KR20200058506A - 면역조정제 - Google Patents

면역조정제 Download PDF

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Publication number
KR20200058506A
KR20200058506A KR1020207012116A KR20207012116A KR20200058506A KR 20200058506 A KR20200058506 A KR 20200058506A KR 1020207012116 A KR1020207012116 A KR 1020207012116A KR 20207012116 A KR20207012116 A KR 20207012116A KR 20200058506 A KR20200058506 A KR 20200058506A
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KR
South Korea
Prior art keywords
dmf
resin
fmoc
solution
frit
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
KR1020207012116A
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English (en)
Korean (ko)
Inventor
마이클 매튜 밀러
마틴 패트릭 앨런
링 리
Original Assignee
브리스톨-마이어스 스큅 컴퍼니
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Application filed by 브리스톨-마이어스 스큅 컴퍼니 filed Critical 브리스톨-마이어스 스큅 컴퍼니
Publication of KR20200058506A publication Critical patent/KR20200058506A/ko
Pending legal-status Critical Current

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/50—Cyclic peptides containing at least one abnormal peptide link
    • C07K7/54—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring
    • C07K7/56—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring the cyclisation not occurring through 2,4-diamino-butanoic acid
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04—Linear peptides containing only normal peptide links
    • C07K7/08—Linear peptides containing only normal peptide links having 12 to 20 amino acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/10—Peptides having 12 to 20 amino acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Epidemiology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
KR1020207012116A 2017-10-03 2018-10-02 면역조정제 Pending KR20200058506A (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201762567323P 2017-10-03 2017-10-03
US62/567,323 2017-10-03
PCT/US2018/053871 WO2019070643A1 (en) 2017-10-03 2018-10-02 IMMUNOMODULATORS

Publications (1)

Publication Number Publication Date
KR20200058506A true KR20200058506A (ko) 2020-05-27

Family

ID=63998773

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1020207012116A Pending KR20200058506A (ko) 2017-10-03 2018-10-02 면역조정제

Country Status (6)

Country Link
US (1) US11492375B2 (enExample)
EP (1) EP3692053A1 (enExample)
JP (1) JP7257393B2 (enExample)
KR (1) KR20200058506A (enExample)
CN (1) CN111051332B (enExample)
WO (1) WO2019070643A1 (enExample)

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Also Published As

Publication number Publication date
CN111051332B (zh) 2024-09-06
EP3692053A1 (en) 2020-08-12
US11492375B2 (en) 2022-11-08
CN111051332A (zh) 2020-04-21
US20200291069A1 (en) 2020-09-17
JP2020536091A (ja) 2020-12-10
WO2019070643A1 (en) 2019-04-11
JP7257393B2 (ja) 2023-04-13

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