KR870003072A - 아릴 피리돈의 제조방법 - Google Patents

아릴 피리돈의 제조방법 Download PDF

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KR870003072A
KR870003072A KR1019860007736A KR860007736A KR870003072A KR 870003072 A KR870003072 A KR 870003072A KR 1019860007736 A KR1019860007736 A KR 1019860007736A KR 860007736 A KR860007736 A KR 860007736A KR 870003072 A KR870003072 A KR 870003072A
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pyridone
trifluoromethyl
trifluoromethylphenyl
chloro
compound
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KR900005369B1 (ko
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로버트 퍼리오르 트레보
드라이스달 턴불 미첼
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그라함 도날드 아놀드
임페리알 케미칼 인더스트리스 피엘씨
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Abstract

내용 없음

Description

아릴 피리돈의 제조방법
본 내용은 요부공개 건이므로 전문내용을 수록하지 않았음

Claims (12)

  1. 다음 일반식의 화합물 :
    식중, 각 X 및 Y는 독립적으로 할로겐,
    n는 1-4까지의 정수 ;
    각 Z는 독립적으로 할로겐 및 트리할로메틸로부터 선택된 것, 및
    A는 산소 또는 황,
  2. 제 1 항에 있어서, n이 1 또는 2인 화합물.
  3. 제 1 항에 있어서, 각 X 및 Y는 독립적으로 염소 또는 불소인 화합물.
  4. 제 2 항에 있어서, n이 1 이고 Z가 트리플루오로메틸이거나 n이 2이고 최소한 하나의 Z가 트리플루오로메틸인 화합물.
  5. 전술한 항의 어느 한 항에서, A가 산소인 화합물.
  6. 1-(2,6-디플루오로-4-트리플루오로메틸페닐)-4-트리플루오로메틸-2-피리돈 ;
    1-(2-클로로-6-플루오로-4-트리플루오로페닐)-3-클로로-5-트리플루오로메틸-2-피리돈 ;1-(2-클로로-6-플루오로-4-트리플루오로페닐)-3,5-디브로모-2-피리돈 ;
    1-(2,6-디플루오르-4-트리플루오로메틸페닐-3-클로로-5-트리플루오로메틸-2-피리돈;
    1-(2,6-디플루오로-4-트리플루오로메틸페닐)-5-클로로-2-피리돈 ;
    1-(2,6-디플루오로-4-트리플루오로메틸페닐)-3,5-비스(트리플루오로메틸)-2-피리돈 ;
    1-(2,6-디플루오로-4-플루오로메틸페닐)-5-클로로-4-트리플루오로메틸-2-피리돈 ;
    1-(2,6-디플루오로-4-트리플루오로메틸페닐)-5-브로모-4-트리플루오로메틸-2-피리돈;
    1-(2-클로로-6-플루오로-4-트리플루오로메틸페닐)-4-트리플루오로메틸-2-피리돈 ;
    1-(2-클로로-6-플루오로-4-트리플루오로메틸페닐)-5-트리플루오로메틸-2-피리돈 ;
    1-(2-클로로-6-플루오로-4-트리플루오로메틸페닐)-5-클로로-2-피리돈 ;
    1-(2-클로로-6-플루오로-4-트리플루오로메틸페닐)-3-브로모-5-트리플루오로메틸-2-피리돈 ;
    1-(2-클로로-6-클로로-4--트리플루오로메틸페닐)-3,5-디클로로-2-피리돈 ;
    1-(2-클로로-6-플루오로-4--트리플루오로메틸페닐)-3,5-비스(트리플루오로메틸)-2-피리돈 ;
    1-(2-클로로-6-플루오로-4--트리플루오로메틸페닐)-5-브로모-4-트리플루오로메틸-2-피리돈 ;
    1-(2-클로로-6-플루오로-4--트리플루오로메틸페닐)-4,5-비스(트리플루오로메틸)-2-피리돈 ;
    1-(2-클로로-6-플루오로-4--트리플루오로메틸페닐)-3,5-디클로로-4-트리플루오로메틸-2-피리돈 ;
    1-(2-클로로-6-플루오로-4--트리플루오로메틸페닐)-3,5-디브로모-4-트리플루오로메틸-2-피리돈 ;
    1-(2,6-디클로로-4-트리플루오로메틸페닐)-3-클로로-5-트리플루오로메틸-2-피리돈 ;
    1-(2,6-디클로로-4-트리플루오로메틸페닐)-3,5-비스(트리플루오로메틸)-2-피리돈 ;
    1-(2,6-디클로로-4-트리플루오로메틸페닐)-4-트리플루오로메틸-2-피리돈;
    1-(2,6-디클로로-4-트리플루오로메틸페닐)-4-클로로디플루오로메틸-2-피리돈 ;
    1-(2,6-디클로로-4-트리플루오로메틸페닐)-5-클로로-4-트리플루오로메틸-2-피리돈 ;
    1-(2,6-디클로로-4-트리플루오로메틸페닐)-5-브로모-4-트리플루오로메틸-2-피리돈 ;
    1-(2,6-디클로로-4-트리플루오로메틸페닐)-4,5-비스(트리플루오로메틸)-2-피리돈 ;
    1-(2,6-디클로로-4-트리플루오로메틸페닐)-3,5-디클로로-4-트리플루오로메틸-2-피리돈 ;
    1-(2-브로모-6-클로로-4-트리플루오로메틸페닐)-4-트리플루오로메틸-2-피리돈 ;
    1-(2,6-디브로모-4-트리플루오로메틸페닐)-4-트리플루오로메틸-2-피리돈 ;
    1-(2,6-디플루오로-4-트리플루오로메틸페닐)-5-트리플루오로메틸-2-피리돈 ;
    1-(2,6-디플루오로-4-트리플루오로메틸페닐)-3,5-디클로로-2-피리돈 ;
    1-(2,6-디플루오로-4-트리플루오로메틸페닐)-3-브로모-5-트리플루오로메틸-2-피리돈 ;
    1-(2-클로로-6-플루오로-4-트리플루오로메틸페닐)-5-클로로-4-트리플루오로메틸-2-피리돈 ;
    1-(2,6-디클롤로-4-트리플루오로메틸페닐)-4-트리플루오로메틸-2-피리돈으로부터 선택된 화합물.
  7. 식중 Hal이 할로겐이고 X 및 Y가 제 1 항에서 전술한 바와 같은 일반식(2)의 화합물을
    식중 Z 및 n이 제 1 항에서 전술한 바와 같은 일반식(3)의 화합물과 반응시킨 후 바란다면
    i) n이 1보다 큰 일반식(1)의 화합물을 제조하기 위해 일반식(2)의 화합물을 할로겐화시키는 것; 및
    ii) A가 황인 일반식(1)의 화합물을 제조하기 위해 A가 산소인 일반식(1)의 화합물을 황화제와 반응시키는 것을 하나 이상 행하는 것으로 구성되는, 제 1 항의 일반식(1)의 화합물의 제조방법.
  8. 다음 일반식(3A) 또는 (3B)의 화합물
    식중, Z4및 Z5는 둘다가 수소이지 않게, 독립적으로 수소, 할로겐, 또는 트리플루오로메틸로부터 선택된 것;
    Z10는 트리플루오로메틸과는 다른 트리할로메틸.
  9. 다음 일반식의 화합물.
  10. 식중 W가 아미노, X가 브롬, 및 Y가 염소이거나 W가 불소, X가 브롬 및 Y가 염소 또는 브롬인 다음 일반식의 화합물.
  11. 활성 성분으로서 살충적으로 효과적인 양의 제 1항의 화합물로 구성된 살충조성도.
  12. 살충적으로 효과적인 양의 제11항의 화합물을 해충 또는 해충의 소재지에 사용하는 것으로 구성되는 해충을 박멸하는 방법.
    ※ 참고사항 : 최초출원 내용에 의하여 공개하는 것임.
KR1019860007736A 1985-09-19 1986-09-15 아릴 피리돈의 제조방법 KR900005369B1 (ko)

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GB858523126A GB8523126D0 (en) 1985-09-19 1985-09-19 Aryl pyridones
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TWI412322B (zh) 2005-12-30 2013-10-21 Du Pont 控制無脊椎害蟲之異唑啉
BRPI0809770B8 (pt) 2007-06-13 2022-12-06 Du Pont Composto e composição para controlar uma praga de invertebrados
BRPI0810929B8 (pt) 2007-06-27 2022-12-06 Du Pont uso de um composto de fórmula 1
TWI518076B (zh) 2008-04-09 2016-01-21 杜邦股份有限公司 製備雜環化合物之方法
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KR101478133B1 (ko) * 2009-05-25 2014-12-31 센트럴 사우스 유니버시티 1-（치환된 벤질기）-5-트리플루오로메틸-2-（1ｈ）피리돈 화합물 및 그 염의 제조방법 및 용도

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HU199372B (en) 1990-02-28
ES2001694A6 (es) 1988-06-01
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GR862336B (en) 1986-12-23
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JPS6270362A (ja) 1987-03-31
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