KR20150116907A - 옥사디아졸 유도체, 및 대사성 글루타메이트 수용체 강화제로서의 그의 용도 - 842 - Google Patents
옥사디아졸 유도체, 및 대사성 글루타메이트 수용체 강화제로서의 그의 용도 - 842 Download PDFInfo
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- KR20150116907A KR20150116907A KR1020157026785A KR20157026785A KR20150116907A KR 20150116907 A KR20150116907 A KR 20150116907A KR 1020157026785 A KR1020157026785 A KR 1020157026785A KR 20157026785 A KR20157026785 A KR 20157026785A KR 20150116907 A KR20150116907 A KR 20150116907A
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US94255307P | 2007-06-07 | 2007-06-07 | |
| US60/942,553 | 2007-06-07 | ||
| PCT/SE2008/050666 WO2008150233A1 (en) | 2007-06-07 | 2008-06-05 | Oxadiazole derivatives and their use as metabotropic glutamate receptor potentiators - 842 |
Related Parent Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1020097025404A Division KR20100017640A (ko) | 2007-06-07 | 2008-06-05 | 옥사디아졸 유도체, 및 대사성 글루타메이트 수용체 강화제로서의 그의 용도 - 842 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| KR20150116907A true KR20150116907A (ko) | 2015-10-16 |
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Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1020157026785A Ceased KR20150116907A (ko) | 2007-06-07 | 2008-06-05 | 옥사디아졸 유도체, 및 대사성 글루타메이트 수용체 강화제로서의 그의 용도 - 842 |
| KR1020097025404A Ceased KR20100017640A (ko) | 2007-06-07 | 2008-06-05 | 옥사디아졸 유도체, 및 대사성 글루타메이트 수용체 강화제로서의 그의 용도 - 842 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1020097025404A Ceased KR20100017640A (ko) | 2007-06-07 | 2008-06-05 | 옥사디아졸 유도체, 및 대사성 글루타메이트 수용체 강화제로서의 그의 용도 - 842 |
Country Status (33)
| Country | Link |
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| US (2) | US8377940B2 (OSRAM) |
| EP (2) | EP2167502B3 (OSRAM) |
| JP (2) | JP5416696B2 (OSRAM) |
| KR (2) | KR20150116907A (OSRAM) |
| CN (2) | CN101679403B (OSRAM) |
| AR (1) | AR066882A1 (OSRAM) |
| AU (1) | AU2008260717B2 (OSRAM) |
| BR (1) | BRPI0812889A2 (OSRAM) |
| CA (1) | CA2690856C (OSRAM) |
| CL (1) | CL2008001667A1 (OSRAM) |
| CO (1) | CO6251287A2 (OSRAM) |
| CY (2) | CY1113422T1 (OSRAM) |
| DK (2) | DK2444399T3 (OSRAM) |
| EC (1) | ECSP109856A (OSRAM) |
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| HR (2) | HRP20120909T4 (OSRAM) |
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| NZ (1) | NZ582445A (OSRAM) |
| PE (1) | PE20090328A1 (OSRAM) |
| PL (2) | PL2444399T3 (OSRAM) |
| PT (2) | PT2167502E (OSRAM) |
| RS (2) | RS53845B1 (OSRAM) |
| RU (2) | RU2470931C2 (OSRAM) |
| SA (1) | SA08290344B1 (OSRAM) |
| SI (2) | SI2444399T1 (OSRAM) |
| TW (1) | TWI417100B (OSRAM) |
| UA (1) | UA99129C2 (OSRAM) |
| UY (1) | UY31124A1 (OSRAM) |
| WO (1) | WO2008150233A1 (OSRAM) |
| ZA (1) | ZA200908285B (OSRAM) |
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| US7868008B2 (en) * | 2005-08-12 | 2011-01-11 | Astrazeneca Ab | Substituted isoindolones and their use as metabotropic glutamate receptor potentiators |
| US7807706B2 (en) * | 2005-08-12 | 2010-10-05 | Astrazeneca Ab | Metabotropic glutamate-receptor-potentiating isoindolones |
| TW200804281A (en) * | 2006-02-16 | 2008-01-16 | Astrazeneca Ab | New metabotropic glutamate receptor-potentiating isoindolones |
| TWI417095B (zh) | 2006-03-15 | 2013-12-01 | Janssen Pharmaceuticals Inc | １，４-二取代之３-氰基-吡啶酮衍生物及其作為ｍＧｌｕＲ２-受體之正向異位性調節劑之用途 |
| TW200900065A (en) | 2007-03-07 | 2009-01-01 | Janssen Pharmaceutica Nv | 3-cyano-4-(4-pyridinyloxy-phenyl)-pyridin-2-one derivatives |
| TW200845978A (en) | 2007-03-07 | 2008-12-01 | Janssen Pharmaceutica Nv | 3-cyano-4-(4-tetrahydropyran-phenyl)-pyridin-2-one derivatives |
| TWI417100B (zh) * | 2007-06-07 | 2013-12-01 | Astrazeneca Ab | 二唑衍生物及其作為代謝型麩胺酸受體增效劑-８４２之用途 |
| TW200911255A (en) | 2007-06-07 | 2009-03-16 | Astrazeneca Ab | Metabotropic glutamate receptor oxadiazole ligands and their use as potentiators-841 |
| TWI475995B (zh) | 2007-09-14 | 2015-03-11 | Janssen Pharmaceuticals Inc | １’，３’－二取代－４－苯基－３，４，５，６－四氫－２ｈ，１’ｈ－〔１，４’〕聯吡啶基－２’－酮化物 |
| ATE516272T1 (de) | 2007-09-14 | 2011-07-15 | Ortho Mcneil Janssen Pharm | 1,3-disubstituierte 4-(aryl-x-phenyl)-1h-pyridin- 2-one |
| JP5433579B2 (ja) | 2007-09-14 | 2014-03-05 | ジャンセン ファーマシューティカルズ， インコーポレイテッド． | １，３−二置換−４−フェニル−１ｈ−ピリジン−２−オン |
| AU2008323287B2 (en) * | 2007-11-14 | 2011-07-14 | Addex Pharma S.A. | Imidazo[1,2-a]pyridine derivatives and their use as positive allosteric modulators of mGluR2 receptors |
| SA109300358B1 (ar) * | 2008-06-06 | 2012-11-03 | استرازينيكا ايه بي | مقويات مستقبل جلوتامات ذي انتحاء أيضي من أيزو إندولون |
| EP2307389B1 (en) | 2008-06-20 | 2013-01-23 | AstraZeneca AB | Dibenzothiazepine derivative and use thereof |
| EP2344470B1 (en) | 2008-09-02 | 2013-11-06 | Janssen Pharmaceuticals, Inc. | 3-azabicyclo[3.1.0]hexyl derivatives as modulators of metabotropic glutamate receptors |
| RU2517181C2 (ru) | 2008-10-16 | 2014-05-27 | Орто-Макнейл-Янссен Фармасьютикалз, Инк. | Производные индола и бензоморфолина в качестве модулятора метаботропных глутаматных рецепторов |
| US8691813B2 (en) | 2008-11-28 | 2014-04-08 | Janssen Pharmaceuticals, Inc. | Indole and benzoxazine derivatives as modulators of metabotropic glutamate receptors |
| CN102439015B (zh) | 2009-05-12 | 2015-05-13 | 杨森制药有限公司 | 1,2,4-三唑并[4,3-a]吡啶衍生物和其作为mGluR2受体的正向变构调节剂的用途 |
| ES2440001T3 (es) | 2009-05-12 | 2014-01-27 | Janssen Pharmaceuticals, Inc. | Derivados de 1,2,4-triazolo[4,3-A]piridina y su uso para el tratamiento o prevención de trastornos neurológicos y psiquiátricos |
| MY153913A (en) | 2009-05-12 | 2015-04-15 | Janssen Pharmaceuticals Inc | 7-aryl-1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive allosteric modulators of mglur2 receptors |
| RU2012134329A (ru) * | 2010-01-07 | 2014-02-20 | Астразенека Аб | Способ получения позитивного аллостерического модулятора метаботропных глутаматных рецепторов-874 |
| JP2013525427A (ja) * | 2010-04-30 | 2013-06-20 | アストラゼネカ・アクチエボラーグ | 代謝調節型グルタミン酸受容体ポジティブアロステリックモジュレーターの多形 |
| WO2012062751A1 (en) | 2010-11-08 | 2012-05-18 | Janssen Pharmaceuticals, Inc. | 1,2,4-TRIAZOLO[4,3-a]PYRIDINE DERIVATIVES AND THEIR USE AS POSITIVE ALLOSTERIC MODULATORS OF MGLUR2 RECEPTORS |
| CN103298810B (zh) | 2010-11-08 | 2016-03-16 | 杨森制药公司 | 1,2,4-三唑并[4,3-a]吡啶衍生物及其作为MGLUR2受体的正变构调节剂的用途 |
| US8993591B2 (en) | 2010-11-08 | 2015-03-31 | Janssen Pharmaceuticals, Inc. | 1,2,4-triazolo[4,3-a] pyridine derivatives and their use as positive allosteric modulators of MGLUR2 receptors |
| CN102180872B (zh) * | 2011-04-01 | 2014-04-02 | 华中科技大学 | [1,3,4]噁二唑类衍生物及其应用 |
| JO3368B1 (ar) | 2013-06-04 | 2019-03-13 | Janssen Pharmaceutica Nv | مركبات 6، 7- ثاني هيدرو بيرازولو [5،1-a] بيرازين- 4 (5 يد)- اون واستخدامها بصفة منظمات تفارغية سلبية لمستقبلات ميجلور 2 |
| JO3367B1 (ar) | 2013-09-06 | 2019-03-13 | Janssen Pharmaceutica Nv | مركبات 2،1، 4- ثلاثي زولو [3،4-a] بيريدين واستخدامها بصفة منظمات تفارغية موجبة لمستقبلات ميجلور 2 |
| PH12019500127B1 (en) | 2014-01-21 | 2022-05-04 | Janssen Pharmaceutica Nv | Combinations comprising positive allosteric modulators or orthosteric agonists of metabotropic glutamatergic receptor subtype 2 and their use |
| EP3424535A1 (en) | 2014-01-21 | 2019-01-09 | Janssen Pharmaceutica NV | Combinations comprising positive allosteric modulators or orthosteric agonists of metabotropic glutamatergic receptor subtype 2 and their use |
| JP6671456B2 (ja) | 2015-07-17 | 2020-03-25 | 武田薬品工業株式会社 | 複素環化合物 |
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| GB2621323A (en) * | 2022-08-03 | 2024-02-14 | Sirgartan Holdings Ltd | Treatments for obsessive compulsive disorder |
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| US7807706B2 (en) * | 2005-08-12 | 2010-10-05 | Astrazeneca Ab | Metabotropic glutamate-receptor-potentiating isoindolones |
| US7868008B2 (en) * | 2005-08-12 | 2011-01-11 | Astrazeneca Ab | Substituted isoindolones and their use as metabotropic glutamate receptor potentiators |
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| TW200911255A (en) * | 2007-06-07 | 2009-03-16 | Astrazeneca Ab | Metabotropic glutamate receptor oxadiazole ligands and their use as potentiators-841 |
| TWI417100B (zh) * | 2007-06-07 | 2013-12-01 | Astrazeneca Ab | 二唑衍生物及其作為代謝型麩胺酸受體增效劑-８４２之用途 |
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2008
- 2008-06-04 TW TW097120762A patent/TWI417100B/zh not_active IP Right Cessation
- 2008-06-05 DK DK11195016T patent/DK2444399T3/en active
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- 2008-06-05 HR HRP20120909AT patent/HRP20120909T4/hr unknown
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- 2008-06-05 AR ARP080102401A patent/AR066882A1/es unknown
- 2008-06-05 US US12/663,371 patent/US8377940B2/en not_active Expired - Fee Related
- 2008-06-05 ES ES11195016.8T patent/ES2531443T3/es active Active
- 2008-06-05 CN CN2008800191548A patent/CN101679403B/zh not_active Expired - Fee Related
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- 2008-06-05 PL PL11195016T patent/PL2444399T3/pl unknown
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- 2008-06-05 UA UAA200911794A patent/UA99129C2/ru unknown
- 2008-06-05 WO PCT/SE2008/050666 patent/WO2008150233A1/en not_active Ceased
- 2008-06-05 PT PT08779348T patent/PT2167502E/pt unknown
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- 2008-06-05 PT PT11195016T patent/PT2444399E/pt unknown
- 2008-06-05 EP EP11195016.8A patent/EP2444399B1/en active Active
- 2008-06-05 SI SI200830807T patent/SI2167502T1/sl unknown
- 2008-06-05 MY MYPI20095187A patent/MY158066A/en unknown
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- 2008-06-05 RU RU2009147708/04A patent/RU2470931C2/ru not_active IP Right Cessation
- 2008-06-05 ME MEP-2012-131A patent/ME01488B/me unknown
- 2008-06-05 DK DK08779348.5T patent/DK2167502T3/da active
- 2008-06-05 KR KR1020097025404A patent/KR20100017640A/ko not_active Ceased
- 2008-06-06 US US12/134,553 patent/US8377939B2/en not_active Expired - Fee Related
- 2008-06-06 UY UY31124A patent/UY31124A1/es not_active Application Discontinuation
- 2008-06-06 PE PE2008000965A patent/PE20090328A1/es not_active Application Discontinuation
- 2008-06-06 CL CL2008001667A patent/CL2008001667A1/es unknown
- 2008-06-07 SA SA08290344A patent/SA08290344B1/ar unknown
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2009
- 2009-11-16 IL IL202158A patent/IL202158A/en not_active IP Right Cessation
- 2009-11-23 ZA ZA200908285A patent/ZA200908285B/xx unknown
- 2009-12-04 CO CO09139153A patent/CO6251287A2/es not_active Application Discontinuation
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2010
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2012
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2013
- 2013-11-14 JP JP2013235538A patent/JP5815644B2/ja not_active Expired - Fee Related
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2015
- 2015-02-24 HR HRP20150210TT patent/HRP20150210T1/hr unknown
- 2015-02-26 CY CY20151100204T patent/CY1116150T1/el unknown
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