KR870003093A - 퀴놀론카복실산 유도체의 제조방법 - Google Patents

퀴놀론카복실산 유도체의 제조방법 Download PDF

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Publication number
KR870003093A
KR870003093A KR1019860007499A KR860007499A KR870003093A KR 870003093 A KR870003093 A KR 870003093A KR 1019860007499 A KR1019860007499 A KR 1019860007499A KR 860007499 A KR860007499 A KR 860007499A KR 870003093 A KR870003093 A KR 870003093A
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KR
South Korea
Prior art keywords
formula
carboxylic acid
acid derivative
quinolone carboxylic
compound
Prior art date
Application number
KR1019860007499A
Other languages
English (en)
Other versions
KR930003072B1 (ko
Inventor
구니요시 마수자와
세이고 수즈에
게이지 히라이
다가요시 이시자기
Original Assignee
하기하라 히데
교린 세이야꾸 가부시끼 가이샤
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 하기하라 히데, 교린 세이야꾸 가부시끼 가이샤 filed Critical 하기하라 히데
Publication of KR870003093A publication Critical patent/KR870003093A/ko
Application granted granted Critical
Publication of KR930003072B1 publication Critical patent/KR930003072B1/ko

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
    • C07D215/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Quinoline Compounds (AREA)

Abstract

내용 없음

Description

퀴놀론카복실산 유도체의 제조방법
본 내용은 요부공개 건이므로 전문내용을 수록하지 않았음

Claims (1)

  1. 다음 일반식(Ⅱ)의 화합물을 다음 일반식(Ⅲ)의 2급 아민과 축합시켜 다음 일반식(Ⅰ)의 화합물을 제조하고, 필요에 따라 일반식(Ⅰ)의 화합물을 가수분해하여 R1이 저급알킬인 일반식(Ⅰ)의 화합물을 제조하는 방법.
    상기식에서,
    R1은 수소원자 또는 저급알킬 그룹이고,
    R2,R2및 R4는 각각 독립적으로 수소원자 또는 저급알킬그룹이며,
    X는 할로겐원자이다.
    ※ 참고사항 : 최초출원 내용에 의하여 공개하는 것임.
KR1019860007499A 1985-09-10 1986-09-08 퀴놀론카복실산 유도체의 제조방법 KR930003072B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP85-200240 1985-09-10
JP60200240A JPS6259263A (ja) 1985-09-10 1985-09-10 キノロンカルボン酸誘導体
JP200240 1985-09-10

Publications (2)

Publication Number Publication Date
KR870003093A true KR870003093A (ko) 1987-04-15
KR930003072B1 KR930003072B1 (ko) 1993-04-17

Family

ID=16421132

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019860007499A KR930003072B1 (ko) 1985-09-10 1986-09-08 퀴놀론카복실산 유도체의 제조방법

Country Status (9)

Country Link
US (1) US4826982A (ko)
EP (1) EP0216245B1 (ko)
JP (1) JPS6259263A (ko)
KR (1) KR930003072B1 (ko)
CN (1) CN1010313B (ko)
AU (1) AU577712B2 (ko)
CA (1) CA1262135A (ko)
DE (1) DE3672931D1 (ko)
HU (1) HU197893B (ko)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU594983B2 (en) * 1985-10-29 1990-03-22 Dainippon Pharmaceutical Co. Ltd. Novel quinoline derivatives and processes for preparation thereof
DE3719764A1 (de) * 1987-06-13 1988-12-22 Bayer Ag Ionenaustauscherharze beladen mit chinoloncarbonsaeurederivaten, ihre herstellung und verwendung
DE3724466A1 (de) * 1987-07-24 1989-02-02 Bayer Ag Verfahren zur herstellung von chinoloncarbonsaeuren
US8220298B2 (en) 2009-02-17 2012-07-17 Channell Commercial Corporation Self-latching locking assembly

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1598915A (en) * 1977-09-20 1981-09-23 Bellon Labor Sa Roger 1,4-dihydro-quinoline-3-carboxylic acid derivatives process for their preparation and composition containing them
US4665079A (en) * 1984-02-17 1987-05-12 Warner-Lambert Company Antibacterial agents
DE3248505A1 (de) * 1982-12-29 1984-07-05 Bayer Ag, 5090 Leverkusen 1-cyclopropyl-6-fluor-1,4-dihydro-4-oxo-7(4- (oxoalkyl)-1-piperazinyl/-3-chinolincarbonsaeuren und ihre derivate, verfahren zu ihrer herstellung sowie diese enthaltende antibakterielle mittel
DE3318145A1 (de) * 1983-05-18 1984-11-22 Bayer Ag, 5090 Leverkusen 7-amino-1-cyclopropyl-6,8-difluor-1,4-dihydro-4-oxo-3-chinolincarbonsaeuren, verfahren zu ihrer herstellung sowie diese enthaltende antibakterielle mittel
DE3420798A1 (de) * 1984-06-04 1985-12-05 Bayer Ag, 5090 Leverkusen 7-(3-aryl-l-piperazinyl)- sowie 7-(3-cyclohexyl-l-piperazinyl)-3-chinoloncarbonsaeuren
JPS6191183A (ja) * 1984-10-11 1986-05-09 Kyorin Pharmaceut Co Ltd キノロンカルボン酸誘導体

Also Published As

Publication number Publication date
CN1010313B (zh) 1990-11-07
HU197893B (en) 1989-06-28
EP0216245B1 (en) 1990-07-25
KR930003072B1 (ko) 1993-04-17
AU577712B2 (en) 1988-09-29
DE3672931D1 (de) 1990-08-30
AU6240086A (en) 1987-03-12
HUT44026A (en) 1988-01-28
EP0216245A1 (en) 1987-04-01
JPS6259263A (ja) 1987-03-14
CA1262135A (en) 1989-10-03
US4826982A (en) 1989-05-02
CN86106169A (zh) 1987-03-18

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