KR20220119169A - Pgi2-수용체 효능제를 포함하는 조성물 및 그의 제조 방법 - Google Patents

Pgi2-수용체 효능제를 포함하는 조성물 및 그의 제조 방법 Download PDF

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KR20220119169A
KR20220119169A KR1020227027530A KR20227027530A KR20220119169A KR 20220119169 A KR20220119169 A KR 20220119169A KR 1020227027530 A KR1020227027530 A KR 1020227027530A KR 20227027530 A KR20227027530 A KR 20227027530A KR 20220119169 A KR20220119169 A KR 20220119169A
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compound
excipient
pharmaceutical composition
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제지 제쓰 샤오
라이자 베라니아 플로리다
칭-유안 리
리 알라니 셀베이
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아레나 파마슈티칼스, 인크.
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    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/27—Esters, e.g. nitroglycerine, selenocyanates of carbamic or thiocarbamic acids, meprobamate, carbachol, neostigmine
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    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1617—Organic compounds, e.g. phospholipids, fats
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    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1617—Organic compounds, e.g. phospholipids, fats
    • A61K9/1623—Sugars or sugar alcohols, e.g. lactose; Derivatives thereof; Homeopathic globules
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    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
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    • A61K9/1629—Organic macromolecular compounds
    • A61K9/1652—Polysaccharides, e.g. alginate, cellulose derivatives; Cyclodextrin
    • A—HUMAN NECESSITIES
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    • A—HUMAN NECESSITIES
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    • A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
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    • A61K9/2022—Organic macromolecular compounds
    • A61K9/2031—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers
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    • A61K9/2833—Organic macromolecular compounds
    • A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
    • A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
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    • A61K9/4816—Wall or shell material
    • A61K9/4825—Proteins, e.g. gelatin
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    • A61K9/4841—Filling excipients; Inactive ingredients
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    • A61K9/4841—Filling excipients; Inactive ingredients
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  • Inorganic Chemistry (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pulmonology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
KR1020227027530A 2017-03-01 2018-03-01 Pgi2-수용체 효능제를 포함하는 조성물 및 그의 제조 방법 Ceased KR20220119169A (ko)

Applications Claiming Priority (10)

Application Number Priority Date Filing Date Title
US201762465675P 2017-03-01 2017-03-01
US62/465,675 2017-03-01
US201762468832P 2017-03-08 2017-03-08
US62/468,832 2017-03-08
US201762526039P 2017-06-28 2017-06-28
US62/526,039 2017-06-28
US201762530515P 2017-07-10 2017-07-10
US62/530,515 2017-07-10
PCT/US2018/020519 WO2018160882A1 (en) 2017-03-01 2018-03-01 Compositions comprising pgi2-receptor agonists and processes for the preparation thereof
KR1020197028214A KR102432505B1 (ko) 2017-03-01 2018-03-01 Pgi2-수용체 효능제를 포함하는 조성물 및 그의 제조 방법

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KR1020197028214A Division KR102432505B1 (ko) 2017-03-01 2018-03-01 Pgi2-수용체 효능제를 포함하는 조성물 및 그의 제조 방법

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KR1020197028214A Active KR102432505B1 (ko) 2017-03-01 2018-03-01 Pgi2-수용체 효능제를 포함하는 조성물 및 그의 제조 방법

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US (3) US11123298B2 (enExample)
EP (2) EP3977985B1 (enExample)
JP (2) JP7023559B2 (enExample)
KR (2) KR20220119169A (enExample)
CN (1) CN110582271B (enExample)
AU (2) AU2018227842B2 (enExample)
CA (1) CA3054835A1 (enExample)
ES (2) ES2897024T3 (enExample)
IL (1) IL268997B2 (enExample)
MA (1) MA47686A (enExample)
WO (1) WO2018160882A1 (enExample)

Cited By (1)

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WO2025009945A1 (ko) * 2023-07-06 2025-01-09 재단법인대구경북과학기술원 셀렉시팍을 포함하는 퇴행성 뇌질환의 예방 또는 치료용 약학 조성물

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JP2022070923A (ja) 2022-05-13
CA3054835A1 (en) 2018-09-07
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US11826471B2 (en) 2023-11-28
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IL268997B2 (en) 2023-09-01
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US20190240159A1 (en) 2019-08-08
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US11123298B2 (en) 2021-09-21
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