KR20160095035A - 알파-이소형 선택성 포스파티딜이노시톨 3-키나제 억제제를 위한 투여 요법 - Google Patents

알파-이소형 선택성 포스파티딜이노시톨 3-키나제 억제제를 위한 투여 요법 Download PDF

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KR20160095035A
KR20160095035A KR1020167017707A KR20167017707A KR20160095035A KR 20160095035 A KR20160095035 A KR 20160095035A KR 1020167017707 A KR1020167017707 A KR 1020167017707A KR 20167017707 A KR20167017707 A KR 20167017707A KR 20160095035 A KR20160095035 A KR 20160095035A
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compound
pharmaceutically acceptable
acceptable salt
administered
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엠마누엘 디 토마소
마리-캐롤린 게르마
크리스티안 마사세시
크리스틴 프리치
크리스티안 렌 슈넬
란자나 타보라스
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노파르티스 아게
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Application filed by 노파르티스 아게 filed Critical 노파르티스 아게
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/427—Thiazoles not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
KR1020167017707A 2013-12-06 2014-12-03 알파-이소형 선택성 포스파티딜이노시톨 3-키나제 억제제를 위한 투여 요법 Ceased KR20160095035A (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP13306679.5 2013-12-06
EP13306679 2013-12-06
PCT/IB2014/066558 WO2015083101A1 (en) 2013-12-06 2014-12-03 Dosage regimen for an alpha-isoform selective phosphatidylinositol 3-kinase inhibitor

Publications (1)

Publication Number Publication Date
KR20160095035A true KR20160095035A (ko) 2016-08-10

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ID=49876516

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KR1020167017707A Ceased KR20160095035A (ko) 2013-12-06 2014-12-03 알파-이소형 선택성 포스파티딜이노시톨 3-키나제 억제제를 위한 투여 요법

Country Status (22)

Country Link
US (4) US20170000778A1 (https=)
EP (2) EP4000619A1 (https=)
JP (1) JP2016539149A (https=)
KR (1) KR20160095035A (https=)
CN (1) CN105979947A (https=)
AU (2) AU2014358773A1 (https=)
BR (1) BR112016011811A2 (https=)
CA (1) CA2930359C (https=)
CL (1) CL2016001361A1 (https=)
DK (1) DK3076969T3 (https=)
ES (1) ES2899167T3 (https=)
HU (1) HUE057092T2 (https=)
IL (1) IL245709B (https=)
MX (1) MX378409B (https=)
PH (1) PH12016501026A1 (https=)
PL (1) PL3076969T3 (https=)
PT (1) PT3076969T (https=)
RU (1) RU2680246C1 (https=)
SI (1) SI3076969T1 (https=)
TN (1) TN2016000179A1 (https=)
TW (1) TWI666019B (https=)
WO (1) WO2015083101A1 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20180280370A1 (en) * 2015-11-02 2018-10-04 Novartis Ag Dosage regimen for a phosphatidylinositol 3-kinase inhibitor
WO2018060833A1 (en) * 2016-09-27 2018-04-05 Novartis Ag Dosage regimen for alpha-isoform selective phosphatidylinositol 3-kinase inhibitor alpelisib
GB202010627D0 (en) * 2020-07-10 2020-08-26 Qbd (Qs-Ip) Ltd Blocking method

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Also Published As

Publication number Publication date
CA2930359C (en) 2022-03-01
JP2016539149A (ja) 2016-12-15
CL2016001361A1 (es) 2017-02-10
AU2017245292A1 (en) 2017-11-02
AU2014358773A1 (en) 2016-06-02
US20210196696A1 (en) 2021-07-01
EP3076969B1 (en) 2021-09-01
CA2930359A1 (en) 2015-06-11
HUE057092T2 (hu) 2022-04-28
BR112016011811A2 (pt) 2017-08-08
SI3076969T1 (sl) 2021-12-31
US20200069670A1 (en) 2020-03-05
HK1223549A1 (zh) 2017-08-04
AU2017245292B2 (en) 2018-09-27
US10434092B2 (en) 2019-10-08
DK3076969T3 (da) 2021-11-22
CN105979947A (zh) 2016-09-28
EP3076969A1 (en) 2016-10-12
PL3076969T3 (pl) 2022-01-17
IL245709A0 (en) 2016-07-31
PT3076969T (pt) 2021-11-23
MX2016007376A (es) 2017-05-11
TN2016000179A1 (en) 2017-10-06
TWI666019B (zh) 2019-07-21
IL245709B (en) 2021-03-25
US20170000778A1 (en) 2017-01-05
US20180078540A1 (en) 2018-03-22
TW201609096A (zh) 2016-03-16
EP4000619A1 (en) 2022-05-25
MX378409B (es) 2025-03-10
PH12016501026A1 (en) 2016-07-04
RU2680246C1 (ru) 2019-02-19
WO2015083101A1 (en) 2015-06-11
ES2899167T3 (es) 2022-03-10

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