KR880002353B1 - 퀴놀린 화합물 및 그의 제조방법 - Google Patents

퀴놀린 화합물 및 그의 제조방법 Download PDF

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Publication number
KR880002353B1
KR880002353B1 KR1019830001302A KR830001302A KR880002353B1 KR 880002353 B1 KR880002353 B1 KR 880002353B1 KR 1019830001302 A KR1019830001302 A KR 1019830001302A KR 830001302 A KR830001302 A KR 830001302A KR 880002353 B1 KR880002353 B1 KR 880002353B1
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KR
South Korea
Prior art keywords
dihydro
fluoro
oxo
compound
alkylamino
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
KR1019830001302A
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English (en)
Korean (ko)
Other versions
KR840004102A (ko
Inventor
필립 웬트랜드 마아크
마아론 베이리 데니스
Original Assignee
스터어링 드럭그 인코포레이팃드
제이므즈 에이취 루서
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Publication date
Application filed by 스터어링 드럭그 인코포레이팃드, 제이므즈 에이취 루서 filed Critical 스터어링 드럭그 인코포레이팃드
Publication of KR840004102A publication Critical patent/KR840004102A/ko
Application granted granted Critical
Publication of KR880002353B1 publication Critical patent/KR880002353B1/ko
Expired legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/58—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems with hetero atoms directly attached to the ring nitrogen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
KR1019830001302A 1982-03-30 1983-03-30 퀴놀린 화합물 및 그의 제조방법 Expired KR880002353B1 (ko)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US36387682A 1982-03-31 1982-03-31
US363,876 1982-03-31
US446,095 1983-02-14
US06/466,095 US4499091A (en) 1982-03-31 1983-02-14 1-Amino (or substituted amino)-1,4-dihydro-4-oxo-6-fluoro-7-heterylquinoline-3-carboxylic acids and their use as antibacterial agents

Publications (2)

Publication Number Publication Date
KR840004102A KR840004102A (ko) 1984-10-06
KR880002353B1 true KR880002353B1 (ko) 1988-10-29

Family

ID=27002249

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019830001302A Expired KR880002353B1 (ko) 1982-03-30 1983-03-30 퀴놀린 화합물 및 그의 제조방법

Country Status (14)

Country Link
US (1) US4499091A (https=)
KR (1) KR880002353B1 (https=)
AU (1) AU557534B2 (https=)
CA (1) CA1198425A (https=)
DK (1) DK162638C (https=)
ES (1) ES8405390A1 (https=)
FI (1) FI77855C (https=)
GR (1) GR77906B (https=)
IE (1) IE54898B1 (https=)
IL (1) IL68236A (https=)
NO (1) NO158060C (https=)
NZ (1) NZ203621A (https=)
PH (1) PH18392A (https=)
PT (1) PT76456B (https=)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4665079A (en) * 1984-02-17 1987-05-12 Warner-Lambert Company Antibacterial agents
US4730000A (en) * 1984-04-09 1988-03-08 Abbott Laboratories Quinoline antibacterial compounds
DE3409922A1 (de) * 1984-03-17 1985-09-26 Bayer Ag, 5090 Leverkusen 1,7-diamino-1,4-dihydro-4-oxo-3-(aza)chinolincarbonsaeuren, verfahren zu ihrer herstellung sowie ihre verwendung bei der bekaempfung bakterieller erkrankungen
FR2574404B1 (fr) * 1984-12-12 1987-04-24 Provesan Sa Derives 1-substitues de l'acide 6-fluoro-7-(pyrrol-1-yl)-1,4-dihydro-4-oxoquinoleine-3-carboxylique, leur preparation et leur application en tant que medicaments
US4578473A (en) * 1985-04-15 1986-03-25 Warner-Lambert Company Process for quinoline-3-carboxylic acid antibacterial agents
IN166416B (https=) * 1985-09-18 1990-05-05 Pfizer
US4692454A (en) * 1986-02-03 1987-09-08 Warner-Lambert Company Opthalmic use of quinolone antibiotics
DE3606698A1 (de) * 1986-03-01 1987-09-03 Bayer Ag 7-(1-pyrrolidinyl)-chinoloncarbonsaeure -derivate
US5153204A (en) * 1986-03-01 1992-10-06 Bayer Aktiengesellschaft 7-(1-Pyrrolidinyl)-quinolonecarboxylic acid derivatives
JPS62215572A (ja) * 1986-03-17 1987-09-22 Kyorin Pharmaceut Co Ltd キノロンカルボン酸誘導体
IL83049A (en) * 1986-07-04 1991-12-12 Chemie Linz Ag 4-quinolinone-3-carboxylic acid derivatives,their manufacture and pharmaceutical compositions containing them
ES2059335T3 (es) * 1986-09-12 1994-11-16 Hoffmann La Roche Derivados de pirido(3,2,1-ij)-1,3,4-benzoxadiazina, procedimiento para su obtencion, preparados farmaceuticos correspondientes y productos intermedios utilizables en el procedimiento.
US4929613A (en) * 1987-08-26 1990-05-29 Warner-Lambert Company Antibacterial agents
US4868305A (en) * 1988-02-16 1989-09-19 Sterling Drug Inc. Improvement in the preparation of intermediates for quinoline antibacterial agents
US4959363A (en) * 1989-06-23 1990-09-25 Sterling Drug Inc. Quinolonecarboxamide compounds, their preparation and use as antivirals.
US5532239A (en) * 1993-08-02 1996-07-02 Assistance Publique - Hopitaux De Paris Therapeutic application of fluoroquinolone derivatives
DE4416622A1 (de) * 1994-05-11 1995-11-16 Bayer Ag 8-Amino-10-(azabicycloalkyl)-pyrido[1,2,3-d.e] [1,3,4]benzoxa-diazinderivate
US6326391B1 (en) 1998-12-04 2001-12-04 Influx, Inc. Inhibitors of multidrug transporters
US6262072B1 (en) 1999-10-12 2001-07-17 Yung Shin Pharmaceutical Industrial Co. Ltd. Orally administered antimicrobial pharmaceutical formulations of ciprofloxacin
US6957105B2 (en) * 2002-03-26 2005-10-18 Cardiac Pacemakers, Inc. Method and apparatus for detecting oscillations in cardiac rhythm with electrogram signals
US7973022B2 (en) * 2006-02-17 2011-07-05 Idexx Laboratories, Inc. Fluoroquinolone carboxylic acid salt compositions
US20070197548A1 (en) * 2006-02-17 2007-08-23 Murthy Yerramilli V S Fluoroquinolone compositions
US20070196398A1 (en) * 2006-02-17 2007-08-23 Murthy Yerramilli V S Fluoroquinolone fatty acid salt compositions

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS53141286A (en) * 1977-05-16 1978-12-08 Kyorin Seiyaku Kk Novel substituted quinolinecarboxylic acid
CA1175836A (en) * 1977-09-20 1984-10-09 Marcel Pesson Production of 1,4-dihydroquinoline-3-carboxylic acid derivatives
DE2808070A1 (de) * 1978-02-24 1979-08-30 Bayer Ag Verfahren zur herstellung von 4-pyridon-3-carbonsaeuren und/oder deren derivaten

Also Published As

Publication number Publication date
PT76456A (en) 1983-04-01
AU557534B2 (en) 1986-12-24
IL68236A0 (en) 1983-06-15
DK145983D0 (da) 1983-03-30
FI77855C (fi) 1989-05-10
KR840004102A (ko) 1984-10-06
NZ203621A (en) 1986-01-24
NO158060B (no) 1988-03-28
IL68236A (en) 1986-09-30
ES521153A0 (es) 1984-06-01
DK162638B (da) 1991-11-25
PH18392A (en) 1985-06-21
NO158060C (no) 1988-07-06
FI831102L (fi) 1983-10-01
PT76456B (en) 1985-12-10
FI77855B (fi) 1989-01-31
US4499091A (en) 1985-02-12
ES8405390A1 (es) 1984-06-01
IE54898B1 (en) 1990-03-14
NO831056L (no) 1983-10-03
DK145983A (da) 1983-10-01
AU1272283A (en) 1983-10-06
IE830608L (en) 1983-09-30
FI831102A0 (fi) 1983-03-30
GR77906B (https=) 1984-09-25
DK162638C (da) 1992-04-21
CA1198425A (en) 1985-12-24

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