en) | 1995-10-18 |
US4931556A (en) | 1990-06-05 |
HU207312B (en) | 1993-03-29 |
HUT58077A (en) | 1992-01-28 |
DE68920264T2 (de) | 1995-05-24 |
JPH02169589A (ja) | 1990-06-29 |
ATE116313T1 (de) | 1995-01-15 |
EP0365212A3 (en) | 1991-11-06 |
IE893322L (en) | 1990-04-17 |
DE68920264D1 (de) | 1995-02-09 |
EP0365212B1 (en) | 1994-12-28 |
ES2065395T3 (es) | 1995-02-16 |
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