KR20150039748A - Gip 수용체 활성을 나타내는 글루카곤의 유사체들 - Google Patents
Gip 수용체 활성을 나타내는 글루카곤의 유사체들 Download PDFInfo
- Publication number
- KR20150039748A KR20150039748A KR20157001447A KR20157001447A KR20150039748A KR 20150039748 A KR20150039748 A KR 20150039748A KR 20157001447 A KR20157001447 A KR 20157001447A KR 20157001447 A KR20157001447 A KR 20157001447A KR 20150039748 A KR20150039748 A KR 20150039748A
- Authority
- KR
- South Korea
- Prior art keywords
- amino acid
- glucagon
- peptide
- seq
- ala
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
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Images
Classifications
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- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/575—Hormones
- C07K14/605—Glucagons
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- A61K38/22—Hormones
- A61K38/26—Glucagons
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones
- A61P5/50—Drugs for disorders of the endocrine system of the pancreatic hormones for increasing or potentiating the activity of insulin
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/12—Antidiuretics, e.g. drugs for diabetes insipidus
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Diabetes (AREA)
- Endocrinology (AREA)
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- Pharmacology & Pharmacy (AREA)
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- Public Health (AREA)
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- Zoology (AREA)
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- Gastroenterology & Hepatology (AREA)
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- General Chemical & Material Sciences (AREA)
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- Immunology (AREA)
- Emergency Medicine (AREA)
- Child & Adolescent Psychology (AREA)
- Peptides Or Proteins (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Measurement And Recording Of Electrical Phenomena And Electrical Characteristics Of The Living Body (AREA)
- Measuring Pulse, Heart Rate, Blood Pressure Or Blood Flow (AREA)
Applications Claiming Priority (5)
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|---|---|---|---|
| US201261662874P | 2012-06-21 | 2012-06-21 | |
| US61/662,874 | 2012-06-21 | ||
| US201361787973P | 2013-03-15 | 2013-03-15 | |
| US61/787,973 | 2013-03-15 | ||
| PCT/US2013/046229 WO2013192130A1 (en) | 2012-06-21 | 2013-06-18 | Analogs of glucagon exhibiting gip receptor activity |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| KR20150039748A true KR20150039748A (ko) | 2015-04-13 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR20157001447A Abandoned KR20150039748A (ko) | 2012-06-21 | 2013-06-18 | Gip 수용체 활성을 나타내는 글루카곤의 유사체들 |
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| AR (1) | AR091478A1 (OSRAM) |
| AU (1) | AU2013277372B2 (OSRAM) |
| BR (1) | BR112014031671A2 (OSRAM) |
| CA (1) | CA2877127A1 (OSRAM) |
| CL (1) | CL2014003421A1 (OSRAM) |
| CO (1) | CO7170125A2 (OSRAM) |
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| HR (1) | HRP20180936T1 (OSRAM) |
| HU (1) | HUE039267T2 (OSRAM) |
| IL (1) | IL236386B (OSRAM) |
| MX (1) | MX356000B (OSRAM) |
| MY (1) | MY185217A (OSRAM) |
| PE (1) | PE20150863A1 (OSRAM) |
| PH (1) | PH12014502857A1 (OSRAM) |
| PL (1) | PL2864350T3 (OSRAM) |
| PT (1) | PT2864350T (OSRAM) |
| RS (1) | RS57347B1 (OSRAM) |
| SG (1) | SG11201408491SA (OSRAM) |
| SI (1) | SI2864350T1 (OSRAM) |
| TR (1) | TR201808818T4 (OSRAM) |
| TW (1) | TWI644920B (OSRAM) |
| WO (1) | WO2013192130A1 (OSRAM) |
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| BR112014026643B1 (pt) | 2012-04-26 | 2023-03-07 | Universite De Montreal | Derivados de imidazotiadiazol e imidazopirazina como inibidores de receptor 4 ativado por protease (par4) para o tratamento de agregação de plaqueta, seus usos e composição farmacêutica |
| PL2864350T3 (pl) * | 2012-06-21 | 2019-01-31 | Indiana University Research And Technology Corporation | Analogi glukagonu wykazujące aktywność wobec receptora GIP |
| UA116217C2 (uk) | 2012-10-09 | 2018-02-26 | Санофі | Пептидна сполука як подвійний агоніст рецепторів glp1-1 та глюкагону |
| SG10201705097PA (en) | 2012-12-21 | 2017-07-28 | Sanofi Sa | Functionalized exendin-4 derivatives |
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