KR910000855B1 - 아릴히드록사메이트 및 그의 제조방법 - Google Patents

아릴히드록사메이트 및 그의 제조방법 Download PDF

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Publication number
KR910000855B1
KR910000855B1 KR1019850003374A KR850003374A KR910000855B1 KR 910000855 B1 KR910000855 B1 KR 910000855B1 KR 1019850003374 A KR1019850003374 A KR 1019850003374A KR 850003374 A KR850003374 A KR 850003374A KR 910000855 B1 KR910000855 B1 KR 910000855B1
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KR
South Korea
Prior art keywords
compound
formula
group
hydroxy
alkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
KR1019850003374A
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English (en)
Korean (ko)
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KR850008660A (ko
Inventor
에스. 카라뉴스키 도날드
에프. 하스랜거 마틴
Original Assignee
이이. 아르. 스퀴부 앤드 산즈 인코오포레이티드
죠오지 제이. 코에서
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Application filed by 이이. 아르. 스퀴부 앤드 산즈 인코오포레이티드, 죠오지 제이. 코에서 filed Critical 이이. 아르. 스퀴부 앤드 산즈 인코오포레이티드
Publication of KR850008660A publication Critical patent/KR850008660A/ko
Application granted granted Critical
Publication of KR910000855B1 publication Critical patent/KR910000855B1/ko
Expired legal-status Critical Current

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C65/00—Compounds having carboxyl groups bound to carbon atoms of six—membered aromatic rings and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
    • C07C65/21—Compounds having carboxyl groups bound to carbon atoms of six—membered aromatic rings and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups containing ether groups, groups, groups, or groups
    • C07C65/24—Compounds having carboxyl groups bound to carbon atoms of six—membered aromatic rings and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups containing ether groups, groups, groups, or groups polycyclic
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C235/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms
    • C07C235/42—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings and singly-bound oxygen atoms bound to the same carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C63/00—Compounds having carboxyl groups bound to a carbon atoms of six-membered aromatic rings
    • C07C63/04—Monocyclic monocarboxylic acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C65/00—Compounds having carboxyl groups bound to carbon atoms of six—membered aromatic rings and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
    • C07C65/21—Compounds having carboxyl groups bound to carbon atoms of six—membered aromatic rings and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups containing ether groups, groups, groups, or groups
    • C07C65/24—Compounds having carboxyl groups bound to carbon atoms of six—membered aromatic rings and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups containing ether groups, groups, groups, or groups polycyclic
    • C07C65/26—Compounds having carboxyl groups bound to carbon atoms of six—membered aromatic rings and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups containing ether groups, groups, groups, or groups polycyclic containing rings other than six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C65/00—Compounds having carboxyl groups bound to carbon atoms of six—membered aromatic rings and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
    • C07C65/21—Compounds having carboxyl groups bound to carbon atoms of six—membered aromatic rings and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups containing ether groups, groups, groups, or groups
    • C07C65/28—Compounds having carboxyl groups bound to carbon atoms of six—membered aromatic rings and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups containing ether groups, groups, groups, or groups having unsaturation outside the aromatic rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
KR1019850003374A 1984-05-17 1985-05-17 아릴히드록사메이트 및 그의 제조방법 Expired KR910000855B1 (ko)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US61125184A 1984-05-17 1984-05-17
US611251 1984-05-17
US611251/84 1984-05-17
US06/719,935 US4607053A (en) 1984-05-17 1985-04-04 Arylhydroxamates useful as antiallergy agents
US719935 1985-04-04

Publications (2)

Publication Number Publication Date
KR850008660A KR850008660A (ko) 1985-12-21
KR910000855B1 true KR910000855B1 (ko) 1991-02-11

Family

ID=27086475

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019850003374A Expired KR910000855B1 (ko) 1984-05-17 1985-05-17 아릴히드록사메이트 및 그의 제조방법

Country Status (13)

Country Link
US (1) US4607053A (enExample)
EP (1) EP0161939B1 (enExample)
KR (1) KR910000855B1 (enExample)
AU (1) AU586973B2 (enExample)
DE (1) DE3587460T2 (enExample)
DK (1) DK217385A (enExample)
ES (7) ES8609201A1 (enExample)
FI (1) FI851970A7 (enExample)
GR (1) GR851203B (enExample)
HU (1) HU200594B (enExample)
IL (1) IL75223A (enExample)
NZ (1) NZ212099A (enExample)
PH (1) PH21267A (enExample)

Families Citing this family (31)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8531839D0 (en) * 1985-12-30 1986-02-05 Wellcome Found Aryl derivatives
IL78157A (en) * 1985-03-16 1989-08-15 Wellcome Found Aryl derivatives,their preparation and pharmaceutical compositions containing them
IE59397B1 (en) * 1985-03-16 1994-02-23 Wellcome Found New aryl derivatives
US5036157A (en) * 1986-03-11 1991-07-30 Burroughs Wellcome Co. Aryl derivatives
US4761403A (en) * 1986-04-09 1988-08-02 Abbott Laboratories Lipoxygenase inhibiting compounds
GB8609282D0 (en) * 1986-04-16 1986-05-21 Roussel Lab Ltd Chemical compounds
US4906667A (en) * 1986-07-30 1990-03-06 E. R. Squibb & Sons, Inc. Phenyl hydroxamic acids including a hetero-containing substituent
GB8619593D0 (en) * 1986-08-12 1986-09-24 Roussel Lab Ltd Chemical compounds
US4769461A (en) * 1986-09-16 1988-09-06 American Home Products Corporation Quinolinyl benzene hydroxamic acids as anti-inflammatory/antiallergic agents
US4681894A (en) * 1986-09-26 1987-07-21 Ortho Pharmaceutical Corporation Hydroxamic acids and esters
US4731382A (en) * 1986-12-29 1988-03-15 Bristol-Myers Company Lipoxygenase inhibitory phenylalkanohydroxamic acids
US4873259A (en) * 1987-06-10 1989-10-10 Abbott Laboratories Indole, benzofuran, benzothiophene containing lipoxygenase inhibiting compounds
US4822809A (en) * 1987-11-13 1989-04-18 Abbott Laboratories Benzazole lipoxygenase inhibiting compounds
GB2212153B (en) * 1987-11-16 1992-01-15 Squibb & Sons Inc Phenyl hydroxamic acids
EP0588785A1 (en) * 1989-03-30 1994-03-30 Abbott Laboratories Urea based lipoxygenase inhibiting compounds
US5028629A (en) * 1990-03-28 1991-07-02 Eli Lilly And Company 5-Lipoxygenase inhibitors
WO1997048694A1 (en) 1996-06-20 1997-12-24 Board Of Regents, The University Of Texas System Compounds and methods for providing pharmacologically active preparations and uses thereof
US8026280B2 (en) 2001-03-27 2011-09-27 Errant Gene Therapeutics, Llc Histone deacetylase inhibitors
US7312247B2 (en) 2001-03-27 2007-12-25 Errant Gene Therapeutics, Llc Histone deacetylase inhibitors
US7842727B2 (en) * 2001-03-27 2010-11-30 Errant Gene Therapeutics, Llc Histone deacetylase inhibitors
US6495719B2 (en) * 2001-03-27 2002-12-17 Circagen Pharmaceutical Histone deacetylase inhibitors
DE10222561B4 (de) 2002-05-17 2009-12-10 Dr. Franz Köhler Chemie GmbH Protektive Lösung zur Verhinderung von Ischämieschäden
EP1511477A4 (en) * 2002-05-22 2008-04-09 Errant Gene Therapeutics Llc HISTONE DEACETYLASE INHIBITORS BASED ON ALPHA-KETO-EPOXYDE COMPOUNDS
JP2006508986A (ja) * 2002-11-20 2006-03-16 エルラント ゲネ セラペウチクス エルエルシー ヒストンデアセチラーゼ阻害剤による肺細胞の治療方法
US7511171B2 (en) * 2004-04-01 2009-03-31 Sumitomo Chemical Company, Limited Method for producing carboxylic acid compound
WO2006052916A2 (en) * 2004-11-08 2006-05-18 Errant Gene Therapeutics, Inc. Histone deacetylase inhibitors
CN108697091B (zh) 2016-01-25 2021-07-23 美国陶氏益农公司 具有杀虫效用的分子，以及与其相关的中间体、组合物和方法
TWI780112B (zh) 2017-03-31 2022-10-11 美商科迪華農業科技有限責任公司 具有殺蟲效用之分子，及其相關之中間物、組成物暨方法
CN114524753B (zh) * 2022-02-24 2024-03-26 安徽大学 一种多取代异羟肟酸衍生物的合成方法
WO2024159287A1 (pt) * 2023-01-30 2024-08-08 Eurofarma Laboratórios S.A. Hidroxamatos bloqueadores de nav 1.7 e/ou nav 1.8, seus processos de obtenção, composições, usos, métodos de tratamento destes e kits
AR131715A1 (es) * 2023-01-30 2025-04-23 Eurofarma Laboratorios S A AMIDAS BLOQUEADORAS DE Nav 1.7 Y/O Nav 1.8, SUS PROCESOS DE OBTENCIÓN, COMPOSICIONES, USOS, MÉTODOS DE TRATAMIENTO DE LOS MISMOS Y KITS

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2279973A (en) * 1940-05-08 1942-04-14 Du Pont Stabilization of organic substances
US2279560A (en) * 1940-05-08 1942-04-14 Du Pont Viscous hydrocarbon oil
CH220744A (de) * 1941-05-09 1942-04-30 Chem Ind Basel Verfahren zur Herstellung eines neuen Acetylderivats der technischen Stearinhydroxamsäure.
US3560519A (en) * 1969-03-28 1971-02-02 Sinclair Research Inc Aromatic mono(nitrile carbonates)
US3900514A (en) * 1971-06-03 1975-08-19 Kerr Mc Gee Chem Corp N-cycloalkyl hydroxamic acids
US3978208A (en) * 1974-01-07 1976-08-31 Eisai Co., Ltd. Deodorizing compositions
US4208205A (en) * 1977-10-03 1980-06-17 E. I. Du Pont De Nemours And Company Herbicidal benzamides
AU1933583A (en) * 1982-09-22 1984-03-29 Meiji Seika K.K. Hydroxylamine derivatives
NL8400852A (nl) * 1983-03-31 1984-10-16 Sandoz Ag Nieuwe anilinen en hun gebruik.
US4528392A (en) * 1984-04-18 1985-07-09 American Home Products Corporation Aromatic compounds as antiallergic agents
US4792560A (en) * 1985-04-03 1988-12-20 Rorer Pharmaceutical Corporation Quinoline hydroxamates and their use as modulators of arachidonic acid metabolic pathways

Also Published As

Publication number Publication date
ES551515A0 (es) 1987-10-16
HUT37742A (en) 1986-02-28
HU200594B (en) 1990-07-28
IL75223A (en) 1988-05-31
ES8609201A1 (es) 1986-09-01
ES551516A0 (es) 1988-05-16
ES551514A0 (es) 1987-04-16
ES8802378A1 (es) 1988-05-16
ES551517A0 (es) 1987-07-01
ES551519A0 (es) 1987-07-01
KR850008660A (ko) 1985-12-21
DK217385A (da) 1985-11-18
ES8704872A1 (es) 1987-04-16
PH21267A (en) 1987-09-28
EP0161939A3 (en) 1986-10-08
ES543192A0 (es) 1986-09-01
ES8706606A1 (es) 1987-07-01
AU586973B2 (en) 1989-08-03
FI851970L (fi) 1985-11-18
DE3587460T2 (de) 1994-02-17
FI851970A0 (fi) 1985-05-17
DK217385D0 (da) 1985-05-15
ES8800129A1 (es) 1987-10-16
EP0161939B1 (en) 1993-07-21
AU4254685A (en) 1985-11-21
NZ212099A (en) 1989-08-29
EP0161939A2 (en) 1985-11-21
FI851970A7 (fi) 1985-11-18
ES8706605A1 (es) 1987-07-01
GR851203B (enExample) 1985-11-25
IL75223A0 (en) 1985-09-29
ES8706604A1 (es) 1987-07-01
US4607053A (en) 1986-08-19
DE3587460D1 (en) 1993-08-26
ES551518A0 (es) 1987-07-01

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