KR830007688A - 비스-테트라졸릴메틸 치환 세팔로스포린 항생물질의 제조방법 - Google Patents

비스-테트라졸릴메틸 치환 세팔로스포린 항생물질의 제조방법 Download PDF

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Publication number
KR830007688A
KR830007688A KR1019810003492A KR810003492A KR830007688A KR 830007688 A KR830007688 A KR 830007688A KR 1019810003492 A KR1019810003492 A KR 1019810003492A KR 810003492 A KR810003492 A KR 810003492A KR 830007688 A KR830007688 A KR 830007688A
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KR
South Korea
Prior art keywords
formula
hydrogen
general formula
compound
group
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
KR1019810003492A
Other languages
English (en)
Korean (ko)
Inventor
사무엘 카르너 알렌
Original Assignee
아더 알. 웨일
일라인 릴리 앤드 캄파니
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 아더 알. 웨일, 일라인 릴리 앤드 캄파니 filed Critical 아더 알. 웨일
Publication of KR830007688A publication Critical patent/KR830007688A/ko
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D257/00—Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms
    • C07D257/02—Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D257/04—Five-membered rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/02—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
    • C07D241/06—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having one or two double bonds between ring members or between ring members and non-ring members
    • C07D241/08—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having one or two double bonds between ring members or between ring members and non-ring members with oxygen atoms directly attached to ring carbon atoms
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
KR1019810003492A 1980-09-17 1981-09-17 비스-테트라졸릴메틸 치환 세팔로스포린 항생물질의 제조방법 Ceased KR830007688A (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US187859 1980-09-17
US06/187,859 US4346076A (en) 1980-09-17 1980-09-17 Bis-tetrazoylmethyl substituted cephalosporin antibiotics

Publications (1)

Publication Number Publication Date
KR830007688A true KR830007688A (ko) 1983-11-04

Family

ID=22690789

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019810003492A Ceased KR830007688A (ko) 1980-09-17 1981-09-17 비스-테트라졸릴메틸 치환 세팔로스포린 항생물질의 제조방법

Country Status (22)

Country Link
US (1) US4346076A (OSRAM)
EP (1) EP0048169A3 (OSRAM)
JP (1) JPS5781492A (OSRAM)
KR (1) KR830007688A (OSRAM)
AU (1) AU7528481A (OSRAM)
CA (1) CA1174668A (OSRAM)
CS (1) CS686781A2 (OSRAM)
DD (1) DD201142A5 (OSRAM)
DK (1) DK412181A (OSRAM)
ES (1) ES8306377A1 (OSRAM)
FI (1) FI812782L (OSRAM)
GB (1) GB2084144B (OSRAM)
GR (1) GR74671B (OSRAM)
HU (1) HU185954B (OSRAM)
IL (1) IL63770A0 (OSRAM)
PH (1) PH16985A (OSRAM)
PL (1) PL132001B1 (OSRAM)
PT (1) PT73680B (OSRAM)
RO (1) RO82970B (OSRAM)
SU (2) SU1087076A3 (OSRAM)
YU (1) YU222681A (OSRAM)
ZA (1) ZA816224B (OSRAM)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR850001206B1 (ko) * 1984-04-27 1985-08-20 한국과학기술원 세펨 유도체의 제조 방법
IT1181672B (it) * 1984-10-25 1987-09-30 Upjohn Co Cefalosporina alogenidrato cristallino
US4868193A (en) * 1986-09-24 1989-09-19 Rorer Pharmaceutical Corporation Styryl tetrazoles and anti-allergic use thereof
EP0333082A3 (en) * 1988-03-15 1991-05-02 Takeda Chemical Industries, Ltd. Cephem compounds, their production and use

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ176206A (en) * 1973-12-25 1978-03-06 Takeda Chemical Industries Ltd Cephalosporins
US4286089A (en) * 1974-12-27 1981-08-25 Smithkline Corporation 7-Acyl-3-(substituted tetrazolyl thiomethyl)cephalosporins
JPS525787A (en) * 1975-06-27 1977-01-17 Bristol Myers Co Antiibacterial agent
US4109085A (en) * 1976-02-17 1978-08-22 Pfizer Inc. 7-amino-3-substituted-cephem compounds
US4113942A (en) * 1976-02-17 1978-09-12 Pfizer Inc. 4-(Tetrazol-5-yl)-Δ3 -cephem compounds
US4278670A (en) * 1976-07-12 1981-07-14 Smithkline Corporation 7-Alpha-oxyiminoacylcephalosporins
US4129732A (en) * 1977-04-27 1978-12-12 Pfizer Inc. 4(Tetrazol-5-yl)-Δ3 -cephem compounds
FR2387235A1 (fr) * 1978-01-23 1978-11-10 Fujisawa Pharmaceutical Co Procede de preparation de composes d'acide 3,7-disubstitue-3-cephem-4-carboxylique et nouveaux produits ainsi obtenus, ayant une forte activite antibacterienne

Also Published As

Publication number Publication date
PL132001B1 (en) 1985-01-31
GB2084144A (en) 1982-04-07
FI812782A7 (fi) 1982-03-18
ZA816224B (en) 1983-04-27
RO82970A (ro) 1984-01-14
SU1087076A3 (ru) 1984-04-15
PT73680A (en) 1981-10-01
ES505550A0 (es) 1983-05-16
HU185954B (en) 1985-04-28
JPS5781492A (en) 1982-05-21
PH16985A (en) 1984-05-04
ES8306377A1 (es) 1983-05-16
DD201142A5 (de) 1983-07-06
FI812782L (fi) 1982-03-18
YU222681A (en) 1983-10-31
RO82970B (ro) 1984-01-30
PT73680B (en) 1982-11-26
GR74671B (OSRAM) 1984-07-02
EP0048169A2 (en) 1982-03-24
DK412181A (da) 1982-04-21
SU1119607A3 (ru) 1984-10-15
PL233058A1 (OSRAM) 1982-10-11
GB2084144B (en) 1985-02-06
CA1174668A (en) 1984-09-18
IL63770A0 (en) 1981-12-31
CS686781A2 (en) 1985-06-13
EP0048169A3 (en) 1983-01-19
AU7528481A (en) 1982-03-25
US4346076A (en) 1982-08-24

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Legal Events

Date Code Title Description
PA0109 Patent application

Patent event code: PA01091R01D

Comment text: Patent Application

Patent event date: 19810917

PG1501 Laying open of application
PE0902 Notice of grounds for rejection

Comment text: Notification of reason for refusal

Patent event date: 19850727

Patent event code: PE09021S01D

PE0601 Decision on rejection of patent

Patent event date: 19851016

Comment text: Decision to Refuse Application

Patent event code: PE06012S01D

Patent event date: 19850727

Comment text: Notification of reason for refusal

Patent event code: PE06011S01I