KR20220156981A - Ｓ１ｐ 조절제 즉시 방출 투여 요법 - Google Patents
Ｓ１ｐ 조절제 즉시 방출 투여 요법 Download PDFInfo
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- KR20220156981A KR20220156981A KR1020227039781A KR20227039781A KR20220156981A KR 20220156981 A KR20220156981 A KR 20220156981A KR 1020227039781 A KR1020227039781 A KR 1020227039781A KR 20227039781 A KR20227039781 A KR 20227039781A KR 20220156981 A KR20220156981 A KR 20220156981A
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/397—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having four-membered rings, e.g. azetidine
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- A61K9/2013—Organic compounds, e.g. phospholipids, fats
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- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P25/00—Drugs for disorders of the nervous system
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- A—HUMAN NECESSITIES
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- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
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| PCT/IB2015/052550 WO2015155709A1 (en) | 2014-04-10 | 2015-04-08 | S1p modulator immediate release dosage regimen |
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| KR20220156981A true KR20220156981A (ko) | 2022-11-28 |
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| KR1020167031062A Ceased KR20160141841A (ko) | 2014-04-10 | 2015-04-08 | Ｓ１ｐ 조절제 즉시 방출 투여 요법 |
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| JP6674903B2 (ja) * | 2014-04-10 | 2020-04-01 | ノバルティス アーゲー | Ｓ１ｐ調節剤即時放出投与レジメン |
| US11434200B2 (en) | 2017-03-09 | 2022-09-06 | Novartis Ag | Solid forms comprising an oxime ether compound and a coformer, compositions and methods of use thereof |
| US11629124B2 (en) | 2017-03-09 | 2023-04-18 | Novartis Ag | Solid forms comprising an oxime ether compound, compositions and methods of use thereof |
| MX2020007326A (es) * | 2017-09-29 | 2020-09-07 | Novartis Ag | Regimen de dosificacion de siponimod. |
| EP3687530A1 (en) * | 2017-09-29 | 2020-08-05 | Novartis AG | Dosing regimen of siponimod |
| PL3758708T3 (pl) | 2018-03-01 | 2025-03-31 | Astrazeneca Ab | Kompozycje farmaceutyczne zawierające (2s)-{(1s)-1-cyjano-2-[4-(3-metylo-2-okso-2,3-dihydro-1,3-benzoksazol-5-ilo)fenylo]etylo}-1,4-oksazepano-2-karboksyamid |
| EP3823627A4 (en) | 2018-07-17 | 2022-04-20 | Insmed Incorporated | CERTAIN (2S)-N-[(1S)-1-CYANO-2-PHENYLETHYL]-1,4-OXAZEPANE-2-CARBOXAMIDES FOR THE TREATMENT OF LUPUS ENEHROPATHY |
| CN109908095A (zh) * | 2019-04-08 | 2019-06-21 | 肇庆学院 | 一种西尼莫德片剂及制备方法 |
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| US11135197B2 (en) | 2020-02-07 | 2021-10-05 | Argentum Pharmaceuticals Llc | Dosage regimen of an S1P receptor modulator |
| EP4646265A1 (en) | 2023-01-06 | 2025-11-12 | Insmed Incorporated | Novel, reversible dpp1 inhibitors and uses thereof |
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| PL2676953T3 (pl) * | 2008-12-18 | 2017-09-29 | Novartis Ag | Sól hemifumaranowa kwasu 1-[4-[1-(4-cykloheksylo-3-trifluorometylobenzyloksyimino)-etylo]-2-etylobenzylo]-azetydyno-3-karboksylowego |
| SI3409274T1 (sl) * | 2008-12-22 | 2020-03-31 | Novartis Ag | Režim odmerjanja za S1P receptor agonist |
| BRPI0923213A2 (pt) | 2008-12-22 | 2016-01-26 | Novaris Ag | regime de dosagem de um agonista do receptor para s1p. |
| AU2010101513B4 (en) * | 2009-09-29 | 2016-05-05 | Novartis Ag | Dosage regimen of an S1P receptor modulator |
| UA114283C2 (uk) * | 2011-01-07 | 2017-05-25 | Новартіс Аг | Композиції імуносупресантів |
| WO2012095853A1 (en) | 2011-01-10 | 2012-07-19 | Novartis Pharma Ag | Modified release formulations comprising sip receptor modulators |
| WO2013057212A1 (en) * | 2011-10-21 | 2013-04-25 | Novartis Ag | Dosage regimen for an s1p receptor modulator or agonist |
| JP6674903B2 (ja) * | 2014-04-10 | 2020-04-01 | ノバルティス アーゲー | Ｓ１ｐ調節剤即時放出投与レジメン |
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2018
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2020
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2024
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| US20190054065A1 (en) | 2019-02-21 |
| CA2943598C (en) | 2023-03-07 |
| AU2020203107B2 (en) | 2021-10-21 |
| US20220016076A1 (en) | 2022-01-20 |
| CA2943598A1 (en) | 2015-10-15 |
| KR20160141841A (ko) | 2016-12-09 |
| CN116650467A (zh) | 2023-08-29 |
| CN106456552A (zh) | 2017-02-22 |
| EP3831378A1 (en) | 2021-06-09 |
| RU2016143979A (ru) | 2018-05-14 |
| IL305337A (en) | 2023-10-01 |
| IL247986A0 (en) | 2016-11-30 |
| RU2016143979A3 (enExample) | 2018-11-12 |
| JP6674903B2 (ja) | 2020-04-01 |
| PH12016501965A1 (en) | 2017-01-09 |
| RU2020107732A (ru) | 2020-03-30 |
| EP3129020A1 (en) | 2017-02-15 |
| AU2015246036A1 (en) | 2016-10-13 |
| US20250041266A1 (en) | 2025-02-06 |
| ZA201606519B (en) | 2017-11-29 |
| MX2016013245A (es) | 2017-01-16 |
| AU2020203107A1 (en) | 2020-05-28 |
| SG11201607894RA (en) | 2016-10-28 |
| WO2015155709A1 (en) | 2015-10-15 |
| US20170027907A1 (en) | 2017-02-02 |
| CL2016002562A1 (es) | 2017-07-28 |
| EP4074312A1 (en) | 2022-10-19 |
| RU2715734C2 (ru) | 2020-03-03 |
| TW201622721A (zh) | 2016-07-01 |
| JP2017510607A (ja) | 2017-04-13 |
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