CL2016002562A1 - Régimen de dosificación de liberación inmediata de moduladores s1p. - Google Patents

Régimen de dosificación de liberación inmediata de moduladores s1p.

Info

Publication number
CL2016002562A1
CL2016002562A1 CL2016002562A CL2016002562A CL2016002562A1 CL 2016002562 A1 CL2016002562 A1 CL 2016002562A1 CL 2016002562 A CL2016002562 A CL 2016002562A CL 2016002562 A CL2016002562 A CL 2016002562A CL 2016002562 A1 CL2016002562 A1 CL 2016002562A1
Authority
CL
Chile
Prior art keywords
modulators
immediate release
dosing regime
regime
dosing
Prior art date
Application number
CL2016002562A
Other languages
English (en)
Inventor
Eric Legangneux
Philippe Michel Rene Bouillot
Emeric Reynaud
Erik Walstroem
Frank Dahlke
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=52988364&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CL2016002562(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of CL2016002562A1 publication Critical patent/CL2016002562A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/397Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having four-membered rings, e.g. azetidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • A61K9/2018Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/2027Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurology (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Immunology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
CL2016002562A 2014-04-10 2016-10-07 Régimen de dosificación de liberación inmediata de moduladores s1p. CL2016002562A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201461977816P 2014-04-10 2014-04-10

Publications (1)

Publication Number Publication Date
CL2016002562A1 true CL2016002562A1 (es) 2017-07-28

Family

ID=52988364

Family Applications (1)

Application Number Title Priority Date Filing Date
CL2016002562A CL2016002562A1 (es) 2014-04-10 2016-10-07 Régimen de dosificación de liberación inmediata de moduladores s1p.

Country Status (16)

Country Link
US (3) US20170027907A1 (es)
EP (3) EP4074312A1 (es)
JP (1) JP6674903B2 (es)
KR (2) KR20160141841A (es)
CN (2) CN106456552A (es)
AU (2) AU2015246036A1 (es)
CA (1) CA2943598C (es)
CL (1) CL2016002562A1 (es)
IL (2) IL305337A (es)
MX (1) MX2016013245A (es)
PH (1) PH12016501965A1 (es)
RU (2) RU2020107732A (es)
SG (1) SG11201607894RA (es)
TW (1) TW201622721A (es)
WO (1) WO2015155709A1 (es)
ZA (1) ZA201606519B (es)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP4074312A1 (en) * 2014-04-10 2022-10-19 Novartis AG Siponimod immediate release dosage regimen for treating autoimmune diseases
US11629124B2 (en) 2017-03-09 2023-04-18 Novartis Ag Solid forms comprising an oxime ether compound, compositions and methods of use thereof
RU2020114750A (ru) * 2017-09-29 2021-10-29 Новартис Аг Схема введения доз сипонимода
CN111132677A (zh) * 2017-09-29 2020-05-08 诺华股份有限公司 西尼莫德的给药方案
EP3758708A1 (en) * 2018-03-01 2021-01-06 AstraZeneca AB Pharmaceutical compositions comprising (2s)--{(1s)-1-cyano-2-[4-(3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-5-yl)phenyl]ethyl}-1,4-oxazepane-2-carboxamide
CN109908095A (zh) * 2019-04-08 2019-06-21 肇庆学院 一种西尼莫德片剂及制备方法
CA3156298A1 (en) 2019-10-31 2021-05-06 Laetitia POUZOL Combination of a cxcr7 antagonist with an s1p1 receptor modulator
WO2021158838A1 (en) * 2020-02-07 2021-08-12 Argentum Pharmaceuticals Llc Dosage regimen of an s1p receptor modulator

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20170062554A (ko) * 2008-12-18 2017-06-07 노파르티스 아게 1-[4-[1-(4-시클로헥실-3-트리플루오로메틸-벤질옥시이미노)-에틸]-2-에틸-벤질]-아제티딘-3-카르복실산의 헤미푸마레이트 염
PL2379069T3 (pl) * 2008-12-22 2015-08-31 Novartis Ag Schemat dawkowania agonisty receptora S1P
SI3409274T1 (sl) * 2008-12-22 2020-03-31 Novartis Ag Režim odmerjanja za S1P receptor agonist
CA3129729A1 (en) * 2009-09-29 2011-04-07 Novartis Ag Dosage regimen of an s1p receptor modulator
PT2661261T (pt) * 2011-01-07 2019-10-25 Novartis Ag Formulações imunossupressoras.
WO2012095853A1 (en) 2011-01-10 2012-07-19 Novartis Pharma Ag Modified release formulations comprising sip receptor modulators
JP2014530835A (ja) * 2011-10-21 2014-11-20 ノバルティスアーゲー S1p受容体モジュレーターまたはs1p受容体アゴニストのための投薬量レジメン
EP4074312A1 (en) * 2014-04-10 2022-10-19 Novartis AG Siponimod immediate release dosage regimen for treating autoimmune diseases

Also Published As

Publication number Publication date
TW201622721A (zh) 2016-07-01
SG11201607894RA (en) 2016-10-28
JP2017510607A (ja) 2017-04-13
CA2943598C (en) 2023-03-07
PH12016501965A1 (en) 2017-01-09
EP4074312A1 (en) 2022-10-19
CA2943598A1 (en) 2015-10-15
EP3831378A1 (en) 2021-06-09
JP6674903B2 (ja) 2020-04-01
RU2715734C2 (ru) 2020-03-03
US20170027907A1 (en) 2017-02-02
ZA201606519B (en) 2017-11-29
CN116650467A (zh) 2023-08-29
EP3129020A1 (en) 2017-02-15
KR20220156981A (ko) 2022-11-28
RU2020107732A (ru) 2020-03-30
IL247986A0 (en) 2016-11-30
US20220016076A1 (en) 2022-01-20
RU2016143979A3 (es) 2018-11-12
CN106456552A (zh) 2017-02-22
WO2015155709A1 (en) 2015-10-15
KR20160141841A (ko) 2016-12-09
US20190054065A1 (en) 2019-02-21
MX2016013245A (es) 2017-01-16
RU2016143979A (ru) 2018-05-14
IL305337A (en) 2023-10-01
AU2020203107A1 (en) 2020-05-28
AU2020203107B2 (en) 2021-10-21
AU2015246036A1 (en) 2016-10-13

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