KR20170103960A - Pet 영상화제 - Google Patents
Pet 영상화제 Download PDFInfo
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- KR20170103960A KR20170103960A KR1020177022757A KR20177022757A KR20170103960A KR 20170103960 A KR20170103960 A KR 20170103960A KR 1020177022757 A KR1020177022757 A KR 1020177022757A KR 20177022757 A KR20177022757 A KR 20177022757A KR 20170103960 A KR20170103960 A KR 20170103960A
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- South Korea
- Prior art keywords
- methyl
- compound
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- alkyl
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Classifications
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-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/05—Isotopically modified compounds, e.g. labelled
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- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Medicinal Chemistry (AREA)
- Physics & Mathematics (AREA)
- Optics & Photonics (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Medical Informatics (AREA)
- Engineering & Computer Science (AREA)
- Surgery (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pathology (AREA)
- Radiology & Medical Imaging (AREA)
- Biomedical Technology (AREA)
- Heart & Thoracic Surgery (AREA)
- Molecular Biology (AREA)
- Biophysics (AREA)
- High Energy & Nuclear Physics (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Enzymes And Modification Thereof (AREA)
- Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
- Nuclear Medicine (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Applications Claiming Priority (3)
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| US201562105336P | 2015-01-20 | 2015-01-20 | |
| US62/105,336 | 2015-01-20 | ||
| PCT/IB2016/050276 WO2016116875A1 (en) | 2015-01-20 | 2016-01-20 | Pet imaging agents |
Publications (1)
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| KR20170103960A true KR20170103960A (ko) | 2017-09-13 |
Family
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| KR1020177022757A Withdrawn KR20170103960A (ko) | 2015-01-20 | 2016-01-20 | Pet 영상화제 |
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| EP (1) | EP3247706B1 (enExample) |
| JP (2) | JP6723264B2 (enExample) |
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| CN (1) | CN107406419B (enExample) |
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| MX (1) | MX2017009452A (enExample) |
| WO (1) | WO2016116875A1 (enExample) |
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| CA2974311A1 (en) | 2015-01-20 | 2016-07-28 | Novartis Ag | Pet imaging agents |
| TWI809597B (zh) * | 2020-12-16 | 2023-07-21 | 美商美國禮來大藥廠 | 預靶向造影劑 |
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| GB0224917D0 (en) * | 2002-10-25 | 2002-12-04 | Novartis Ag | Organic compounds |
| WO2005043300A2 (en) | 2003-10-20 | 2005-05-12 | Empirix, Inc. | Computer language interpretation and optimization for server testing |
| BRPI0510512A (pt) | 2004-04-28 | 2007-10-30 | Icos Corp | derivados de arilfenilamino, arilfenilamida e sulfeto de arilfeniléter |
| WO2005121094A1 (en) | 2004-06-09 | 2005-12-22 | Pfizer Limited | Piperazine and piperidine derivatives as anti-hiv-agents |
| CN101429161A (zh) * | 2008-12-05 | 2009-05-13 | 常熟理工学院 | Pet显像剂前体异喹啉甲酰胺衍生物的合成方法 |
| JP5767205B2 (ja) * | 2009-04-02 | 2015-08-19 | メルク パテント ゲゼルシャフト ミット ベシュレンクテル ハフツングＭｅｒｃｋ Ｐａｔｅｎｔ Ｇｅｓｅｌｌｓｃｈａｆｔ ｍｉｔ ｂｅｓｃｈｒａｅｎｋｔｅｒ Ｈａｆｔｕｎｇ | オートタキシン阻害剤としての複素環式化合物 |
| US8999974B2 (en) | 2010-08-09 | 2015-04-07 | Raqualia Pharma Inc. | Acyl piperazine derivatives as TTX-S blockers |
| JP2013536200A (ja) * | 2010-08-20 | 2013-09-19 | アミラ ファーマシューティカルス，インコーポレーテッド | オートタキシン阻害剤およびその使用 |
| PT2861566T (pt) * | 2012-06-13 | 2017-02-08 | Hoffmann La Roche | Novos diazaspirocicloalcanos e azaspirocicloalcanos |
| CN104968656B (zh) * | 2012-12-19 | 2017-08-11 | 诺华股份有限公司 | 自分泌运动因子抑制剂 |
| SG11201600241RA (en) | 2013-07-18 | 2016-02-26 | Novartis Ag | Autotaxin inhibitors comprising a heteroaromatic ring-benzyl-amide-cycle core |
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2016
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- 2016-01-20 JP JP2017555866A patent/JP6723264B2/ja not_active Expired - Fee Related
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2019
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2020
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| CN107406419A (zh) | 2017-11-28 |
| US20200017474A1 (en) | 2020-01-16 |
| US20180273509A1 (en) | 2018-09-27 |
| EA201791643A1 (ru) | 2017-11-30 |
| EP3247706A1 (en) | 2017-11-29 |
| MX2017009452A (es) | 2017-11-08 |
| US10450298B2 (en) | 2019-10-22 |
| AU2016209906A1 (en) | 2017-08-03 |
| EP3247706B1 (en) | 2020-07-08 |
| ES2828715T3 (es) | 2021-05-27 |
| CA2974311A1 (en) | 2016-07-28 |
| BR112017015455A2 (pt) | 2018-01-23 |
| JP6723264B2 (ja) | 2020-07-15 |
| US10865195B2 (en) | 2020-12-15 |
| CN107406419B (zh) | 2020-09-11 |
| CN107406419A8 (zh) | 2018-01-12 |
| JP2018511648A (ja) | 2018-04-26 |
| JP2020158532A (ja) | 2020-10-01 |
| WO2016116875A1 (en) | 2016-07-28 |
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