KR20240152410A - 아티카프란트를 포함하는 조성물 - Google Patents

아티카프란트를 포함하는 조성물 Download PDF

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Publication number
KR20240152410A
KR20240152410A KR1020247033299A KR20247033299A KR20240152410A KR 20240152410 A KR20240152410 A KR 20240152410A KR 1020247033299 A KR1020247033299 A KR 1020247033299A KR 20247033299 A KR20247033299 A KR 20247033299A KR 20240152410 A KR20240152410 A KR 20240152410A
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KR
South Korea
Prior art keywords
articaprant
pharmaceutical composition
treatment
anhedonia
patient
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
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KR1020247033299A
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English (en)
Korean (ko)
Inventor
니콜라스 마사 펠릭스 고이바에르츠
마크 쉬밋
바니나 포포바
아담 제이. 사비츠
라마 멜코트
웨인 씨. 드레베츠
엠디 스리하리 고팔
데럴 펨버톤
차크라다르 라기셰티
아이바 케직
마헤쉬 엔. 삼타니
톰 후이브레히츠
게르트 반 더 아부츠
매티유 래블링겐
로라 마르티네즈 마르코스
타티아나 마르코지
카타리나 요키체비치
Original Assignee
얀센 파마슈티칼즈, 인코포레이티드
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Application filed by 얀센 파마슈티칼즈, 인코포레이티드 filed Critical 얀센 파마슈티칼즈, 인코포레이티드
Publication of KR20240152410A publication Critical patent/KR20240152410A/ko
Pending legal-status Critical Current

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2009—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/2853—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers, poly(lactide-co-glycolide)
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4816—Wall or shell material
    • A61K9/4825—Proteins, e.g. gelatin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841—Filling excipients; Inactive ingredients
    • A61K9/4858—Organic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841—Filling excipients; Inactive ingredients
    • A61K9/4866—Organic macromolecular compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Psychiatry (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pain & Pain Management (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Inorganic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
KR1020247033299A 2022-03-07 2023-03-06 아티카프란트를 포함하는 조성물 Pending KR20240152410A (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202263317471P 2022-03-07 2022-03-07
US63/317,471 2022-03-07
PCT/IB2023/052097 WO2023170554A1 (en) 2022-03-07 2023-03-06 Compositions comprising aticaprant

Publications (1)

Publication Number Publication Date
KR20240152410A true KR20240152410A (ko) 2024-10-21

Family

ID=85980700

Family Applications (1)

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KR1020247033299A Pending KR20240152410A (ko) 2022-03-07 2023-03-06 아티카프란트를 포함하는 조성물

Country Status (16)

Country Link
US (3) US20230277500A1 (https=)
EP (1) EP4489730B1 (https=)
JP (1) JP2025508069A (https=)
KR (1) KR20240152410A (https=)
CN (1) CN119156202A (https=)
AU (1) AU2023231767A1 (https=)
CA (1) CA3254546A1 (https=)
CL (1) CL2024002648A1 (https=)
CO (1) CO2024012454A2 (https=)
ES (1) ES3064226T3 (https=)
IL (1) IL315415A (https=)
JO (1) JOP20240196A1 (https=)
MX (1) MX2024010977A (https=)
TW (1) TW202400135A (https=)
UY (1) UY40173A (https=)
WO (1) WO2023170554A1 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US12161622B2 (en) 2021-05-04 2024-12-10 Janssen Pharmaceuticals, Inc. Compositions and methods for the treatment of depression
CN119156211A (zh) 2022-03-07 2024-12-17 杨森制药公司 用于治疗重性抑郁障碍的多晶型形式的阿替卡普兰
EP4489730B1 (en) 2022-03-07 2026-01-21 Janssen Pharmaceuticals, Inc. Compositions comprising aticaprant

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MX2024010977A (es) 2024-12-06
IL315415A (en) 2024-11-01
US12201610B2 (en) 2025-01-21
US20240269110A1 (en) 2024-08-15
CO2024012454A2 (es) 2024-09-30
ES3064226T3 (en) 2026-04-23
UY40173A (es) 2023-09-29
AU2023231767A1 (en) 2024-10-24
CL2024002648A1 (es) 2025-01-24
TW202400135A (zh) 2024-01-01
US20230277500A1 (en) 2023-09-07
CN119156202A (zh) 2024-12-17
CA3254546A1 (en) 2023-09-14
EP4489730B1 (en) 2026-01-21
WO2023170554A1 (en) 2023-09-14
JP2025508069A (ja) 2025-03-21
JOP20240196A1 (ar) 2024-09-05
EP4489730C0 (en) 2026-01-21
US20250228819A1 (en) 2025-07-17
EP4489730A1 (en) 2025-01-15

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