KR20160145833A - 티에노트리아졸로디아제핀 화합물을 사용한 급성 골수성 백혈병 및/또는 급성 림프아구성 백혈병의 치료 방법 - Google Patents

티에노트리아졸로디아제핀 화합물을 사용한 급성 골수성 백혈병 및/또는 급성 림프아구성 백혈병의 치료 방법 Download PDF

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KR20160145833A
KR20160145833A KR1020167033946A KR20167033946A KR20160145833A KR 20160145833 A KR20160145833 A KR 20160145833A KR 1020167033946 A KR1020167033946 A KR 1020167033946A KR 20167033946 A KR20167033946 A KR 20167033946A KR 20160145833 A KR20160145833 A KR 20160145833A
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compound
leukemia
formula
solid dispersion
acute
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케이 노엘
마리아 이 리베이로
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온코에틱스 게엠베하
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
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    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A61K31/167—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the nitrogen of a carboxamide group directly attached to the aromatic ring, e.g. lidocaine, paracetamol
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    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
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    • A61K31/4045—Indole-alkylamines; Amides thereof, e.g. serotonin, melatonin
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    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
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    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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KR1020167033946A 2014-05-02 2015-05-01 티에노트리아졸로디아제핀 화합물을 사용한 급성 골수성 백혈병 및/또는 급성 림프아구성 백혈병의 치료 방법 Withdrawn KR20160145833A (ko)

Applications Claiming Priority (15)

Application Number Priority Date Filing Date Title
US201461987822P 2014-05-02 2014-05-02
US61/987,822 2014-05-02
US201461990465P 2014-05-08 2014-05-08
US61/990,465 2014-05-08
US201462012135P 2014-06-13 2014-06-13
US201462012128P 2014-06-13 2014-06-13
US62/012,128 2014-06-13
US62/012,135 2014-06-13
US201462080804P 2014-11-17 2014-11-17
US201462080771P 2014-11-17 2014-11-17
US62/080,804 2014-11-17
US62/080,771 2014-11-17
US201462086456P 2014-12-02 2014-12-02
US62/086,456 2014-12-02
PCT/US2015/028891 WO2015168621A1 (en) 2014-05-02 2015-05-01 Method of treating acute myeloid leukemia and/or acute lymphoblastic leukemia using thienotriazolodiazepine compounds

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KR20160145833A true KR20160145833A (ko) 2016-12-20

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KR1020167033946A Withdrawn KR20160145833A (ko) 2014-05-02 2015-05-01 티에노트리아졸로디아제핀 화합물을 사용한 급성 골수성 백혈병 및/또는 급성 림프아구성 백혈병의 치료 방법

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US (1) US9956228B2 (cg-RX-API-DMAC7.html)
EP (1) EP3137085A4 (cg-RX-API-DMAC7.html)
JP (1) JP2017514909A (cg-RX-API-DMAC7.html)
KR (1) KR20160145833A (cg-RX-API-DMAC7.html)
CN (1) CN107073014A (cg-RX-API-DMAC7.html)
AU (1) AU2015252844A1 (cg-RX-API-DMAC7.html)
CA (1) CA2947601A1 (cg-RX-API-DMAC7.html)
MX (1) MX2016014301A (cg-RX-API-DMAC7.html)
RU (1) RU2016146099A (cg-RX-API-DMAC7.html)
WO (1) WO2015168621A1 (cg-RX-API-DMAC7.html)

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US20170049784A1 (en) 2017-02-23
AU2015252844A1 (en) 2016-11-03
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