KR20230002656A - 아미노피리미딘 유도체, 또는 이의 약학적으로 허용 가능한 염, 수화물, 또는 용매화물을 포함하는 경구 투여용 약학 조성물 - Google Patents
아미노피리미딘 유도체, 또는 이의 약학적으로 허용 가능한 염, 수화물, 또는 용매화물을 포함하는 경구 투여용 약학 조성물 Download PDFInfo
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| US63/014,277 | 2020-04-23 | ||
| PCT/IB2021/053035 WO2021209893A1 (en) | 2020-04-14 | 2021-04-13 | Pharmaceutical composition for oral administration comprising amin op yrimidine derivative or pharmaceutically acceptable salt, hydrate, or solvate thereof |
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| PH (1) | PH12022552454A1 (https=) |
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| KR20210061457A (ko) * | 2018-10-18 | 2021-05-27 | 주식회사유한양행 | 아미노피리미딘 유도체 또는 이의 염을 포함하는 경구 투여용 약학 조성물 |
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| WO2022253261A1 (zh) * | 2021-06-01 | 2022-12-08 | 杭州领业医药科技有限公司 | Lazertinib甲磺酸盐的水合物晶型及其制备方法和用途 |
| CN118251220A (zh) * | 2022-01-19 | 2024-06-25 | 江苏奥赛康药业有限公司 | 一种包含嘧啶基团的三并环类化合物的组合物及其制备方法和应用 |
| CA3228195A1 (en) | 2023-05-23 | 2025-06-30 | Janssen Biotech, Inc. | Methods for treatment of non-small cell lung cancer (nsclc) |
| WO2025052273A1 (en) | 2023-09-05 | 2025-03-13 | Janssen Biotech, Inc. | Methods of treating non-small cell lung cancer |
| WO2026042017A1 (en) | 2024-08-19 | 2026-02-26 | Janssen Biotech, Inc. | Amivantamab in combination with lazertinib for the treatment of non-small cell lung cancer (nsclc) |
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| US6437006B1 (en) * | 1999-09-27 | 2002-08-20 | American Cyanamid Company | Pharmaceutical carrier formulation |
| US6399591B1 (en) * | 2000-01-19 | 2002-06-04 | Yung-Shin Pharmaceutical Ind. Co., Ltd. | Chargeable pharmaceutical tablets |
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| EP2198857A1 (en) * | 2008-12-19 | 2010-06-23 | Ratiopharm GmbH | Oral dispersible tablet |
| US9278063B2 (en) * | 2009-12-11 | 2016-03-08 | Sumitomo Dainippon Pharma Co., Ltd. | Press-coated orally-disintegrating tablets |
| JP2013523833A (ja) * | 2010-04-07 | 2013-06-17 | バーテックス ファーマシューティカルズ インコーポレイテッド | ３−（６−（１−（２，２−ジフルオロベンゾ［ｄ］［１，３］ジオキソール−５−イル）シクロプロパンカルボキサミド）−３−メチルピリジン−２−イル）安息香酸の医薬組成物およびその投与 |
| CN113201073A (zh) | 2012-11-21 | 2021-08-03 | 詹森生物科技公司 | 双特异性EGFR/c-Met抗体 |
| WO2015006753A2 (en) * | 2013-07-12 | 2015-01-15 | The Regents Of The University Of California | Therapies for diseases caused by arthropod-borne parasites |
| JP6581088B2 (ja) * | 2013-12-12 | 2019-09-25 | アルミラル・ソシエダッド・アノニマＡｌｍｉｒａｌｌ， Ｓ．Ａ． | フマル酸ジメチルを含む医薬組成物 |
| GB201402070D0 (en) * | 2014-02-07 | 2014-03-26 | Galapagos Nv | Pharmaceutical compositions for the treatment of inflammatory disorders |
| EP3929190B1 (en) | 2014-10-13 | 2024-12-25 | Yuhan Corporation | Compounds and compositions for modulating egfr mutant kinase activities |
| CN109310677A (zh) | 2016-04-07 | 2019-02-05 | 凯莫森特里克斯股份有限公司 | 通过联合施用ccr1拮抗剂与pd-1抑制剂或pd-l1拮抗剂降低肿瘤负荷 |
| KR20230169458A (ko) * | 2017-01-20 | 2023-12-15 | 엑셀리시스, 인코포레이티드 | 암을 치료하기 위한 카보잔티닙 및 아테졸리주맙의 조합 |
| CN110520110A (zh) * | 2017-03-08 | 2019-11-29 | 阿瑞雅德制药公司 | 包含5-氯-n4-[2-(二甲基磷酰基)苯基]-n2-{2-甲氧基-4-[4-(4-甲基哌嗪-1-基)哌啶-1-基]苯基}嘧啶-2,4-二胺的药物制剂 |
| AR111469A1 (es) * | 2017-04-21 | 2019-07-17 | Yuhan Corp | Sal de un compuesto del derivado de aminopiridina, una forma cristalina de la misma, y un proceso para preparar la misma |
| FI3658552T3 (fi) | 2017-07-28 | 2023-11-16 | Yuhan Corp | Menetelmä n-(5-((4-(4-((dimetyyliamino)metyyli)-3-fenyyli-1h-pyratsol-1-yyli)pyrimidin-2-yyli)amino)-4-metoksi-2-morfolinofenyyli)akryyliamidin valmistamiseksi saattamalla vastaava amiini reagoimaan 3-halopropionyylikloridin kanssa |
| EP3658553B1 (en) | 2017-07-28 | 2022-06-15 | Yuhan Corporation | Intermediates useful for the synthesis of aminopyrimidine derivatives, process for preparing the same, and process for preparing aminopyrimidine derivatives using the same |
| ES2959967T3 (es) | 2017-07-28 | 2024-02-29 | Yuhan Corp | Procedimiento de preparación deN-(5-(4-(4-formil-3-fenil-1h-pirazol-1-il)pirimidin-2-ilamino)-4-metoxi-2-morfolinofenil)acrilamida |
| CN110580014B (zh) * | 2018-06-11 | 2021-03-30 | 北京京东尚科信息技术有限公司 | 用于控制自动导引运输车的方法、装置和系统 |
| JP7455807B2 (ja) * | 2018-07-20 | 2024-03-26 | アイメリーズ ユーエスエー，インコーポレーテッド | 鋳造砂廃棄物からの砂、ベントナイト、及び有機物の回収 |
| KR20200043618A (ko) | 2018-10-18 | 2020-04-28 | 주식회사유한양행 | 아미노피리미딘 유도체 또는 이의 염을 포함하는 경구투여용 약학 조성물 |
| CA3136632A1 (en) * | 2019-04-11 | 2020-10-15 | Goldfinch Bio, Inc. | Spray-dried formulation of a pyridazinone trpc5 inhibitor |
| FI3920891T3 (fi) * | 2019-04-17 | 2024-03-19 | Nordiccan As | Nopeasti hajoavat kannabinoiditabletit |
| US11850248B2 (en) | 2019-05-14 | 2023-12-26 | Yuhan Corporation | Therapies with 3rd generation EGFR tyrosine kinase inhibitors |
| AU2020319662B2 (en) * | 2019-07-31 | 2024-02-29 | F. Hoffmann-La Roche Ag | New pharmaceutical formulation |
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| Publication number | Priority date | Publication date | Assignee | Title |
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| KR20210061457A (ko) * | 2018-10-18 | 2021-05-27 | 주식회사유한양행 | 아미노피리미딘 유도체 또는 이의 염을 포함하는 경구 투여용 약학 조성물 |
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| JP2023522634A (ja) | 2023-05-31 |
| AU2021257662A1 (en) | 2022-12-15 |
| US20210322323A1 (en) | 2021-10-21 |
| BR112022020609A2 (pt) | 2022-11-29 |
| IL297240A (en) | 2022-12-01 |
| PH12022552454A1 (en) | 2024-02-05 |
| JP7787824B2 (ja) | 2025-12-17 |
| TW202207940A (zh) | 2022-03-01 |
| JP2025179094A (ja) | 2025-12-09 |
| US20250177311A1 (en) | 2025-06-05 |
| CA3180184A1 (en) | 2021-10-21 |
| WO2021209893A1 (en) | 2021-10-21 |
| WO2021209893A8 (en) | 2022-10-13 |
| UY39171A (es) | 2021-10-29 |
| AU2021257662B2 (en) | 2025-06-12 |
| CN115484937A (zh) | 2022-12-16 |
| AU2025203347A1 (en) | 2025-05-29 |
| US12138351B2 (en) | 2024-11-12 |
| MX2022012898A (es) | 2023-01-24 |
| EP4135669A1 (en) | 2023-02-22 |
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