KR20170125951A - 화학요법에 의해 유도되는 통증의 예방 또는 치료를 위한 시그마 리간드 - Google Patents
화학요법에 의해 유도되는 통증의 예방 또는 치료를 위한 시그마 리간드 Download PDFInfo
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- KR20170125951A KR20170125951A KR1020177028558A KR20177028558A KR20170125951A KR 20170125951 A KR20170125951 A KR 20170125951A KR 1020177028558 A KR1020177028558 A KR 1020177028558A KR 20177028558 A KR20177028558 A KR 20177028558A KR 20170125951 A KR20170125951 A KR 20170125951A
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- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
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- A—HUMAN NECESSITIES
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- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
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| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP09382144.5 | 2009-08-14 | ||
| EP09382144A EP2292236A1 (en) | 2009-08-14 | 2009-08-14 | Sigma ligands for the prevention or treatment of pain induced by chemotherapy |
| PCT/EP2010/061720 WO2011018487A1 (en) | 2009-08-14 | 2010-08-12 | Sigma ligands for the prevention or treatment of pain induced by chemotherapy |
Related Parent Applications (1)
| Application Number | Title | Priority Date | Filing Date |
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| KR1020157034281A Division KR20150140419A (ko) | 2009-08-14 | 2010-08-12 | 화학요법에 의해 유도되는 통증의 예방 또는 치료를 위한 시그마 리간드 |
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| KR20170125951A true KR20170125951A (ko) | 2017-11-15 |
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| KR1020157034281A Ceased KR20150140419A (ko) | 2009-08-14 | 2010-08-12 | 화학요법에 의해 유도되는 통증의 예방 또는 치료를 위한 시그마 리간드 |
| KR1020127006715A Expired - Fee Related KR101605151B1 (ko) | 2009-08-14 | 2010-08-12 | 화학요법에 의해 유도되는 통증의 예방 또는 치료를 위한 시그마 리간드 |
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| Application Number | Title | Priority Date | Filing Date |
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| KR1020157034281A Ceased KR20150140419A (ko) | 2009-08-14 | 2010-08-12 | 화학요법에 의해 유도되는 통증의 예방 또는 치료를 위한 시그마 리간드 |
| KR1020127006715A Expired - Fee Related KR101605151B1 (ko) | 2009-08-14 | 2010-08-12 | 화학요법에 의해 유도되는 통증의 예방 또는 치료를 위한 시그마 리간드 |
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Families Citing this family (14)
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| EP2116539A1 (en) | 2008-04-25 | 2009-11-11 | Laboratorios Del. Dr. Esteve, S.A. | 1-aryl-3-aminoalkoxy-pyrazoles as sigma ligands enhancing analgesic effects of opioids and attenuating the dependency thereof |
| EP2353598A1 (en) | 2010-02-04 | 2011-08-10 | Laboratorios Del. Dr. Esteve, S.A. | Sigma ligands for use in the prevention and/or treatment of postoperative pain |
| EP2353591A1 (en) | 2010-02-04 | 2011-08-10 | Laboratorios Del. Dr. Esteve, S.A. | Sigma ligands for potentiating the analgesic effect of opioids and opiates in post-operative pain and attenuating the dependency thereof |
| EP2388005A1 (en) * | 2010-05-21 | 2011-11-23 | Laboratorios Del. Dr. Esteve, S.A. | Sigma ligands for the prevention and/or treatment of emesis induced by chemotherapy or radiotherapy |
| EP2415471A1 (en) | 2010-08-03 | 2012-02-08 | Laboratorios Del. Dr. Esteve, S.A. | Use of sigma ligands in opioid-induced hyperalgesia |
| EP2426111A1 (en) * | 2010-08-09 | 2012-03-07 | Laboratorios Del. Dr. Esteve, S.A. | 4-[-2-[[5-methyl-1-(2-naphtalenyl)-1h-pyrazol-3-yl]oxy]ethyl]morpholine hydrochloride amorphous solid forms |
| EP2524694A1 (en) * | 2011-05-19 | 2012-11-21 | Laboratorios Del. Dr. Esteve, S.A. | Use of sigma ligands in diabetes type-2 associated pain |
| EP2792352A1 (en) | 2013-04-16 | 2014-10-22 | Laboratorios Del. Dr. Esteve, S.A. | Alpha-2 adrenoreceptor and sigma receptor ligand combinations |
| EP3043795A1 (en) * | 2013-09-12 | 2016-07-20 | Laboratorios Del. Dr. Esteve, S.A. | Nsaid and sigma receptor ligand combinations |
| JP2017503765A (ja) | 2013-12-17 | 2017-02-02 | ラボラトリオス・デル・ドクトル・エステベ・ソシエダッド・アノニマ | ガバペンチノイドおよびシグマ受容体の組み合わせ |
| AU2014364647A1 (en) | 2013-12-17 | 2016-06-23 | Laboratorios Del Dr. Esteve, S.A. | Serotonin-Norepinephrine Reuptake Inhibitors (SNRIs) and Sigma receptor ligands combinations |
| EP3463339B1 (en) * | 2016-06-06 | 2023-12-06 | Esteve Pharmaceuticals, S.A. | Use of sigma receptor ligands in cancer |
| CA3121202A1 (en) | 2018-11-30 | 2020-06-04 | Nuvation Bio Inc. | Pyrrole and pyrazole compounds and methods of use thereof |
| WO2024105225A1 (en) * | 2022-11-18 | 2024-05-23 | Universitat De Barcelona | Synergistic combinations of a sigma receptor 1 (s1r) antagonist and a soluble epoxide hydrolase inhibitor (sehi) and their use in the treatment of pain |
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| Publication number | Priority date | Publication date | Assignee | Title |
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| SU11248A1 (ru) | 1927-03-29 | 1929-09-30 | В.С. Григорьев | Способ очистки антрацена |
| FR2301250A1 (fr) * | 1975-02-21 | 1976-09-17 | Bellon Labor Sa Roger | Nouveaux diaryl-1, 4o-aminoalcoxy-3 pyrazoles et leurs sels |
| PL1781618T3 (pl) * | 2004-08-27 | 2013-03-29 | Esteve Labor Dr | Inhibitory receptora sigma |
| DK1781618T3 (da) * | 2004-08-27 | 2012-10-29 | Esteve Labor Dr | Sigma-receptorinhibitorer |
| EP1634872A1 (en) * | 2004-08-27 | 2006-03-15 | Laboratorios Del Dr. Esteve, S.A. | Pyrazole derivatives as sigma receptor inhibitors |
| CN101395157A (zh) * | 2006-03-01 | 2009-03-25 | 伊斯特芬博士实验室有限公司 | 作为西格玛受体抑制剂的吡唑衍生物 |
| MX2008011016A (es) * | 2006-03-01 | 2008-09-08 | Esteve Labor Dr | Inhibidores de receptor sigma. |
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